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N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]butanamide
N-({1-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
4-{1-[(4-fluoro-2-methylphenyl)methyl]pyrrolidin-3-yl}-2-(pyridin-3-yl)pyridine
5-(azocan-1-yl)-1-ethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazole
(3aR,6aR)-N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(2-methoxyacetyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-(2,1,3-benzothiadiazol-5-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}[(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
6-ethyl-N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-2-oxo-1,2-dihydropyridine-4-carboxamide
3-(2-chlorophenyl)-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-3-phenylpropanamide
1-{[6-(2-fluoro-3-methoxyphenyl)pyridin-3-yl]methyl}-4-methylpiperazine
(2S)-2-amino-2-cyclohexyl-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
5-methyl-3-{[3-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-1H-indole
4-(1,3-dimethyl-1H-pyrazol-4-yl)-N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyrimidin-2-amine
{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
(1S,5R)-3-benzoyl-N-(3-cyanophenyl)-3,6-diazabicyclo[3.2.2]nonane-6-carboxamide
[(3S,5R)-5-[(dimethylamino)methyl]-1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)piperidin-3-yl]methanol
N-methyl-5-{[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]methyl}furan-2-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl]benzamide
4-{[1-(3-methyl-1H-indole-2-carbonyl)pyrrolidin-3-yl]methyl}benzoic acid
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl){[1-(2-methylpropyl)piperidin-4-yl]methyl}amine
4-[4-(3-chlorophenyl)pyrimidin-2-yl]-1,4-oxazepan-6-ol
N-[(3-chloro-2-fluorophenyl)methyl]-1-methylazepane-2-carboxamide
2-(4-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-1,4-diazepan-1-yl)-N,N-dimethylacetamide
3-[3-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-6-(propan-2-yl)pyridazine
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]acetamide
6-(2-{4-[(dimethylamino)methyl]phenyl}piperidine-1-carbonyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-[(3,4-difluorophenyl)methyl]-2-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)-2,7-diazaspiro[4.5]decane
(1R,7S)-N-methyl-4-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
3-[(oxolan-3-yl)sulfamoyl]-N-[3-(1H-1,2,4-triazol-1-yl)propyl]benzamide
2-hydroxy-N-{[2-(morpholin-4-yl)pyridin-3-yl]methyl}-2-phenylpropanamide
1-{[2-(ethanesulfonyl)-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
3-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-6-methoxypyridazine
2-(3-{2-[methyl(2-phenylethyl)amino]ethyl}-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl)pyridine-3-carbonitrile
N-({4-[(3-phenylpropyl)amino]quinazolin-2-yl}methyl)-1,3-thiazole-5-carboxamide
2-(2-{[2,2-bis(prop-2-en-1-yl)piperidin-1-yl]methyl}phenoxy)acetic acid
methyl (2S,4S,5R)-4-(cyclopentylcarbamoyl)-5-(2,3-difluorophenyl)-1-methylpyrrolidine-2-carboxylate
1-[2-butyl-4-(3-chlorophenyl)-5-oxopiperazine-1-carbonyl]cyclopropane-1-carboxamide
N-{1-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]ethyl}-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-7-methoxy-N,4-dimethylquinazolin-2-amine
2-{3-[(3,4-difluorophenyl)amino]piperidin-1-yl}-N,N-diethylacetamide
1-(4-methylpiperazin-1-yl)-3-{1-[4-(methylsulfanyl)benzoyl]piperidin-3-yl}propan-1-one
3-{[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}imidazolidine-2,4-dione
1-[(3-methylphenyl)methyl]-3-(oxolan-3-yl)-5-(1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethylquinoline-3-carboxamide
1-[3-(pyridin-3-ylmethoxy)piperidin-1-yl]-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(2-phenoxyethyl)piperidine
N-[3-(1H-pyrazol-1-yl)phenyl]-1-(thian-4-yl)pyrrolidine-2-carboxamide
1-[3-(1-butyl-1H-imidazol-2-yl)piperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
3-[1-(2-chloropyridine-4-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
N,6-dimethyl-N-(thiophen-3-ylmethyl)imidazo[1,2-a]pyridine-2-carboxamide