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N-cyclohexyl-N,7-dimethylimidazo[1,2-a]pyridine-2-carboxamide
N-(3-{2-azatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}propyl)-N-methylmorpholine-2-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2-propyl-1H-1,3-benzodiazol-1-yl)propanamide
(2S,4S)-4-amino-N,N-diethyl-1-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]pyrrolidine-2-carboxamide
N-cyclopropyl-2-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]propanamide
8-(1-benzothiophen-2-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(pyridin-2-yl)thiophen-2-yl]methyl}pyrazolo[1,5-a]pyridine-7-carboxamide
2-[({2-[(dimethylamino)methyl]phenyl}methyl)(methyl)amino]-2-(2-methoxy-5-methylphenyl)acetic acid
2-({2-[1-(benzenesulfonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N3-cyclooctyl-N5-(furan-2-ylmethyl)-4-oxo-1-(oxolan-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
4-oxo-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(4-methyl-1-propyl-1H-pyrazol-5-yl)-2-[4-(2-methyl-5-propylpyrimidin-4-yl)-1H-pyrazol-1-yl]acetamide
1-[(3R,4S)-3-amino-4-phenylpyrrolidin-1-yl]-3-(1H-1,2,3-benzotriazol-1-yl)propan-1-one
N-[2-(2-amino-1,3-thiazol-4-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
(2S,4S,5R)-4-(tert-butylcarbamoyl)-2-ethyl-5-(4-methoxyphenyl)-1-methylpyrrolidine-2-carboxylic acid
5-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-2-phenylpyrimidine
1-methyl-5-{3-[(1-propylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1H-1,2,3-benzotriazole
N-{[2-(4-acetylpiperazin-1-yl)pyridin-3-yl]methyl}-5-methylthiophene-2-carboxamide
N-[(3R,4R)-3-hydroxy-1-(6-methyl-4-oxo-4H-pyran-2-carbonyl)piperidin-4-yl]pyridine-3-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
4-(1H-pyrazol-4-yl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}butan-1-one
4-{[3-(3-methoxyphenoxy)azetidin-1-yl]methyl}-5-methyl-2-(thiophen-2-yl)-1,3-oxazole
(1R,9S)-5-amino-13-methyl-3-(1-methyl-1H-pyrazol-4-yl)-6,13-diazatricyclo[7.3.1.02,7]trideca-2,4,6-triene-4-carbonitrile
N-cyclopropyl-1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}piperidine-4-carboxamide
(1S,5R)-6-[4-(2-methoxyphenyl)benzoyl]-3-methyl-3,6-diazabicyclo[3.2.2]nonane
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[2-(pyridine-2-sulfonyl)ethyl]amine
methyl({2-[(4-methylpyrimidin-2-yl)oxy]hex-5-en-1-yl})(pyridin-3-ylmethyl)amine
6-(2-chlorophenyl)-2-[(3S)-3-hydroxypyrrolidine-1-carbonyl]-7-methyl-7H,8H-imidazo[1,2-a]pyrazin-8-one
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[(1-methyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]acetamide
N-[2-(furan-2-yl)-2-(pyrrolidin-1-yl)ethyl]-6-methylimidazo[2,1-b][1,3]thiazole-5-carboxamide
N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
methyl({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
2-(1H-pyrazol-1-yl)-N-[2-(4-sulfamoylphenyl)ethyl]benzamide
3-(5-methyl-1H-pyrazol-1-yl)-1-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
N-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyl-1,2,3,4-tetrahydronaphthalen-1-amine
methyl (2S)-2-{[6-(3-fluorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-3-methylbutanoate
3-{2-[3-(2-chlorophenoxy)azetidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(2-hydroxyethyl)-1H-1,2,4-triazol-3-yl]benzamide
6-methyl-2-(3-{[3-(1H-pyrazol-1-yl)azetidin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
(4aR,8aR)-2-(5-methyl-1,2-oxazole-3-carbonyl)-7-(pyrrolidine-1-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
ethyl 5-(3,5-dimethyl-1H-pyrrole-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-({2-[2-hydroxy-3-(morpholin-4-yl)propoxy]-3-methoxyphenyl}methyl)piperazin-2-one
1-(3,5-dimethylphenyl)-4-[5-(methoxymethyl)furan-2-carbonyl]piperazin-2-one
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)piperidine-4-carboxamide
1-[benzyl(methyl)amino]-3-{4-[(cyclohexylamino)methyl]phenoxy}propan-2-ol
4-ethyl-1-methyl-3-[1-(5-propylthiophene-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(5-ethyl-2-methylpyrimidin-4-yl)-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-amine
5-methoxy-9-(6-methoxy-1-methyl-1H-indole-2-carbonyl)-1-oxa-9-azaspiro[5.5]undecane
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carboxamide