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1-[2-(dimethylamino)acetyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
3-methyl-8-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4-{3-azaspiro[5.5]undecan-9-yl}-1λ6-thiomorpholine-1,1-dione
2-{6-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-methylpyrimidin-4-yl}ethan-1-amine
6-[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
2-({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)-1-[2-(trifluoromethyl)phenyl]ethan-1-ol
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
3-{[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]methyl}-1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]urea
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl})amine
N-[2-(3-{[methyl(1,3-thiazol-4-ylmethyl)amino]methyl}phenoxy)propyl]cyclohexanecarboxamide
4-ethyl-1-methyl-3-[1-(quinolin-2-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(3R,5R)-5-(morpholin-4-ylmethyl)-1-(pyrrolidine-1-sulfonyl)piperidin-3-yl]methanol
4-oxo-4-(3-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-1-yl)butanamide
2-acetamido-N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)acetamide
(3S,4S)-1-{[2-(ethylamino)pyrimidin-5-yl]methyl}-4-(naphthalen-2-yl)piperidin-3-ol
2-{2-[4-phenyl-5-(2,4,6-trimethylphenyl)-1H-imidazol-1-yl]ethoxy}ethan-1-ol
2-{4-[4-(6-ethylpyrimidin-4-yl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
N-[(3-chloro-4,5-dimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
6-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]pyridine-2-carboxylic acid
(3S)-1-({5-[(3-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-fluoropyrrolidine
methyl (2S)-1-(2-cyclobutaneamido-7-oxo-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carbonyl)pyrrolidine-2-carboxylate
3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-(3-fluorophenyl)-5-(thian-4-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-[2-(methylamino)ethyl]-decahydro-1,6-naphthyridin-2-one
3-[(2-amino-6-ethyl-5-methylpyrimidin-4-yl)amino]-N-cyclohexylpropanamide
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(pyridine-4-carbonyl)piperidin-3-amine
N-cyclopentyl-N-[(5-methylthiophen-2-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
1-(1-benzothiophen-2-ylmethyl)-4-[2-(oxolan-2-yl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
methyl 2-{[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]sulfonyl}benzoate
(3R,4S)-3,4-dimethyl-1-[1-(morpholin-4-yl)cyclohexanecarbonyl]piperidin-4-ol
4-[(2-aminopyridin-3-yl)methyl]-3-methyl-1-(2-methylpropyl)piperazin-2-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(2,5-dioxoimidazolidin-1-yl)acetamide
N-[(3R,4S)-1-acetyl-4-(propan-2-yl)pyrrolidin-3-yl]-3-(morpholin-4-yl)benzamide
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-6-fluoroquinolin-4-ol
N-cyclopentyl-1-(2-methylpropyl)-5-(pyridine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-ethoxy-3-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]pyridine
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-[3-(1H-pyrazol-1-yl)propyl]-1,2-oxazole-3-carboxamide
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-cyclopropyl-5-(3-methyl-1-propyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(2-ethyl-1H-1,3-benzodiazol-1-yl)butanamide
3-{[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,3-oxazolidin-2-one
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]-5-(2-fluorophenyl)-1,2,4-triazin-3-amine
2-methyl-6-{1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidin-3-yl}-3,4-dihydropyrimidin-4-one
2-(2,4-dimethoxyphenyl)-2-[methyl(quinolin-4-ylmethyl)amino]acetic acid
5-{1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-imidazol-2-yl}-2-(thiophen-2-yl)pyrimidine
N-(4-fluorophenyl)-1-[2-(pyridin-4-ylsulfanyl)acetyl]piperazine-2-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-N-[2-(pyridin-4-yl)ethyl]acetamide
1-[2-(4-phenyl-1,4-diazepan-1-yl)pyrimidin-4-yl]piperidin-3-ol
2-[(2-hydroxyethyl)({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})amino]ethan-1-ol
1-[4-(4-{[5-methyl-2-(5-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one