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2-[2-(1H-imidazol-4-yl)ethyl]-8-(pent-4-enoyl)-2,8-diazaspiro[5.5]undecan-3-one
7-{1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
2-[4-(oxolane-2-carbonyl)-1,4-diazepan-1-yl]-N,N-bis(prop-2-en-1-yl)acetamide
1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
1-[4-(2-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(4H-1,2,4-triazol-4-yl)propan-1-one
3-[({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)(methyl)amino]-2,2-dimethylpropan-1-ol
2-(1-ethylpiperidin-4-yl)-N-[2-(2-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]acetamide
4-(2,6-dimethoxypyridine-3-carbonyl)-6-[(2-fluorophenyl)methoxy]-1-(2-methylpropyl)-1,4-diazepan-2-one
N-(furan-2-ylmethyl)-2-(1H-imidazol-2-yl)-N-(thiophen-2-ylmethyl)benzamide
4-{[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
1-{[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
2-{4-[(1-ethyl-1H-indol-3-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
N-[2-hydroxy-2-(3-hydroxyphenyl)ethyl]-2,6,8-trimethylquinoline-4-carboxamide
1-cyclobutanecarbonyl-4-(piperidin-4-yl)-1,4-diazepane
1-methyl-4-[5-(1-methyl-3-propyl-1H-pyrazol-5-yl)-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-1-yl]piperidine
4-[(2-fluorophenyl)methyl]-1-[(5-methyl-1,2-oxazol-3-yl)methyl]piperidine
3-methyl-4-{4-[1-(morpholin-4-yl)ethyl]phenyl}benzoic acid
{[4-chloro-2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}({1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
2-{4-[3-(1,2,3,6-tetrahydropyridine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
4-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-3,4-dihydro-2H-1,4-benzothiazin-3-one
6-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)-3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
6-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-2,3,4,5-tetrahydropyridazin-3-one
2-(dimethylamino)-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(3-methylphenyl)acetamide
(2R,6S)-4-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,6-dimethylmorpholine
N-[2-(2,6-dimethoxyphenyl)phenyl]-2-methylpropanamide
N-{[1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-3-yl]methyl}acetamide
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-3-{[(3-hydroxypropyl)(methyl)amino]methyl}piperidin-2-one
2-[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]pyridine-3-carboxamide
1-(5-methyl-1,2-oxazole-3-carbonyl)-4-[(4-phenyl-1H-1,2,3-triazol-1-yl)methyl]piperidine
3-[(4-benzoylpiperidin-1-yl)methyl]pyrrolidin-3-ol
2-ethyl-5-({4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)pyrimidine
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,3S,5S)-3-(4-methoxyphenyl)-8-[(6-methylpyridin-2-yl)methyl]-8-azabicyclo[3.2.1]octane
N-[2-(dimethylamino)ethyl]-N-[(2-methylphenyl)methyl]-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-3-(methylsulfanyl)propan-1-one
N-cyclopentyl-4-{[(3S,4R)-4-ethoxyoxolan-3-yl]sulfamoyl}benzamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(dimethylamino)azepan-1-yl]propan-1-one
8-[3-(dimethylamino)pyrazin-2-yl]-2-(3-methoxypropyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
1-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(methylamino)ethan-1-one
4-methyl-1-{[2-(trifluoromethoxy)phenyl]methyl}piperidine-4-carbonitrile
N5-tert-butyl-N2-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2,5-dicarboxamide
1-{[2-(3,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(4-methoxybenzoyl)piperazine
[(1,3-dimethylpyrrolidin-3-yl)methyl]({[4-(1H-imidazol-1-yl)phenyl]methyl})methylamine
N,5-dimethyl-N-[3-(oxolan-2-yl)propyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(4-methyl-1H-pyrazol-1-yl)-1-(1-propyl-1H-pyrazole-5-carbonyl)piperidine-4-carboxylic acid
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(thiophen-2-yl)acetamide
[(3R,4S)-1-{[3-(furan-2-yl)phenyl]methyl}-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(1H-pyrrole-2-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-(furan-2-ylmethyl)-N-{[2-(4-hydroxypiperidin-1-yl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-4-methoxybenzamide