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ethyl 3-[(2-cyclohexyl-1,3-benzoxazol-6-yl)formamido]propanoate
1,7-dimethyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-2-ylmethyl)-1H-indole-2-carboxamide
2-amino-N-[(1S,2R)-2-aminocyclobutyl]-4-methyl-1,3-benzothiazole-6-carboxamide
6-methyl-5-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]-2-(pyrimidin-2-yl)-1,2,3,4-tetrahydro-2,7-naphthyridine
3-{2-[(3aR,6aS)-octahydropyrrolo[3,4-c]pyrrol-2-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
N'-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-N,N-dimethylbutanediamide
4-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[3-(1H-pyrazol-5-yl)piperidin-1-yl]butan-1-one
(1S,5R)-3-[3-(4-methyl-1H-pyrazol-1-yl)propanoyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-(cyclohex-3-en-1-ylmethyl)-4-(4-methylphenoxy)piperidine-4-carboxylic acid
3-(1-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
5-[3-(aminomethyl)pyrrolidin-1-yl]-2-[2-(ethylsulfanyl)ethyl]-2,3-dihydropyridazin-3-one
3-(azetidine-1-carbonyl)-N-(oxolan-3-ylmethyl)benzene-1-sulfonamide
4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-[(5-methylfuran-2-yl)methyl]piperidine
[(1-benzylpyrrolidin-3-yl)methyl]({[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
3-(2-amino-1,3-thiazol-4-yl)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylpropanamide
5-({[1-(2-phenylethyl)piperidin-3-yl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(1-methylpiperidin-4-yl)piperidine-3-carboxamide
(2R,4S)-4-hydroxy-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine-2-carboxylic acid
N-cyclohexyl-1-methyl-N-(pyridin-3-ylmethyl)-1H-indole-4-carboxamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-4-(3-hydroxy-3-methylbutyl)benzamide
N-cyclopropyl-3-{1-[1-(3,5-dimethylphenyl)piperidin-4-yl]piperidin-4-yl}propanamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(4-propanoylphenoxy)acetamide
(2S,4R)-1-[(4-chlorophenyl)methyl]-N-[2-(3-fluorophenyl)ethyl]-4-[(4-fluorophenyl)sulfanyl]pyrrolidine-2-carboxamide
1-{2-methoxy-4-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}-3-(thiomorpholin-4-yl)propan-2-ol
2-methyl-4-[4-({[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]but-3-yn-2-ol
4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
1-{[(2-methylpropyl)[(2E)-3-phenylprop-2-en-1-yl]carbamoyl]methyl}piperidine-4-carboxamide
(2E)-1-[4-(4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(thiophen-3-ylmethyl)benzamide
N-[2-(5-methyl-4-phenyl-1H-imidazol-1-yl)ethyl]aniline
1-{[1-(3-methylphenyl)-1H-imidazol-2-yl]methyl}-3-(pyrrolidin-1-yl)piperidine
N-[1-(2,4-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]acetamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(2-phenyl-1H-imidazol-1-yl)acetamide
2-({[(3R,4R)-1-[(2,6-difluoro-4-methoxyphenyl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-(3-methoxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
5-{2-oxo-2-[3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}imidazolidine-2,4-dione
N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[(pyridin-2-ylmethyl)amino]benzamide
{4-fluoro-3-[2-(propan-2-yloxy)phenyl]phenyl}methanamine
5-(3-fluoro-4-methoxyphenyl)-1-propyl-1H,4H-pyrazolo[3,4-d]imidazole
4-[(4-fluorophenyl)methyl]-1-(3-fluoropyridine-4-carbonyl)-3-(propan-2-yl)-1,4-diazepan-5-one
1-{2-[2-(3-methoxyphenyl)azetidin-1-yl]-2-oxoethyl}piperidin-2-one
methyl 3-[(3S,4R)-4-(dimethylamino)-1-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}piperidin-3-yl]propanoate
N-(1H-1,3-benzodiazol-2-ylmethyl)-N-methyl-5-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)pentanamide
N-{[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]methyl}furan-2-carboxamide
N,N-dimethyl-2-({[2-(3-phenylpropoxy)phenyl]carbamoyl}amino)acetamide
ethyl 4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carboxylate
5-{4-[(3-hydroxypyrrolidin-3-yl)methyl]piperazin-1-yl}-6-phenyl-2,3-dihydropyridazin-3-one
N-ethyl-N-(oxolan-2-ylmethyl)-2-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
6-methyl-2-[3-(1H-pyrazol-3-yl)phenyl]pyridine-3-carboxamide
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(1H-pyrrole-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane