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N-(2-{4-[(5-ethylpyridin-2-yl)methyl]morpholin-2-yl}ethyl)acetamide
1-(2-methoxyethyl)-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-6-oxopiperidine-3-carboxamide
methyl 8-{[4-(benzyloxy)phenyl]methyl}-2-oxo-1-(prop-2-en-1-yloxy)-1,8-diazaspiro[4.5]decane-4-carboxylate
1-(2-ethoxyethyl)-5-(pyrrolidine-1-carbonyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(8-methoxyquinolin-5-yl)methyl]-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
(2S,4R)-1-[(2-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]-N-(2-methyl-1,3-benzothiazol-5-yl)pyrrolidine-2-carboxamide
1-[4-(2-methoxybenzoyl)piperazin-1-yl]-3-(thiophen-2-yl)propan-1-one
4-[4-(2-chlorophenyl)piperidin-4-yl]-2-(1H-1,2,4-triazol-1-ylmethyl)pyrimidine
propan-2-yl 4-chloro-3-({[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]carbamoyl}amino)benzoate
5,6-dimethyl-N-[4-(1H-pyrazol-1-yl)butan-2-yl]pyrimidin-4-amine
1-[(3S,4S)-3,4-dihydroxypiperidin-1-yl]-3-[(4-phenylphenyl)amino]propan-1-one
4-(2-hydroxy-4-methylpentanoyl)-1-(2-methylphenyl)piperazin-2-one
2-{3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]piperidin-1-yl}acetamide
3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridin-2-amine
1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-5-oxopyrrolidine-3-carboxylic acid
3-[2-(3-methyl-1,2-oxazol-5-yl)acetamido]-4-(2-methylpiperidin-1-yl)benzamide
1-[2-(furan-2-yl)-2-oxoacetyl]-3-methylpiperidine-3-carbonitrile
N-ethyl-2-{4-[2-(3-phenylpyrrolidin-1-yl)acetyl]piperazin-1-yl}acetamide
1-(oxane-4-carbonyl)-3-(4-phenylbenzoyl)piperidine
methyl 4-[5-({2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}methyl)-1,2,4-oxadiazol-3-yl]benzoate
2-(cyclopropylmethyl)-8-(6-methoxypyrimidin-4-yl)-2,8-diazaspiro[5.5]undecan-3-one
6-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-2-carboxylic acid
1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(1-methyl-1H-imidazol-2-yl)piperidine
methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
(1R,2S)-1-(2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazol-1-yl)-2,3-dihydro-1H-inden-2-ol
1-(4-butoxyphenyl)-3-(oxan-4-yl)urea
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]propan-1-one
N-cyclopentyl-4-(4-methylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
2-{[1-(4-methoxy-3-methylphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}pyridine
(3S,4R)-1-{[cyclohexyl(methyl)carbamoyl]methyl}-4-phenylpyrrolidine-3-carboxylic acid
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
ethyl 3-[(3,5-dimethyl-1-benzofuran-2-yl)formamido]hexanoate
8-fluoro-3-(morpholin-2-ylmethyl)-3,4-dihydroquinazolin-4-one
N-[(2R,3R)-1'-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-2-(pyridin-4-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]acetamide
methyl 4-{2-amino-3-cyano-5H,6H,7H,8H,9H-cyclohepta[b]pyridin-4-yl}-1H-pyrazole-3-carboxylate
2-{8-methylimidazo[1,2-a]pyridin-3-yl}-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(1,3-dihydroxypropan-2-yl)-1,3-oxazole-4-carboxamide
1-[1-(3-aminopropanoyl)piperidin-4-yl]-N-(2-phenylethyl)piperidine-3-carboxamide
4-chloro-N-cyclopropyl-1-ethyl-N-[(2-methoxyphenyl)methyl]-1H-pyrazole-5-carboxamide
N-phenyl-5-{1-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
4-{[5-(1-cyclohexylpiperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}morpholine
7-(1-benzothiophen-3-yl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-(2-hydroxyphenyl)-6-methylpyrimidin-4-yl]azetidin-3-ol
2-(3-methoxypropyl)-8-(pyridine-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4,6-dimethyl-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazolo[3,4-b]pyridin-3-amine
2-{4-[3-(1H-pyrazol-1-yl)benzoyl]morpholin-2-yl}ethan-1-ol
(3aS,6aS)-2-methyl-5-[2-(phenylformamido)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-chloro-N-{[1-(dimethylsulfamoyl)piperidin-3-yl]methyl}benzamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
2-(3-hydroxypropyl)-8-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,8-diazaspiro[5.5]undecan-3-one