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N-methyl-5-(oxolan-2-yl)-N-(quinoxalin-2-ylmethyl)thiophene-2-carboxamide
N,N-dimethyl-2-phenyl-7-(pyridine-4-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
4-[({2-methylthieno[2,3-d]pyrimidin-4-yl}amino)methyl]hepta-1,6-dien-4-ol
3-(4-methoxyphenyl)-N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-1H-pyrazole-5-carboxamide
N-cyclopropyl-N-(thiophen-3-ylmethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-{[1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)piperidin-3-yl]methyl}-1H-indole-2-carboxamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-4-phenyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
8-[4-(dimethylamino)-5-methylpyrimidin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[1-(4-fluorophenyl)-2-methylpropan-2-yl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-{1-[2-(3-chlorophenyl)acetyl]piperidin-4-yl}-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
(3S,4S)-1-(1-benzoxepine-4-carbonyl)-4-methylpiperidine-3,4-diol
6-ethyl-N-[(5-methylpyrazin-2-yl)methyl]-2-oxo-1,2-dihydropyridine-4-carboxamide
5-[2-methyl-6-(piperidin-3-yl)pyrimidin-4-yl]-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
[(3-ethoxy-4-methoxyphenyl)methyl]({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-[2-(ethylamino)pyrimidin-5-yl]-N,7,8-trimethyl-N-(propan-2-yl)quinoline-4-carboxamide
1-{4-[(prop-2-en-1-yl)(pyridin-2-ylmethyl)amino]piperidin-1-yl}ethan-1-one
1-(3,4-dimethylphenyl)-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-cyclopentyl-8-[2-(3-methyl-1H-1,2,4-triazol-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
methyl 3-[(furan-2-ylformamido)methyl]-5-[3-(trifluoromethyl)benzenesulfonamido]benzoate
{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}(methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
6-methyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
2-(2-fluoro-4-methoxyphenyl)-4-(1H-imidazol-1-ylmethyl)-5-methyl-1,3-oxazole
6-(4-methylpiperazin-1-yl)-N4-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}pyrimidine-2,4-diamine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(1H-imidazol-4-ylmethyl)piperidine
2-(morpholin-4-yl)-2-(pyridin-3-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
5-(2,4-difluorophenoxymethyl)-N-{[2-(trifluoromethyl)phenyl]methyl}-1,2-oxazole-3-carboxamide
2-ethyl-4-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-1-(propan-2-yl)piperazine
N,N-diethyl-3-(5-phenyl-1,3,4-oxadiazol-2-yl)propanamide
dimethyl[(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-4-yl)methyl]amine
8-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-N-methyl-6-azaspiro[2.5]octane-1-carboxamide
methyl 6-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}-3-(1-phenylcyclopropaneamido)thieno[2,3-b]pyridine-2-carboxylate
4-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
4-[({4-[(diethylamino)methyl]-5-ethylfuran-2-yl}formamido)methyl]benzoic acid
N-butyl-2-methyl-N-(3-phenylprop-2-yn-1-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
(2S)-1-acetyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-methyl-N-(2-{4-[(3-methylthiophen-2-yl)methyl]morpholin-2-yl}ethyl)propanamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-2-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-2-yl}acetamide
(2S,4S)-1-[(3-chlorophenyl)methyl]-4-{[(4-methoxy-2,3-dimethylphenyl)methyl]amino}-N-methylpyrrolidine-2-carboxamide
2-[(2-methylprop-2-en-1-yl)oxy]-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}benzamide
1-(3-{1-methyl-2-oxo-1,2-dihydrospiro[indole-3,4'-piperidine]-1'-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(2-fluorophenyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}cyclopropane-1-carboxamide
(2S)-3-methyl-2-{2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}butanamide
1-[(3-methoxyphenyl)methyl]-4-(2-phenylbutanoyl)piperazin-2-one
4-(1-{[4-(cyclopentyloxy)phenyl]methyl}azetidin-3-yl)morpholine
1-{1-[(3-chloropyridin-4-yl)methyl]piperidin-4-yl}-3-phenylpropan-1-ol
2-({1-[1-(2H-1,3-benzodioxol-5-yl)-1H-1,2,4-triazol-5-yl]ethyl}sulfanyl)pyridine
N-{1-[(5-methylfuran-2-yl)methyl]-1H-pyrazol-5-yl}-2-[4-(pyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-(propan-2-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide