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ethyl 4-[(4-chlorophenyl)methyl]-1-[2-(dimethylamino)benzoyl]piperidine-4-carboxylate
8-(4-aminopyrimidin-2-yl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(4aS,8aR)-1-(3-methoxypropyl)-6-[3-(2-methylphenyl)propanoyl]-decahydro-1,6-naphthyridin-2-one
(2,1,3-benzoxadiazol-5-ylmethyl)[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]amine
[(1-cyclohexylpiperidin-3-yl)methyl][(5-methylfuran-2-yl)methyl](pyridin-3-ylmethyl)amine
(2S,4S)-4-amino-N,N-diethyl-1-(1-methyl-2-oxo-1,2-dihydroquinoline-3-carbonyl)pyrrolidine-2-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[1-(pyridin-3-yl)propyl]benzamide
(1-{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)methanol
2-{[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}benzonitrile
6-[3-(hydroxymethyl)piperidin-1-yl]-N-[(3-propyl-1,2-oxazol-5-yl)methyl]pyridine-3-carboxamide
5-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)furan-2-carboxylic acid
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(pyrrolidin-3-yl)benzamide
{[1-(3-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-pyrazol-4-yl]methyl}[3-(pyridin-3-yl)propyl]amine
3-(3-fluorophenyl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1H-pyrazole-4-carboxamide
3-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
N-{3-oxo-3-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propyl}methanesulfonamide
3-methanesulfonamido-N-phenyl-5-[({[4-(trifluoromethoxy)phenyl]methyl}amino)methyl]benzamide
{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}(methyl){[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amine
2-(2-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}ethyl)-1H-1,3-benzodiazole
1,3-dimethyl-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
ethyl[(2-fluorophenyl)methyl]({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amine
methyl (2S,4S)-1-benzyl-4-(4-methylbenzamido)pyrrolidine-2-carboxylate
(2S,4S)-N-ethyl-1-[(4-methyl-1,3-thiazol-5-yl)methyl]-4-(thiophene-3-amido)pyrrolidine-2-carboxamide
5-(2-ethylpiperidine-1-carbonyl)-1-(2-methoxyethyl)-4-oxo-N-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3-carboxamide
N-methyl-N-[3-(1-methyl-1H-pyrazol-4-yl)propyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[2-(pyrimidin-2-ylsulfanyl)acetyl]piperidin-4-yl}propanamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butan-1-one
1-(cyclopropylmethyl)-5-(furan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
2-({3-[2-(4-ethylpiperazin-1-yl)ethyl]-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)benzonitrile
(2R,6S)-4-(6-chloro-3-{4H,5H,6H,7H-thieno[3,2-c]pyridin-5-ylmethyl}imidazo[1,2-a]pyridine-2-carbonyl)-2,6-dimethylmorpholine
4,7-dimethyl-2-(3-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}piperidin-1-yl)quinazoline
(3R,4R)-4-ethyl-1-(2-methyl-1,3-benzoxazole-6-carbonyl)piperidine-3,4-diol
N-[4-(3-methylphenyl)phenyl]-1-[3-(methylsulfanyl)propanoyl]piperidine-4-carboxamide
N-(1-carbamoylcycloheptyl)-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
4-(5-acetylthiophene-3-carbonyl)-6-[(3,5-dimethoxyphenyl)methoxy]-1-(propan-2-yl)-1,4-diazepan-2-one
2-{1-[(2-butyl-1H-imidazol-4-yl)methyl]piperidin-4-yl}-4-methyl-1H-1,3-benzodiazole
3-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzonitrile
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-[2-({[1-(2-cyclohexylethyl)-3-hydroxy-2-oxopiperidin-3-yl]methyl}amino)ethyl]acetamide
N-{[7-(pyrimidin-2-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-1,3-thiazole-5-carboxamide
1-{2-[(4-methoxyphenyl)methyl]morpholin-4-yl}-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(pyridin-3-yl)ethan-1-one
1-methyl-6-oxo-N-[3-(1H-pyrazol-1-yl)propyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-[2-({[3-(1H-pyrazol-1-yl)phenyl]methyl}amino)propyl]-3,4-dihydroquinazolin-4-one
N-[2-(2-chloro-6-fluorophenyl)ethyl]-2-(phenylamino)pyrimidine-5-carboxamide
3-(2-phenylethyl)-8-(pyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
methyl (1R,5S,6R)-6-{[(2,3-dihydro-1H-inden-2-yl)(methyl)amino]methyl}-3-azabicyclo[3.1.0]hexane-3-carboxylate
N-cyclohexyl-4-(1H-pyrazol-4-yl)-N-(pyridin-3-ylmethyl)butanamide
3-chloro-6-{4-[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}pyridazine
N-ethyl-N-methyl-2-(1H-pyrazol-3-yl)pyrimidin-4-amine