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4-(benzyloxy)-1-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(4aR,7aS)-4-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(5-methylhexanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
5-ethyl-1'-{[3-(morpholin-4-yl)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(piperidin-1-yl)-N-(piperidin-4-yl)-2,3-dihydro-1H-indene-2-carboxamide
1-[3-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)phenyl]ethan-1-one
(1R,3S)-N3-ethyl-N1-[2-hydroxy-2-(prop-2-en-1-yl)pent-4-en-1-yl]-1,2,2-trimethylcyclopentane-1,3-dicarboxamide
4-(6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridazin-3-yl)thiomorpholine
1-(4-cyclopentylpyrimidin-2-yl)-N-ethylpyrrolidine-3-carboxamide
(3aS,6aS)-2-(2-methoxyethyl)-5-[(2-methylpyridin-3-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-cyclopropyl-8-{[4-(2-hydroxyethoxy)phenyl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
4-tert-butyl-6-[(1S,5R)-3-methyl-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,2-dihydropyrimidin-2-one
(5-methyl-3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,2-oxazol-4-yl)methanol
(3R,4R)-1-[2-(benzenesulfonyl)ethyl]-3-methyl-4-(oxan-4-yl)piperidin-4-ol
2-(2,3-dihydro-1H-inden-1-yl)-N-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}acetamide
(1S,5R)-6-[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
5-{[3-(3,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
4-{6-[2-(pyridin-2-yl)pyrrolidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
4-{pyrazolo[1,5-a]pyridine-7-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
4-[4-(1-hydroxyethyl)phenyl]benzamide
2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]quinoxaline
2-methyl-4-(4-{[(2S)-2,4,5,5-tetramethylpiperazin-1-yl]methyl}phenyl)butan-2-ol
2-[2-(propan-2-yl)-1H-imidazol-1-yl]-N-{2-[2-(pyrazin-2-yl)-1,3-thiazol-4-yl]ethyl}propanamide
N-[(4-methylphenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
(1S,5R)-6-[(4-chloro-2-fluorophenyl)methyl]-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
8-(3-fluoropyridine-4-carbonyl)-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
2-({3-[4-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)-1,3-benzothiazole
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-methyl-N-[1-(pyridin-4-yl)ethyl]acetamide
2-(pyridin-4-yl)-5-[4-(thiophen-2-ylmethyl)piperazine-1-carbonyl]pyrimidine
4-(isoquinolin-5-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
6-({3-[4-(pyridin-4-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methoxy)quinoline
methyl 2-{2,8-diazaspiro[4.5]decane-2-sulfonyl}benzoate
N-methyl-3-[5-(4-phenylbutyl)-1,3,4-oxadiazol-2-yl]-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]propanamide
1-(5-acetyl-2-ethoxyphenyl)-3-[(1-methyl-1H-imidazol-2-yl)methyl]-3-propylurea
1-(4-hydroxypiperidin-1-yl)-2-(4-{4-[(oxan-4-ylmethyl)amino]piperidin-1-yl}phenyl)ethan-1-one
1-[benzyl(methyl)amino]-3-(4-{[4-(3-methoxypropyl)piperidin-1-yl]methyl}phenoxy)propan-2-ol
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-propyl-1,3-thiazole-4-carboxamide
4-fluoro-3-[3-(3-methoxypropyl)piperidine-1-carbonyl]benzene-1-sulfonamide
3-(1-ethyl-1H-1,2,3,4-tetrazol-5-yl)-1-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]urea
6-{methyl[(4-methyl-1,3-thiazol-2-yl)methyl]amino}-N-[2-(1-methylpiperidin-2-yl)ethyl]pyridine-3-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2,5-dimethylpyrimidine
[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl][3-(pyridin-3-yloxy)propyl]amine
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-2,5,6-trimethylpyrimidin-4-amine
7-(1H-imidazole-2-carbonyl)-N2,N2,N4,N4-tetramethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
1-(1-{[4-ethoxy-3-(hydroxymethyl)phenyl]methyl}piperidin-4-yl)piperidine-3-carboxylic acid
N-[(1-ethylpiperidin-3-yl)methyl]-N-methyl-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-4-(1H-pyrazol-4-yl)butan-1-one
2-amino-1-[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2,3-dimethylbutan-1-one
2-cyclopropyl-5-{2-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl}pyrimidin-4-ol