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5-methoxy-9-(2-methyl-1-benzofuran-7-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
3-(1-{[2-(piperidin-1-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
1-{[3-(difluoromethoxy)phenyl]methyl}-3-[5-methyl-1-(propan-2-yl)-1H-1,2,4-triazol-3-yl]urea
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-1-methyl-1H-pyrrole-2-carboxamide
2-acetyl-8-(2-methyl-5-propylpyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(3-methoxyphenyl)methyl]-N-(2-methylpropyl)acetamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-ethylpiperidine-4-carboxamide
1-[3-(2-ethyl-1H-imidazol-1-yl)propanoyl]-N-(pyridin-4-ylmethyl)piperazine-2-carboxamide
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-[2-(oxan-2-yl)ethyl]acetamide
(1S,9R)-11-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
2-(5-amino-3-methyl-1H-pyrazol-1-yl)-1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]ethan-1-one
1-{[3-(3-chlorophenyl)-1-methyl-1H-pyrazol-4-yl]methyl}-1,4-diazepan-5-one
N-[(2-chlorophenyl)methyl]-6-({methyl[1-(trimethyl-1H-pyrazol-4-yl)ethyl]amino}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
ethyl 1-{3-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}-4-[(2-chlorophenyl)methyl]piperidine-4-carboxylate
[(3-methyl-1-benzofuran-2-yl)methyl]bis(1,3-oxazol-4-ylmethyl)amine
1-(4-{5-cyclopropyl-1-[4-(2,5-dimethoxyphenyl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
N-[(3-methylpyridin-4-yl)methyl]-4-{[1-(2-phenylethyl)piperidin-4-yl]oxy}benzamide
3-ethyl-4-methyl-N-{2-[2-(trifluoromethoxy)phenyl]ethyl}-1H-pyrazole-5-carboxamide
8-(butan-2-yl)-1-methyl-3-(naphthalen-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[(2S,6S)-4-(oxan-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
7-[1-(furan-2-ylmethyl)piperidine-3-carbonyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridine-4-carbonitrile
5-ethyl-N-[3-(1H-imidazol-1-yl)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
methyl 3-(furan-3-amido)-5-[(5-methylhex-5-en-2-yl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
methyl 2-{[2-(cyclohex-1-en-1-yl)ethyl]sulfamoyl}-6-(4-methyl-2-oxopentanoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-({7-[(2,6-difluorophenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)-5-(methoxymethyl)furan-2-carboxamide
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]acetamide
N-({3-[2-(2-hydroxyethyl)-4-methyl-1H-1,3-benzodiazol-1-yl]phenyl}methyl)propanamide
(3S,4R)-1-[3-(3-chloro-1,2-oxazol-5-yl)propanoyl]-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxypyridine-3-carboxamide
2,3-dimethyl-N-{[4-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-3-ylmethyl)-1H-indole-5-carboxamide
1-(2-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)-4-phenylpyrrolidin-2-one
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-methoxyphenyl)ethan-1-one
2-amino-N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-6-methylpyrimidine-4-carboxamide
2-(2-fluorophenyl)-1-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
1-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-[4-(pyrrolidine-1-carbonyl)phenoxy]piperidine
3-chloro-5-[3-(oxan-4-yl)-1-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]-1,2-dihydropyridin-2-one
N-[(3,5-dimethoxyphenyl)methyl]-N-(1-methoxypropan-2-yl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
4,6-dimethyl-3-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
(2S,4R)-4-amino-N-methyl-1-[2-(2-methylpropanamido)benzoyl]pyrrolidine-2-carboxamide
N-[(4-hydroxy-3-methoxyphenyl)methyl]-1-[(4-methylphenyl)methyl]-5-oxopyrrolidine-3-carboxamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
7-amino-4-[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]-1,2,3,4-tetrahydro-1,8-naphthyridin-2-one
7-methyl-2-[2-(phenylamino)pyrimidine-5-carbonyl]-2,7-diazaspiro[4.5]decan-6-one
N-(2-hydroxyethyl)-N-(thiophen-2-ylmethyl)-2,3-dihydro-1-benzofuran-7-carboxamide
(4aR,8aS)-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-[2-(3-methoxyphenyl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}-1-propyl-1H-pyrazole
N-(1-methyl-1H-1,2,3-benzotriazol-5-yl)-4-(4H-1,2,4-triazol-4-yl)piperidine-1-carboxamide
(3S,4R)-1-(1H-indole-6-carbonyl)-4-methyl-3-(2-methylpropyl)piperidin-4-ol
2-[2-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]acetamide
2-methyl-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}butan-1-one