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[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]({[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
2-(5-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl)ethan-1-ol
2-[methyl({4-methyl-5-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)amino]ethan-1-ol
7-fluoro-N-(2-methoxyethyl)-3-methyl-N-[(trimethyl-1H-pyrazol-4-yl)methyl]-1H-indole-2-carboxamide
(3S)-1-{[2,5-dimethoxy-4-(methylsulfanyl)phenyl]methyl}-N,N-dimethylazepan-3-amine
(3S,4R)-4-(3-methoxyphenyl)-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidine-3-carboxylic acid
methyl 3-(4-{1-[2-(4-methoxyphenyl)ethyl]-4-methyl-2,5-dioxoimidazolidin-4-yl}piperidine-1-carbonyl)benzoate
4-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}-1-(pyridin-3-ylmethyl)pyrrolidin-2-one
4-cyclohexyl-9-methoxy-7-(4-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(8aS)-2-[(3-phenoxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
ethyl 2-(4-{[(oxan-4-yl)carbamoyl]amino}phenyl)-1,3-oxazole-4-carboxylate
4-{4-[4-(1-methoxyethyl)phenyl]-6-methylpyrimidin-2-yl}morpholine
(3R,4R)-4-ethyl-1-(1H-pyrrole-2-carbonyl)piperidine-3,4-diol
N-{[1-methyl-2-(methylsulfanyl)-1H-imidazol-5-yl]methyl}-3-(1H-pyrazol-1-yl)benzamide
2-amino-6-[2-fluoro-4-(trifluoromethyl)phenyl]-4-(piperidin-4-yl)pyridine-3-carbonitrile
methyl 2-{[(2,6-dimethoxyphenyl)methyl]amino}pyridine-4-carboxylate
4-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}oxane-4-carbonitrile
2-(4-fluorophenyl)-N-(2-{7-[(3-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)acetamide
N-{[4-(3-fluorophenyl)oxan-4-yl]methyl}-[1,2,4]triazolo[1,5-a]pyrimidine-2-carboxamide
methyl 3-[({5-[(2-chloroprop-2-en-1-yl)sulfanyl]-4-(4-methoxyphenyl)-4H-1,2,4-triazol-3-yl}methyl)sulfamoyl]thiophene-2-carboxylate
2-{2-[3-(methoxymethyl)piperidin-1-yl]-4-(morpholin-4-yl)pyrimidin-5-yl}-2-methylpropanoic acid
2-{[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}benzonitrile
(benzylsulfamoyl)(methyl){[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}amine
ethyl 1-[(2-fluorophenyl)carbamoyl]-3-[(2-methylphenyl)methyl]piperidine-3-carboxylate
4-chloro-2-fluoro-N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N-methylbenzamide
1-cyclopentyl-6-oxo-N-[(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)methyl]piperidine-3-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(furan-2-ylmethyl)-2,8-diazaspiro[4.5]decan-3-one
3-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}urea
6-[(4aS,8aR)-4a-(hydroxymethyl)-decahydro-1,6-naphthyridine-6-carbonyl]-5-methyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
4-(4-ethyl-1H-pyrazol-5-yl)-1-[3-(5-methylfuran-2-yl)-1H-pyrazole-5-carbonyl]piperidine
dimethyl({2-[2-(quinolin-8-yl)phenoxy]ethyl})amine
1-(4-acetylpiperazin-1-yl)-3-(3-chlorophenyl)-3-phenylpropan-1-one
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(furan-2-ylmethyl)pyrrolidin-3-yl]-2,4-dimethyl-1,3-thiazole-5-carboxamide
4-{[5-(3-chlorophenyl)furan-2-yl]methyl}-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
N2,N2-dimethyl-6-({[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}methyl)-1,3,5-triazine-2,4-diamine
5-[(1S,3R,3aR,6aS)-3-ethyl-3-(hydroxymethyl)-5-phenyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]-2-methoxyphenol
7-methyl-2-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{[3-(2-fluoro-4-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-4-ol
N-(cyclopropylmethyl)-2-(2,4-dioxo-1,3-diazinan-1-yl)-N-(propan-2-yl)benzamide
N-cyclopropyl-1-{1-[2-(pyridin-2-yl)ethyl]piperidin-4-yl}piperidine-3-carboxamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,9-dioxaspiro[5.5]undecan-4-amine
N-ethyl-1-(2-methoxyacetyl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-methyl-1-{2-[(4-methylphenyl)sulfanyl]ethyl}urea
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4-(4-methylphenoxy)piperidine-4-carboxamide
2-[(3,5-difluorophenyl)methyl]-N,N-dimethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carboxamide
1-phenyl-5-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
1-(2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)azocane
3-benzyl-5-(2,4-difluoro-3-methoxyphenyl)-1H-1,2,4-triazole