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N-methyl-6-oxo-4-[(1E)-1-phenylprop-1-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridine-3-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-6-methyl-4-oxo-1,4-dihydropyridine-3-carboxamide
N'-(3-ethylphenyl)-N-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]butanediamide
7-cyclopropanecarbonyl-N-methyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-benzyl-N-(2-methyl-2H-1,2,3-triazol-4-yl)piperidin-4-amine
N-[(2-ethyl-4-methyl-1,3-thiazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
5-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
N-{3-[(4aS,8aR)-1-(2-methylpropyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-3-oxopropyl}methanesulfonamide
1-(butane-1-sulfonyl)-4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine
4-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(2-fluorophenyl)methyl]piperidine
N-[3-(4-fluorophenyl)-3-(furan-2-yl)propyl]-3-(2-{[4-(methylsulfanyl)phenyl]methyl}-5-oxopyrrolidin-2-yl)propanamide
9-[(4-methoxy-2,3-dimethylphenyl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]piperidin-4-yl}methyl)-3-methylbut-2-enamide
2-[(4-methoxyphenyl)methyl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,3-benzoxazole-6-carboxamide
(3aR,6aS)-1-oxo-5-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(3,4-dimethoxyphenyl)-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
4-(3-methoxypyrazin-2-yl)-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
5-(2-{[(dimethyl-1,3-thiazol-5-yl)methyl]amino}pyrimidin-4-yl)-2-ethoxybenzoic acid
2-{1-[(2-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yl)ethyl]acetamide
(1R,9aR)-1-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
1'-(5-propyl-1,2-oxazole-3-carbonyl)-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
2-[3-(morpholin-4-ylmethyl)phenyl]benzamide
9-{[2-(morpholin-4-yl)quinolin-3-yl]methyl}-6-oxa-9-azaspiro[4.5]decane
N-[1-(3-fluoro-4-hydroxyphenyl)ethyl]-2,3-dimethylquinoxaline-6-carboxamide
1-ethyl-2-[1-(1-methylpiperidin-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-1,3-benzodiazole
{4-[(3-methoxyphenyl)methyl]-1-(1-methyl-1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl}methanol
[3-(azepan-1-yl)propyl](methyl)[(4-methyl-1H-imidazol-5-yl)methyl]amine
4-chloro-5-{[7-(cyclobutylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
N-{1-[5-methyl-1-(pyridin-2-yl)-1H-pyrazol-4-yl]ethyl}-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
1-(3-fluorophenyl)-3-(1-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
2-[(dimethylamino)methyl]-N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-1,3-thiazole-4-carboxamide
3-(furan-2-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
3-hydroxy-1-methyl-3-({[(2-phenylphenyl)methyl]amino}methyl)piperidin-2-one
2-{3-cyclopropyl-5-[2-(3,4-difluorophenyl)ethyl]-1H-1,2,4-triazol-1-yl}-4-methylpyridine
(4aR,6R,8aS)-8a-(methoxymethyl)-2-(6-methoxypyrimidin-4-yl)-6-(morpholin-4-yl)-decahydroisoquinoline
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(isoquinoline-5-carbonyl)pyrrolidin-3-yl]methanol
2-[2-(pyrrolidin-1-yl)ethyl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}acetamide
2-hydroxy-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}benzoic acid
6-amino-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]pyridine-3-carboxamide
N-[1-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-(3-methoxy-1,5-dimethyl-1H-pyrazol-4-yl)-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carboxamide
methyl 4-(5-{[3-(3-phenylpropanoyl)piperidin-1-yl]methyl}-1,2,4-oxadiazol-3-yl)benzoate
6-methyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}pyridazin-3-amine
1-[(8-chloroquinolin-2-yl)methyl]-2-methyl-1,4-diazepan-5-one
4-[(3-fluorophenyl)methyl]-1-[3-(thiophen-2-yl)propanoyl]-1,4-diazepan-5-one
2-[methyl(4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}phenyl)amino]ethan-1-ol
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide