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N-(2-methyl-1-{3-[(3-methylphenyl)methyl]-1,2,4-oxadiazol-5-yl}propyl)acetamide
(4R)-N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-oxo-1,3-thiazolidine-4-carboxamide
3-(3-fluorophenyl)-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
1-(cyclopentylcarbamoyl)-4-[(2-methylpyridin-3-yl)oxy]piperidine-4-carboxylic acid
(3S,7S,8aS)-7-[({3-[(diethylamino)methyl]-4-methoxyphenyl}methyl)amino]-3-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
3-{2-[4-(2-chlorophenyl)-3-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-hydroxy-1-{[4-(propan-2-yl)phenyl]methyl}-3-({[2-(pyridin-2-yl)ethyl]amino}methyl)piperidin-2-one
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopentanecarboxamide
N-(3-chloro-4-fluorophenyl)-3-{4-[(2-methyl-1,3-thiazol-4-yl)methyl]piperazin-1-yl}-3-oxopropanamide
1-{1-[1-(1-butyl-1H-1,2,4-triazol-5-yl)propan-2-yl]-3,5-dimethyl-1H-pyrazol-4-yl}ethan-1-one
(4S)-4-(methoxymethyl)-1-[5-(methoxymethyl)furan-2-carbonyl]-3,3-dimethylpiperidin-4-ol
(2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazol-4-yl)methanol
N-[(4-hydroxyphenyl)methyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
1-ethyl-5-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1H-pyrazole-4-carboxamide
7-[(2,3-dimethoxyphenyl)methyl]-3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
1-(3-{[4-(2-methoxyethyl)piperazin-1-yl]methyl}-7-methylimidazo[1,2-a]pyridine-2-carbonyl)azepane
N-cyclopropyl-1-{1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
2-[(1-ethylpyrrolidin-2-yl)methyl]-6-(thiomorpholine-4-carbonyl)-2,3-dihydro-1H-isoindol-1-one
ethyl 4-({1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}amino)piperidine-1-carboxylate
1-(7-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-2,7-diazaspiro[4.5]decan-2-yl)-2,2-dimethylpropan-1-one
1-(2-methyl-1-benzofuran-5-carbonyl)piperazine-2-carboxylic acid
7-cyclopentyl-2-(morpholine-4-sulfonyl)-2,7-diazaspiro[4.5]decan-6-one
3-(pyridin-4-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
N-[2-(3-ethylphenoxy)ethyl]-N,2-dimethylpyrido[2,3-d]pyrimidin-4-amine
(4aS,8aR)-6-[(5-ethylpyridin-2-yl)methyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
(4aS,7aR)-1-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)pyrrolidine
3-[1-(2-amino-6-methylpyrimidin-4-yl)piperidin-3-yl]-N-[(2-fluorophenyl)methyl]propanamide
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-6-oxopiperazine-2-carboxamide
(1R,3S)-N-(2,4-dichlorophenyl)-1,3-dihydroxy-7-azaspiro[3.5]nonane-7-carboxamide
1-{7-methylimidazo[1,2-a]pyridine-2-carbonyl}-4-(2-methylpyridin-4-yl)piperazine
N-[2-(1-methylpyrrolidin-2-yl)ethyl]-5-(morpholin-4-ylmethyl)furan-3-carboxamide
(2S)-N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-(1,3-oxazole-5-carbonyl)pyrrolidine-2-carboxamide
ethyl 1-[3-(furan-2-yl)propanoyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
3-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carbonyl)-N,N-dimethylaniline
6-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carbonitrile
5-{[4-(3-methylphenoxy)piperidin-1-yl]methyl}-N-propylpyrimidin-2-amine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[3-(methylsulfanyl)propyl]piperidine-3-carboxamide
3-(piperidine-1-carbonyl)-2-(pyridin-4-yl)pyridine
N-methyl-4-(1H-pyrazol-4-yl)-N-[1-(pyridin-3-yl)propyl]butanamide
2-benzyl-4-[1-(pyridin-3-ylmethyl)piperidin-4-yl]morpholine
5-methyl-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-{1-[(3-hydroxypyrrolidin-3-yl)methyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
4-(1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidine-4-carbonyl)morpholine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]piperidine-4-carboxamide
5-[4-(1,3-benzoxazol-2-yl)piperazine-1-carbonyl]-2-tert-butylpyrimidin-4-ol
4-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1-propylpiperidine
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-2-phenylethyl}-N,2-dimethylfuran-3-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-{3-oxo-1-[(4-phenylphenyl)methyl]piperazin-2-yl}acetamide
3-{[2-(4,5-dimethylfuran-2-yl)-1H-imidazol-1-yl]methyl}-1λ6-thiolane-1,1-dione