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5-(azepane-1-carbonyl)-N-methyl-1-(2-methylpropyl)-4-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N,N-dimethyl-3-({2-[(trifluoromethyl)sulfanyl]ethyl}sulfamoyl)benzamide
3-(2,5-dimethylfuran-3-yl)-5-{thieno[3,2-d]pyrimidin-4-yl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
ethyl 2-{[(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxylate
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridine
3-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]benzonitrile
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-2-methylphenol
3,5-dimethyl-1-(1-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}azetidin-3-yl)-1H-pyrazole
3-(4-butoxyphenyl)-5-(oxolan-3-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}-4-oxo-1,4-dihydroquinoline-2-carboxamide
5-benzyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
4-methoxy-N-(2,3,4,9-tetrahydro-1H-carbazol-6-ylmethyl)piperidine-1-sulfonamide
4-[(1S)-1-phenylpropyl]-3-propyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(oxan-4-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]piperidine-3-carboxamide
2-amino-3-ethyl-N-{[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[1-(piperidin-1-yl)cyclohexyl]methyl}amine
4-(4-fluorophenoxy)-1-[2-(pyridin-4-yl)acetyl]piperidine-4-carboxylic acid
6-ethyl-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-2-(morpholin-4-yl)pyrimidin-4-amine
8-(1H-indol-2-ylmethyl)-1-methyl-3-(propan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-1-(2,2-diphenylacetyl)piperazine-2-carboxamide
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]benzamide
(4aS,7aR)-1-(1-methyl-1H-pyrazole-3-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
3-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
5-methyl-4-[(oxolan-2-ylmethyl)amino]-N-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
methyl (2S,4R)-1-({4-[(dimethyl-1,2-oxazol-4-yl)carbamoyl]phenyl}methyl)-4-hydroxypyrrolidine-2-carboxylate
2-methanesulfonyl-6-methyl-5-[5-(thiophen-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
N-ethyl-N-(1-hydroxypropan-2-yl)-5-methyl-2-phenylfuran-3-carboxamide
N-cyclopropyl-1-{2-[(2-ethyl-6-methylpyridin-3-yl)oxy]acetyl}piperazine-2-carboxamide
2-(3-methoxyphenyl)-6-(3-propoxypiperidine-1-carbonyl)-1,3-benzoxazole
5-(pyridin-3-yl)-5-[1-(1H-pyrrole-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[(3-fluorophenyl)methyl]-3-[2-oxo-2-(4-phenylpiperidin-1-yl)ethyl]piperazin-2-one
2-(1,3-dimethyl-2,5-dioxoimidazolidin-4-yl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-(1-{1-[3-(furan-2-yl)propanoyl]piperidin-4-yl}-2-(3-methoxyphenyl)ethyl)-N-methylpyridine-3-carboxamide
3-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-N-phenylpropanamide
(3S,4S)-1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
(1-{[2-(difluoromethoxy)phenyl]methyl}-4-(2-phenoxyethyl)piperidin-4-yl)methanol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-ol
3-[(1S,3S,3aR,6aS)-3-(hydroxymethyl)-5-methyl-3-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-2-chlorophenol
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
N-ethyl-2,4-dimethyl-N-[2-(3-methylphenoxy)ethyl]-1,3-oxazole-5-carboxamide
2-[3-(3,4-difluorophenyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1H-1,2,4-triazol-1-yl]ethan-1-ol
1-{4-[hydroxy(1-methyl-1H-imidazol-2-yl)methyl]piperidin-1-yl}-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
N-[2-(1-ethyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-azaspiro[5.5]undecan-9-amine
1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]pentane-1,4-dione
1-methyl-4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazine
N-[1-benzyl-4-(propan-2-yloxy)-1H-indazol-3-yl]-1-methylpyrrolidine-3-carboxamide