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4-methyl-N-{[7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-oxazole-5-carboxamide
({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl){[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}amine
5-[(2-fluoro-5-methoxyphenyl)methyl]-5-(3-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-3-oxopropyl)pyrrolidin-2-one
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(4-methylpiperazine-1-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
ethyl 1-(1-{[2-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carbonyl)piperidine-3-carboxylate
[(2-ethylpyrimidin-5-yl)methyl][(2-phenoxypyridin-3-yl)methyl]amine
1-[1-(3-ethyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]-3-(pyrrolidine-1-carbonyl)piperidine
4-[1-(4-chlorophenyl)-1H-1,2,4-triazol-5-yl]-N,N-dimethylpiperidine-1-carboxamide
1-(3,6-dimethyl-1-benzofuran-2-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-{4-[(3-phenylpiperidin-1-yl)methyl]phenyl}acetamide
1-[2-(1,3-benzothiazol-2-yl)pyrrolidin-1-yl]-3-(3-chloro-1,2-oxazol-5-yl)propan-1-one
[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl](phenyl)methanol
4-{1-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydrophthalazin-1-one
2-methyl-5-(3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine-1-carbonyl)pyrimidine
2-methyl-3-{[methyl({[2-(2-methylpropoxy)phenyl]methyl})carbamoyl]amino}benzamide
1-cycloheptanecarbonyl-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
5-ethyl-N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-2-methylpyrimidin-4-amine
6-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-1,4-oxazepan-6-ol
4-(2-methyl-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-2-yl)morpholine
1-{[4-(2-hydroxyethoxy)phenyl]methyl}-4-(2-methylquinolin-6-yl)piperidin-4-ol
N-({2-[benzyl(methyl)amino]-2,3-dihydro-1H-inden-2-yl}methyl)-2-(thiophen-2-yl)acetamide
4-(5-fluoropyridin-2-yl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-{5-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]pyrimidin-2-yl}morpholine
[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
6-methoxy-3-({4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}methyl)-1,2-dihydroquinolin-2-one
6-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}pyridine-2-carboxylic acid
N1-cycloheptyl-N3-(pyridin-3-yl)propane-1,3-diamine
5-ethyl-2-{1-[1-(3-methyl-1,2,4-oxadiazol-5-yl)propyl]-1H-imidazol-2-yl}pyridine
1-butyl-3-methyl-4-[(2E)-pent-2-en-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{[1-(dimethylamino)cyclohexyl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
6-methyl-4-oxo-N-[(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-4H-pyran-2-carboxamide
3-(1-methyl-1H-pyrrol-2-yl)-N-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1H-pyrazole-5-carboxamide
(1R,3S)-3-amino-N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}cyclohexane-1-carboxamide
6-methoxy-N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(2-methyl-4-oxo-1,4-dihydroquinolin-1-yl)-N-(2-methylpropyl)acetamide
4-(azepan-1-yl)-N-[3-(dimethylamino)propyl]pyridine-2-carboxamide
5-(4-acetyl-2-methoxyphenoxymethyl)-N-(2,2,2-trifluoroethyl)-1,2-oxazole-3-carboxamide
N,N-dimethyl-2-[2-(morpholin-4-ylmethyl)phenyl]pyridine-3-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-2,5,6-trimethylpyrimidin-4-amine
2-(4-phenylpiperidin-1-yl)-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}acetamide
methyl (2S,4R)-1-[(2-chloro-6-fluorophenyl)methyl]-4-[4-(1H-pyrazol-1-yl)benzamido]pyrrolidine-2-carboxylate
1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}azetidin-3-ol
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-5-phenylpentan-1-one
3-{2-[3-(3-fluorophenoxymethyl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
N-cyclopentyl-1-(1-{[4-(trifluoromethoxy)phenyl]methyl}piperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
N-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-ylmethyl}-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
1-{2-[(2,2-dimethylpropyl)(methyl)amino]ethyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[(5-methyl-1H-imidazol-4-yl)methyl]piperidin-4-amine
N-[(3S,4R)-1-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4-(4-methylphenyl)pyrrolidin-3-yl]acetamide