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1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
3-chloro-N-(4-methoxy-3-pentanamidophenyl)pyridine-4-carboxamide
1-[1-ethyl-5-(propan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl]pyrrolidine
2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperazin-1-yl}-4-(pyridin-2-yl)pyrimidine
3-(3-methoxybenzoyl)-1-[3-(methylsulfanyl)propyl]piperidine
8-chloro-2-({[1-(pyrazin-2-yl)piperidin-3-yl]amino}methyl)quinolin-4-ol
1-{4-[(3,4-dichlorophenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(1H-pyrazol-3-yl)benzamide
N-[(4-ethylphenyl)methyl]-N-(2-methylpropyl)-2-(morpholin-2-yl)acetamide
4-[4-(4-chlorophenyl)-1H-imidazol-2-yl]-1-(propan-2-yl)pyrrolidin-2-one
3-chloro-5-{3-[(3-chlorophenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}-1,2-dihydropyridin-2-one
3-{2-[4-(2-hydroxyethyl)piperazin-1-yl]-2-oxoethyl}-4-[(2-methoxyphenyl)methyl]piperazin-2-one
2-methyl-6-({5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-2,3,4,5-tetrahydropyridazin-3-one
5-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-N-methyl-N-(pyridin-2-ylmethyl)pyridin-2-amine
4-(1-aminocyclopropanecarbonyl)-7-(1-benzothiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N'-[2-(4-fluorophenyl)ethyl]-N'-{[2-(3-hydroxypiperidin-1-yl)-8-methylquinolin-3-yl]methyl}-N,N-dimethylbutanediamide
3-{[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}-N-(1,3-thiazol-2-yl)propanamide
5-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(3-fluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepine
5-[1-ethyl-3-(propan-2-yl)-1H-pyrazol-5-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[3-(5-methylfuran-2-yl)butyl]amine
4-[(2,4-difluorophenyl)methyl]-8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
1-[1-methyl-3-(trifluoromethyl)-1H-thieno[2,3-c]pyrazole-5-carbonyl]-3-(1H-pyrazol-5-yl)piperidine
N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}piperidin-3-amine
[(1-methyl-1H-imidazol-2-yl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})(propan-2-yl)amine
N-(4-methoxy-2-methylphenyl)-3-{1-[4-(propan-2-yloxy)benzoyl]piperidin-3-yl}propanamide
N-[(4-fluorophenyl)methyl]-1-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2H-1,3-benzodioxol-5-ylmethyl)bis(pyridin-3-ylmethyl)amine
6-[(1,4-dioxan-2-ylmethyl)amino]-N-[3-(pyridin-2-yl)propyl]pyridine-3-carboxamide
methyl 4-{methyl[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]carbamoyl}butanoate
N-butyl-N-(furan-2-ylmethyl)-2H-1,3-benzodioxole-5-carboxamide
N-({5-[(3-methyl-1,2-oxazol-5-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)acetamide
2-(furan-2-yl)-N-(6-methylpyridin-3-yl)pyrrolidine-1-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclopropanecarbonyl-2-{3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl}piperidine
4-{3-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidine-1-carbonyl]phenyl}-1λ6-thiomorpholine-1,1-dione
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-{1-[3-(1H-pyrrol-1-yl)propyl]piperidin-4-yl}-3-(pyrrolidine-1-carbonyl)piperidine
N-[2-(2-chlorophenyl)ethyl]-5-methyl-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-(3,5-dimethyl-4-{[2-methyl-4-(2-methylphenyl)piperazin-1-yl]methyl}-1H-pyrazol-1-yl)ethan-1-ol
(3S,5R)-5-(4-methylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxylic acid
2-methoxy-5-oxo-6-{[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
4-(4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)pyridin-2-amine
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-(4-methylpiperidin-1-yl)-N-(2-methylpropyl)propanamide
4-{[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}benzamide
ethyl 1-(oxan-4-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
N-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(naphthalen-1-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
2-{5-[(2-methylphenyl)methyl]-3-(oxolan-3-yl)-1H-1,2,4-triazol-1-yl}ethan-1-ol
methyl 2-[2,4-dioxo-1-(2-phenylethyl)-8-(thiophen-3-ylmethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
9-(6-aminopyridine-3-carbonyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one