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1-[(1S,3R)-3-hydroxy-1-methoxy-1-methyl-7-azaspiro[3.5]nonan-7-yl]-2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
(3aR,6aR)-2-cyclobutanecarbonyl-5-(3-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-(2-hydroxyethyl)-8-[2-(2-methylphenoxy)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(oxolan-2-ylmethyl)-N-(thiophen-3-ylmethyl)acetamide
5-(4,4-difluoropiperidine-1-carbonyl)-2-(phenoxymethyl)pyrimidin-4-ol
1-{2-[2-(3-propanamidophenoxy)acetamido]ethyl}piperidine-3-carboxamide
1-{5-[3-(methoxymethyl)piperidine-1-carbonyl]pyridin-2-yl}-4-(2-methylpropyl)-1,4-diazepane
1-[(2-fluoro-5-methylphenyl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-2-(2-methoxyethyl)piperidine
(1R,5R)-6-[5-(methoxymethyl)furan-2-carbonyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-[5-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propanoic acid
N-[(1R,2S)-1-hydroxy-1-phenylpropan-2-yl]-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
5-[1-(4-methoxyphenyl)-3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]-1H-1,2,3-benzotriazole
N-(1-{[5-(piperidin-1-ylmethyl)thiophen-2-yl]methyl}pyrrolidin-3-yl)acetamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(1,2-oxazol-3-ylmethyl)piperidine-4-carboxylate
N-[(2S,4R,6S)-2-[2-(methoxymethyl)pyrimidin-5-yl]-6-(2-methylpropyl)oxan-4-yl]benzamide
1-(4-{4-[(4aS,8aS)-decahydroisoquinolin-2-ylmethyl]-1H-1,2,3-triazol-1-yl}piperidin-1-yl)ethan-1-one
N-{[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-(2-phenylethyl)benzamide
N-[(2,3-dimethylphenyl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
methyl({[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}){[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}amine
3-{[1-(1H-imidazol-2-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[(4-methyl-1H-imidazol-2-yl)methyl]benzamide
3-hydroxy-1-(2-methoxyethyl)-3-[({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)methyl]piperidin-2-one
6-[1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-3-yl]-2-ethyl-3,4-dihydropyrimidin-4-one
4-[6-(4-methanesulfonylphenyl)pyridazin-3-yl]thiomorpholine
7-[(4-fluorophenyl)methyl]-2-(1H-imidazol-2-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(1H-indol-1-yl)ethyl]-2-methanesulfonyl-N-methylacetamide
benzyl({[2-(cyclopentanesulfonyl)-1-(3-methoxypropyl)-1H-imidazol-5-yl]methyl})ethylamine
1-phenyl-4-[(2,3,4-trifluorophenyl)methyl]piperazin-2-one
ethyl 2-{[3-(4-phenylpiperazin-1-yl)piperidine-1-carbonyl]amino}acetate
1-ethyl-N-[2-(furan-2-yl)ethyl]-5-oxopyrrolidine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-[(5-fluoro-2-methylphenyl)methyl]piperazine
1-{3-[(4-methoxyphenyl)amino]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
3-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-(7-methanesulfonyl-4-methylquinazolin-2-yl)pyrrolidine-2-carboxamide
3-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
3-[4-(3-cyclohexyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]phenol
1-(2,1,3-benzothiadiazol-4-yl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-(1-benzylpiperidin-3-yl)-2-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-methoxy-1-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
1-[1-(5-ethylpyrimidin-2-yl)piperidin-4-yl]-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[3-(3,3-diphenylpiperidin-1-yl)-3-oxopropyl]acetamide
ethyl 4-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)carbamoyl]piperazine-1-carboxylate
[3-(1H-imidazol-1-yl)propyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3-methanesulfonylpropanamide
2-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrazine
1-[1-(hydroxymethyl)cyclopropanecarbonyl]-4-{thieno[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol