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3-(1-{1-[(2,4-difluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-1-(2-methoxyphenyl)urea
2-(6-methoxynaphthalen-2-yl)-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)morpholine
N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
4-{1-[5-(2,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}morpholine
2-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-6-methylpyridine-3-carbonitrile
1-{3-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-3-oxopropyl}-6-methyl-1,2-dihydropyridin-2-one
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperidin-4-yl}propanamide
2-amino-4-(2-butyl-1H-imidazol-4-yl)-6-(4-hydroxyphenyl)pyridine-3-carbonitrile
2-(1-oxo-1,2-dihydrophthalazin-2-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]acetamide
2-[4-(2-chloro-6-fluorobenzoyl)morpholin-3-yl]-1-(4-hydroxypiperidin-1-yl)ethan-1-one
{[3-(3-fluorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(1H-pyrazol-1-yl)ethyl]amine
N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
3-(3-chloro-1,2-oxazol-5-yl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(morpholin-4-yl)piperidin-1-yl]propan-1-one
N-{[2-(diethylamino)pyridin-3-yl]methyl}thiophene-3-sulfonamide
2,5-dimethyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[(1-cyclooctylpyrrolidin-3-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)acetamide
(1S,3R)-3-amino-N-(2-methoxyethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopentane-1-carboxamide
1-[2-(1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-(dimethylamino)-N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-2-(3-methylphenyl)acetamide
4-[2-(1H-pyrazol-1-yl)ethyl]-1-[5-(pyrrolidin-2-yl)thiophene-2-carbonyl]piperidine
5-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-1H-1,2,3-triazole
5-[1-(4-methylpentanoyl)piperidin-4-yl]-5-(pyridin-2-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
1-[(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-3-hydroxypiperidin-1-yl]-2-methoxyethan-1-one
5-(3-ethoxypropanoyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
5-methyl-4-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,3-oxazole
2-(4,5-dimethyl-1H-imidazol-1-yl)-1-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)ethan-1-one
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N,2-dimethyl-6-(piperidin-4-yl)pyrimidin-4-amine
(1R,3s,6r,8S)-4-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-azatricyclo[4.3.1.13,8]undecane
4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1-[2-(piperidin-1-yl)ethyl]-1,2,3,6-tetrahydropyridine
4-(3-fluorophenoxy)-1-{thieno[2,3-d]pyrimidin-4-yl}piperidine-4-carboxylic acid
N3-cyclooctyl-4-oxo-1-(oxolan-2-ylmethyl)-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N,2,5-trimethyl-N-(quinolin-5-ylmethyl)-1,3-oxazole-4-carboxamide
N-[(1S)-1-(4-chlorophenyl)ethyl]-2-methyl-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
4-(2-methoxyethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(2,4-difluorophenoxy)-N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]acetamide
1-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-[2-(1H-pyrrol-1-yl)ethyl]piperazine
1-(2-methoxyethyl)-8-methyl-3-(naphthalen-1-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4S)-4-amino-N-methyl-1-{3-[(4-methylphenyl)formamido]propanoyl}pyrrolidine-2-carboxamide
N-{1-[(3-{4-oxo-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}phenyl)methyl]pyrrolidin-3-yl}acetamide
1-[(3,5-dimethylphenyl)methyl]-4-[4-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
1-[4-(4-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)phenyl]ethan-1-one
1-[3-(hydroxymethyl)-3-[(2-methylphenyl)methyl]piperidin-1-yl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
[(1-cyclopentylpiperidin-4-yl)methyl][(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl](oxolan-2-ylmethyl)amine
3-methoxy-N-{[7-methoxy-2-(pyrrolidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-(4-methoxyphenyl)-4-{4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}butane-1,4-dione
2-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)quinolin-8-ol
[(3-methoxyphenyl)methyl](prop-2-en-1-yl){[3-(pyrimidin-2-yloxy)phenyl]methyl}amine
(3S,4S)-4-(4-fluoropiperidin-1-yl)-1-{[2-(thiophen-2-yl)pyrimidin-5-yl]methyl}pyrrolidin-3-ol
3-(4-fluorophenyl)-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
N-ethyl-1-methyl-3-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide