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9-oxo-N-propyl-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
2-[(6-amino-2-{[(4-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)amino]-N,N-dimethylethane-1-sulfonamide
4-{1-[2-(4-phenyl-1,3-thiazol-2-yl)-1H-imidazol-1-yl]ethyl}pyrimidine
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetamide
methyl 2-[2-(2-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}acetamido)-1,3-thiazol-5-yl]acetate
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
N-cyclopentyl-3-[5-(2-methylpentanoyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanamide
7-[(3-methoxyphenyl)methyl]-2-[3-(methylsulfanyl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-1,4-diazepane
ethyl 4-[1-(2-methoxyethyl)-2,4-dioxo-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-8-yl]piperidine-1-carboxylate
1-[(2-fluoro-4-methylphenyl)methyl]-4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
6-oxo-1-(2-phenylethyl)-N-[2-(pyridin-3-yloxy)ethyl]piperidine-3-carboxamide
N-[(1S,2S)-2-(benzyloxy)cyclohexyl]-2-methyl-1,3-thiazole-4-carboxamide
1-(2-{[2-amino-6-(propan-2-yloxy)pyrimidin-4-yl]amino}ethyl)-4,6-dimethyl-1,2-dihydropyrimidin-2-one
1-(2-methoxyethyl)-6-oxo-N-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine
2-(3,5-dimethyl-1H-pyrazol-4-yl)-N-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]acetamide
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-3-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1,4-dihydropyridin-4-one
2-benzyl-9-(4,4,4-trifluorobutyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(cyclopropylamino)-2-ethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
{2-[1-(3-chloro-2-methylphenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]ethyl}urea
N-(4-fluoro-3-methylphenyl)-3-(morpholin-4-ylmethyl)piperidine-1-carboxamide
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
2-{[3-(methoxymethyl)pyrrolidin-1-yl]methyl}-1-(2-methylpropyl)-1H-1,3-benzodiazole
{4-[(4-chlorophenyl)methyl]-1-(1-methoxypropan-2-yl)piperidin-4-yl}methanol
1-(4-{[3-(2-hydroxyethyl)-4-(2-phenylethyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
N-methyl-N-(oxan-4-yl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
1-cyclohexyl-N3-[1-(4-fluorophenyl)ethyl]-N5-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
(4S)-1-{2-[(dimethylamino)methyl]benzoyl}-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
(1R,7S)-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(6-aminopyridin-3-yl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
7-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-(4-{2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamido}phenyl)pentanamide
(3S,4R)-3-benzyl-4-methyl-1-propylpiperidin-4-ol
(1S,3R)-N-(4-chloro-3-methylphenyl)-3-[2-(2-oxo-1,3-oxazolidin-3-yl)acetamido]cyclopentane-1-carboxamide
1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-3-(2-ethyl-1H-1,3-benzodiazol-6-yl)urea
(2S)-2-amino-4-methyl-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]pentan-1-one
4-oxo-N-[3-(pyridin-2-yl)propyl]-3,4-dihydrophthalazine-1-carboxamide
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]acetamide
2-[(4-chlorophenyl)methyl]-8-[(2S)-2-(methylamino)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-[2-(4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
2-[(2,6-dichlorophenyl)methyl]-4-hydroxy-N-[2-(1H-imidazol-1-yl)propyl]pyrimidine-5-carboxamide
[(2-fluoro-4,5-dimethoxyphenyl)methyl](methyl)(1H-pyrazol-3-ylmethyl)amine
{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[1-(1,3-thiazol-2-yl)ethyl]amine
3-butanamido-N-{1-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]ethyl}benzamide
1-{[3,5-dimethyl-2-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyridin-3-yl)piperidin-4-ol
3-[(3R,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-fluorophenyl)urea
1-benzyl-8-(cyclohex-3-en-1-ylmethyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
7-(5-ethoxyfuran-2-carbonyl)-3,5-dimethyl-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyrazine
3-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1-[4-(2-oxopyrrolidin-1-yl)phenyl]urea