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(3R,4S)-3,4-dimethyl-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-4-ol
2-(2-aminopyrimidin-5-yl)-N,N,6-trimethylquinoline-4-carboxamide
N-({1-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperidin-4-yl}methyl)acetamide
3-methoxy-2-[(4-{1-[(2-methoxyethyl)(pyridin-2-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
3-{[(4-methanesulfonylmorpholin-2-yl)methyl]amino}-N-(1,3-thiazol-2-yl)propanamide
1-methyl-3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
2-{2-[(4aS,8aR)-4a-(hydroxymethyl)-6-propyl-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
2-ethyl-5-[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]pyrimidine
3-{[2-(4-ethylphenyl)-1H-imidazol-1-yl]methyl}-1-methylpiperidine
3-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4,5,6,7-tetrahydro-1,2-benzoxazole
(2S,4R)-4-amino-1-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-N-methylpyrrolidine-2-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
methyl (2S,4R)-1-(2-chloro-6-methylbenzenesulfonyl)-4-(dimethylamino)pyrrolidine-2-carboxylate
4-{[2-(4-methoxyphenyl)ethyl]amino}-5-methyl-N-(pyridin-4-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
1-cyclopentyl-4-{4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}pyrrolidin-2-one
N-cyclooctyl-2-[3-oxo-1-(pyridin-2-ylmethyl)piperazin-2-yl]acetamide
(1-{1-[3-(furan-2-yl)benzoyl]piperidin-4-yl}-2-phenylethyl)(methyl)(pyridin-4-ylmethyl)amine
2-(2-hydroxyethyl)-8-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[2-(3-benzoylpiperidin-1-yl)-2-oxoethyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-({1-[4-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)propan-1-ol
1-[3-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)propyl]-1H-indazole
N-{[2-(azocane-1-carbonyl)-6-chloroimidazo[1,2-a]pyridin-3-yl]methyl}-1-methylpiperidin-4-amine
2-(1H-imidazol-1-yl)-1-[4-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
4-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)-3-fluoropyridine
2-[2-(4-fluorophenyl)piperidine-1-carbonyl]-N,N-dimethylaniline
N-[(4-ethoxyphenyl)methyl]-3-ethynyl-N-(2-methoxyethyl)benzamide
6-({[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}amino)pyridine-3-carbonitrile
3-chloro-N-cyclopentyl-4-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}oxy)benzamide
4-{4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethyl-6-methylpyrimidine
1-(2-fluorophenyl)-4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
3-(1-methyl-1H-pyrazol-4-yl)-1-[4-(piperidine-1-carbonyl)piperidin-1-yl]propan-1-one
(3aS,6aS)-2-cyclopentanecarbonyl-5-(5-ethylpyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[(1-acetylpiperidin-4-yl)oxy]-N-[(3-chlorophenyl)methyl]-4-methoxybenzamide
3-(2-fluorophenyl)-1-(pyridin-4-ylmethyl)-6-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(1S,5R)-6-(cyclobutylmethyl)-3-[2-(pyridin-2-ylsulfanyl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-cyclopropyl-3-[1-(3-methyl-5,6-dihydro-1,4-dioxine-2-carbonyl)piperidin-3-yl]propanamide
N-(4-methylpyridin-3-yl)-2-(4-phenylmethanesulfonylmorpholin-3-yl)acetamide
1-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
2-[2-(1-{3-[4-(dimethylamino)phenyl]propanoyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
4-[(1S,5R)-6-benzyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-methoxypyridine-3-carbonitrile
3-[1-(1-benzofuran-2-ylmethyl)piperidin-4-yl]-N-cyclopropylpropanamide
2,3-dimethyl-7-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
5-[4-(oxolan-2-ylmethyl)piperazine-1-carbonyl]-N-phenylpyrimidin-2-amine
(2S,4S)-4-amino-1-[(2S)-2-acetamido-4-methylpentanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
(1S,3R)-3-amino-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)cyclopentane-1-carboxamide
2-[4-(6-methoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]-N-methylethane-1-sulfonamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-1-propylpiperidin-4-amine
3-[1-(1-benzothiophen-2-ylmethyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-[2-(dimethylamino)-2-(3-methylthiophen-2-yl)ethyl]-1-propylpiperidin-4-amine
1-{3-[2-(3-methoxyphenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one