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5-butyl-1'-(5-methylthiophene-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-benzyl-N-butyl-1-[1,3-dioxo-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
2-methyl-N-[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]thieno[3,2-d]pyrimidin-4-amine
(2S,4R)-4-benzamido-N,N-diethyl-1-(3-hydroxypropanoyl)pyrrolidine-2-carboxamide
4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]benzamide
2-[({1-[3-(furan-2-yl)benzoyl]piperidin-3-yl}oxy)methyl]pyridine
N-[(5-chloro-2,3-dimethoxyphenyl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
(2S,4S)-4-[2-(2,4-dichlorophenoxy)acetamido]pyrrolidine-2-carboxylic acid
N,4-dimethyl-N-{[1-(propan-2-yl)piperidin-3-yl]methyl}-1,3-thiazol-2-amine
5-({4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidin-1-yl}methyl)-2-(propylsulfanyl)pyrimidine
1-[1-(1-benzoxepine-4-carbonyl)pyrrolidin-3-yl]-3,5-dimethyl-1H-pyrazole
6-cyano-N-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}pyridine-3-carboxamide
5-ethyl-N-[4-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-1,3-oxazole-4-carboxamide
1-{4-[2-(3-phenylpropyl)morpholine-4-carbonyl]piperidin-1-yl}ethan-1-one
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-fluoro-3-(trifluoromethyl)benzamide
4-[2-(3-methoxyphenyl)ethyl]-11-[(2-phenylethyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[({[1-(hydroxymethyl)cyclobutyl]methyl}carbamoyl)amino]-N-(2-methoxyethyl)benzamide
methyl[(2-methyl-1H-imidazol-4-yl)methyl][(2-phenyl-1,3-thiazol-4-yl)methyl]amine
N-[(5-ethylpyridin-2-yl)methyl]-3-(3-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
1-[(3-methoxyphenyl)methyl]-4-[2-(methylamino)pyridine-4-carbonyl]piperazin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-{imidazo[1,2-a]pyridin-2-yl}propanamide
N-{2-[3-(2-ethyl-1H-imidazol-1-yl)propanamido]-5-methoxyphenyl}-2-methylpropanamide
N-(prop-2-en-1-yl)-N-(propan-2-yl)-1,2,3,4-tetrahydronaphthalene-2-carboxamide
4-ethyl-3-[1-(isoquinoline-5-carbonyl)piperidin-3-yl]-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1,3-dimethylpyrrolidin-3-yl)methyl]-5-[(isoquinolin-5-yloxy)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N,N-dimethyl-7-(4-methylnaphthalene-1-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
3-(3-{[4-(pyrimidin-2-yloxy)piperidin-1-yl]methyl}-1H-indol-1-yl)propanamide
5-chloro-N-[2-(3-{[(furan-3-ylmethyl)(methyl)amino]methyl}phenoxy)propyl]-3-methyl-1H-indole-2-carboxamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-[1-(2-methoxyethyl)-3-(3-methoxyphenyl)-2,5-dioxopyrrolidin-3-yl]-N-methylacetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(pyridine-4-carbonyl)piperazin-2-one
[(3-fluoro-2-methylphenyl)methyl]({[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl})methylamine
methyl({[4-(5-methylpyridin-2-yl)piperidin-4-yl]methyl}){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
9-(2,5-dimethylfuran-3-carbonyl)-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(4S)-4-hydroxy-4-(methoxymethyl)-3,3-dimethylpiperidin-1-yl]-2-{[(2-methylphenyl)methyl]sulfanyl}ethan-1-one
4-[(4-fluorophenyl)methyl]-11-{[2-(pyridin-3-yl)ethyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-{5-[(2S)-1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]pyrrolidin-2-yl]-1,2,4-oxadiazol-3-yl}pyridine
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
[1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-3-(2-methoxyethyl)piperidin-3-yl]methanol
5-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-5-oxopentanamide
5-(azepane-1-carbonyl)-1-(butan-2-yl)-4-oxo-N-{[3-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-(5-methylhexan-2-yl)-5-{[2-(propan-2-yl)-1H-imidazol-1-yl]methyl}-1H-pyrazole-3-carboxamide
2-ethoxy-1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
1-benzyl-4-(furan-3-carbonyl)-1,4-diazepan-6-ol
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-[2-(pyridin-2-yl)pyrrolidin-1-yl]pyridine-3-carboxamide
6-methyl-9-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]-9H-purine
N-[(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
{1-[3-(5-methylfuran-2-yl)benzoyl]piperidin-2-yl}methanamine
N-ethyl-2-{4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperazin-1-yl}acetamide
N-[(1-cyclopropyl-5-oxopyrrolidin-3-yl)methyl]-3-{4-[2-(3-methylphenyl)acetamido]-1H-pyrazol-1-yl}benzamide
1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(morpholin-4-yl)ethan-1-one