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N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]pyridine-4-carboxamide
3-methanesulfonamido-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}propanamide
2-(2-{[5-(methoxymethyl)furan-2-yl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)-6-methylpyridine
[(3R,4R)-4-[(dimethylamino)methyl]-1-(5-{[(4-methylphenyl)sulfanyl]methyl}furan-2-carbonyl)pyrrolidin-3-yl]methanol
5-chloro-2-{4-[(3-methylpyridin-2-yl)methyl]piperazine-1-carbonyl}-2,3-dihydro-1H-indole
3-(oxolan-2-yl)-7-[1-(trifluoromethyl)cyclopropanecarbonyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
(1S,6R)-9-{6-methylimidazo[2,1-b][1,3]thiazole-3-carbonyl}-3,9-diazabicyclo[4.2.1]nonan-4-one
5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)pyrrolidin-1-yl]methyl}-2-(furan-2-yl)pyrimidine
(1R,3S)-7-(2-cyclopropylpyrimidine-5-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
1-{1-[(4-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-{[2-(pyridin-3-yl)-1H-imidazol-1-yl]methyl}-2,1,3-benzothiadiazole
(4aS,7aR)-1-(2,4-dimethylbenzoyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-1,3-diazinane-2,4-dione
8-(6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1-{1-[(dimethylcarbamoyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-methylbenzamide
2-(oxan-2-ylmethoxy)-1-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecan-4-yl]ethan-1-one
6-cyano-N-[(1R,3S)-3-[(2-ethoxyphenyl)carbamoyl]cyclopentyl]pyridine-3-carboxamide
N-(adamantan-2-yl)-2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
4-{5-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}pyridine
N,N-dimethyl-5-{[3-(naphthalene-1-carbonyl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine
N-benzyl-5-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5-{[2-(5-fluoro-1H-1,3-benzodiazol-2-yl)pyrrolidin-1-yl]methyl}-2-methyl-4H,7H-pyrazolo[1,5-a]pyrimidin-7-one
N-methyl-5-{[methyl(2-phenylethyl)amino]methyl}-N-propyl-1,2-oxazole-3-carboxamide
7-(5-butylpyridine-2-carbonyl)-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
1-(2-oxo-2-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
2-[5-(2-fluoro-6-methoxyphenyl)-4-phenyl-1H-imidazol-1-yl]-1-phenylethan-1-ol
2-(5-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}furan-2-yl)benzonitrile
methyl 5-(2-acetylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
7-[(3-oxo-3,4-dihydroquinoxalin-2-yl)methyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-methyl-5-phenyl-N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
N-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
2-(3-{[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}phenoxy)ethan-1-ol
2-(2-hydroxyethyl)-8-{[4-(trifluoromethyl)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
N-[(4-fluorophenyl)methyl]-3-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]propanamide
1-{1-[(4-methanesulfonylphenyl)methyl]azetidin-3-yl}-3,5-dimethyl-1H-pyrazole
2-(2,3-dimethoxyphenyl)-5,6-dimethylpyridine-3-carboxamide
10-methoxy-N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine-5-carboxamide
4-(5-{[carbamoyl(methyl)amino]methyl}-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl)benzamide
2-methyl-4-[4-({methyl[1-(1,3-thiazol-2-yl)ethyl]amino}methyl)phenyl]butan-2-ol
1-[(4-chlorophenyl)methyl]-N-({4-[2-(pyrimidin-5-yl)ethynyl]phenyl}methyl)piperidin-3-amine
4-[4-(morpholine-4-carbonyl)phenoxy]thiane-4-carboxylic acid
1-{2-[({5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)methyl]morpholin-4-yl}ethan-1-one
2-cyclopentyl-N-[1-(pyrazin-2-yl)propan-2-yl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-methoxy-6-{4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-2-amine
1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}-4-phenyl-1,4-diazepane
(4-{[4-(3,5-dimethyl-1-benzofuran-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methanol
5-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-N,N-dimethylpyridin-2-amine
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)propanamide
N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide
[1-(1-{[2-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol