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N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
3-[5-(1H-1,2,3-benzotriazole-5-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-1-(9H-purin-6-yl)piperidin-4-amine
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl](methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N-{2-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-1,2,3,4-tetrahydroisoquinolin-7-yl}pyridine-2-carboxamide
1-[(4aS,8aS)-4a-hydroxy-7-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-3-methylbut-2-en-1-one
5-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-1H-indole
(2R,4S)-1-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-4-hydroxypiperidine-2-carboxylic acid
1-[(2R,3R,6R)-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-2-amine
2-(cyclopropylmethyl)-9-[3-(pyridin-3-yl)propyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopropyl-4-methoxy-2-{[1-(1-phenoxypropan-2-yl)piperidin-4-yl]oxy}benzamide
[1-(6-methylpyridazin-3-yl)piperidin-4-yl](pyridin-2-yl)methanol
1-{1'-[(2-ethoxyphenyl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-cyclobutyl-3-[3-(trifluoromethyl)benzoyl]piperidine
3-{5-[(benzyloxy)methyl]-4-phenyl-1H-imidazol-1-yl}-1-(pyrrolidin-1-yl)propan-1-one
N-(3-methyl-1-{7-[(2E)-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}butyl)furan-2-carboxamide
4-[(2-aminopyridin-3-yl)methyl]-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(1S,6R)-9-(pyrimidin-5-ylmethyl)-3,9-diazabicyclo[4.2.1]nonane
N-(4-fluorophenyl)-1-(1H-pyrazol-3-ylmethyl)piperidin-3-amine
N-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
N-(oxolan-2-ylmethyl)-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-3,4-dimethoxy-N-(oxolan-2-ylmethyl)benzamide
2-methyl-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]oxolane-2-carboxamide
2-(3-{[4-(4,6,7-trimethylquinazolin-2-yl)-1,4-diazepan-1-yl]methyl}phenoxy)ethan-1-ol
6-methoxy-1-(7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepin-3-yl)hexan-1-one
3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(3-methylphenyl)-4H-1,2,4-triazole
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-2-methyl-N-(2-methylpropyl)furan-3-carboxamide
4-benzyl-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3-methyl-6-{5-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}pyridazine
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-3-(piperidin-4-ylmethyl)benzamide
7-(2-methoxyacetamido)-N-methyl-1-(2-phenylethyl)-N-(thiophen-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(4-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}morpholin-3-yl)acetic acid
4-(3-methoxy-6-methylpyridin-2-yl)-N-(pyridin-4-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-({2-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-imidazol-1-yl}methyl)pyridine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[(3-fluoro-2-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]pyridin-3-ol
N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-6-(2-methylphenyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
2-methyl-4-[5-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)furan-2-yl]but-3-yn-2-ol
N,5-dimethyl-N-(1-methylpyrrolidin-3-yl)-7-(trifluoromethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-(4-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}phenyl)ethan-1-amine
N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-1,2-oxazole-3-carboxamide
9-[2-(morpholin-4-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecan-5-ol
1-(4-chloro-1,3-dimethyl-1H-pyrazole-5-carbonyl)-4-(2-phenoxyethyl)piperazine
1-cyclopropyl-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]piperidin-2-one
6-methyl-N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carboxamide
N-({1-[(3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}methyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
3-(3-methoxyphenoxymethyl)-1-(2-methylfuran-3-carbonyl)piperidine
1-(2-chlorophenyl)-3-(1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-(3-methyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane