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3-(4-chloro-1H-pyrazol-1-yl)-1-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]propan-1-one
2-amino-4-{3-[(dimethylamino)methyl]-4-hydroxyphenyl}-8-hydroxy-5H-indeno[1,2-b]pyridine-3-carbonitrile
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-cyclopentyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
7-(cyclopropylmethyl)-N-ethyl-N-methyl-8-oxo-6-(thiophen-2-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-cyclopropyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]quinoline-4-carboxamide
N-(1-ethyl-1H-1,2,4-triazol-3-yl)-3-(3-methoxyphenoxy)azetidine-1-carboxamide
methyl (2S,4R)-1-(5-{[benzyl(methyl)amino]methyl}-1,2-oxazole-3-carbonyl)-4-hydroxypyrrolidine-2-carboxylate
1-[5-(2,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-2-(1,3-thiazol-2-yl)piperidine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
N-cyclopentyl-3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
5-(3-methoxyphenyl)-N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]furan-2-carboxamide
(2E)-N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-3-(1-methyl-1H-pyrazol-4-yl)prop-2-enamide
4-{2-[(4aR,8aR)-6-(3-phenylpropanoyl)-decahydro-1,6-naphthyridin-1-yl]-2-oxoethyl}-7-methyl-2H-chromen-2-one
[3-(furan-2-carbonyl)-9-[3-(1H-pyrazol-1-yl)propyl]-3,9-diazaspiro[5.5]undecan-1-yl]methanol
4-[(1-{[2-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)methyl]morpholine
5-chloro-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
5-(methoxymethyl)-N-{[7-(pyridin-3-yl)-1H,2H-naphtho[2,1-b]furan-2-yl]methyl}furan-2-carboxamide
2-cyclopropanecarbonyl-8-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(1S,5R)-6-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-3,5-dimethyl-N-[2-(1-methylpiperidin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-(3-methoxyphenyl)propanamide
4-{4-[1-(morpholin-4-yl)ethyl]phenyl}-6-(pyrrolidin-1-yl)pyrimidin-2-amine
[3-(1H-imidazol-1-yl)propyl]({[5-(1H-pyrazol-5-yl)furan-2-yl]methyl})(pyridin-4-ylmethyl)amine
1-[2-(dimethylamino)ethyl]-N-[2-(5-methylfuran-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
(4aS,7aR)-1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-(1-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}pyrrolidin-3-yl)acetamide
ethyl 2-{4-[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]piperazin-1-yl}acetate
3-methyl-8-(2,3,6-trimethylquinoline-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2-methoxyphenyl)-2-methyl-1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperazine
9-[(2-aminopyridin-3-yl)methyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
N3-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-1,3-dicarboxamide
4-(2-fluorophenoxy)-1-(3-phenylpropyl)piperidine-4-carboxylic acid
({3-methoxy-2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)[2-(1H-1,2,4-triazol-1-yl)propyl]amine
3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine
1-{1-[(4-ethoxyphenyl)methyl]piperidin-4-yl}-4-(pyrrolidine-1-carbonyl)piperidine
[(3R,5R)-1-[(5-cyclopentylthiophen-2-yl)methyl]-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
(3R,5S)-N3-(2,3-dihydro-1H-inden-5-yl)-1-[(4-hydroxyphenyl)methyl]-N5-[(2-methoxyphenyl)methyl]piperidine-3,5-dicarboxamide
methyl 6-[(2-chloro-6-fluorophenyl)methyl]-2-[(2-methoxyethyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-butyl-8-[2-(methylamino)-1,3-thiazole-4-carbonyl]-2,8-diazaspiro[5.5]undecan-3-one
6-(2-chlorophenyl)-N-(2-hydroxyethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
methyl 3-(oxolane-2-amido)-1-(2-phenylethyl)-5-[(propan-2-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
3-{3-[3-(dimethylamino)pyrrolidin-1-yl]propyl}-8-(pyridine-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(3-methyl-1H-pyrazol-5-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
5-cyclobutanecarbonyl-1'-(1,3-thiazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(1H-indol-4-yl)-2-oxo-7-(pyrrolidin-1-yl)-1,2,3,4-tetrahydroquinoline-6-carboxamide
1-(2-methyl-5-{1-methyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}phenyl)imidazolidin-2-one
1-[3-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenoxy]-3-(morpholin-4-yl)propan-2-ol
N-[3-hydroxy-2-(thiophen-3-ylmethyl)propyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol