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4-(1-methyl-3-propyl-1H-pyrazole-5-amido)oxane-4-carboxylic acid
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydro-1H-inden-2-yl)-1,3-oxazole-4-carboxamide
1-methyl-N-[3-(5-methyl-4-{[3-(4-methyl-1,3-thiazol-5-yl)propanamido]methyl}-1,3-oxazol-2-yl)phenyl]piperidine-3-carboxamide
ethyl 4-{4-cyclopropyl-5-[(dimethylamino)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
3-[4-(3-chlorophenyl)-3-oxopiperazine-1-carbonyl]benzonitrile
N-ethyl-6-(4-methoxypiperidin-1-yl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-[(3,4-dimethylphenyl)methyl]-4-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}piperazin-2-one
(4aS,8aS)-4a-hydroxy-N-[2-(methylsulfanyl)phenyl]-decahydroisoquinoline-2-carboxamide
N-[(3S,4R)-1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]-4-propylpyrrolidin-3-yl]methanesulfonamide
4-[(2-{[(3S)-3-fluoropyrrolidin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)methyl]-2,1,3-benzoxadiazole
1-[4-(4-hydroxypiperidin-1-yl)piperidin-1-yl]-4-(2-methyl-1H-imidazol-1-yl)butan-1-one
4-({1-[3-(2-methylphenyl)benzoyl]piperidin-4-yl}methyl)morpholine
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
3-methoxy-N-[1-methyl-2-phenyl-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]propanamide
methyl 3-[(2E)-3-(3-fluorophenyl)prop-2-enamido]-6-(pyrrolidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N-cyclopropyl-N-(1-{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)pyridine-2-carboxamide
N-(furan-2-ylmethyl)-N,5-dimethyl-4-{[2-(morpholin-4-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
6-[(dimethyl-1,2-oxazol-4-yl)methoxy]-1-(2-methylpropyl)-4-{[4-(pyrimidin-2-yloxy)phenyl]methyl}-1,4-diazepan-2-one
N-tert-butyl-5-[3-(diethylamino)pyrrolidine-1-carbonyl]-1-(3-methylbutyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N-methyl-2-(1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
4-[(2-chlorophenyl)methyl]-1-(3,6-dimethylpyrazin-2-yl)piperidine-4-carboxylic acid
1-[4-(4-{[methyl(1-methylpiperidin-4-yl)amino]methyl}phenoxy)piperidin-1-yl]-2-(thiophen-3-yl)ethan-1-one
N-[3-(3-ethylphenoxy)propyl]-N,1-dimethyl-6-oxo-1,6-dihydropyridine-3-carboxamide
ethyl[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl][(6-methylpyridin-2-yl)methyl]amine
3-({methyl[1-(pyrazin-2-yl)propan-2-yl]amino}methyl)pyridin-2-amine
N-[(2-fluorophenyl)methyl]-N-(2-hydroxyethyl)-1-methyl-1H-1,3-benzodiazole-5-carboxamide
4-[4-(hydroxymethyl)benzoyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2R,3R)-3-(1,4-oxazepan-4-yl)-1'-(pyridin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[1-(2,7,8-trimethylquinoline-4-carbonyl)piperidin-2-yl]ethan-1-ol
6-{1-[(4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-2-(6-methylpyridin-3-yl)-3,4-dihydropyrimidin-4-one
N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-ethyl-5-methoxy-1-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-1H-indole-2-carboxamide
1-(cyclohexylmethyl)-N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
1-{4-[5-(azepan-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-ethoxyethan-1-one
5-[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]pyridin-2-amine
1-[(1S,5R)-6-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl}){[3-(1H-pyrazol-1-yl)phenyl]methyl}amine
5-(2-methoxy-5-methylphenoxymethyl)-3-(phenoxymethyl)-1,2,4-oxadiazole
N-[(3-chloro-2-methylphenyl)methyl]-2-(2-oxopiperidin-1-yl)acetamide
ethyl 4-(oxan-2-ylmethyl)-1-{[2-(trifluoromethyl)phenyl]carbamoyl}piperidine-4-carboxylate
7-{2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidine-6-carbonyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-2,6,8-trimethylquinoline
1-(4-ethylphenyl)-3-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)urea
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(thiolan-3-yl)pyridin-2-amine
N-methyl-4-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}-1,3-thiazol-2-amine
N-(1-ethyl-1H-pyrazol-5-yl)-5-[1-(furan-3-ylmethyl)pyrrolidin-2-yl]thiophene-2-carboxamide
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
2-methyl-8-{6-methylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-(pyridin-2-ylmethyl)-4-[4-(pyridin-3-yl)piperazine-1-carbonyl]pyrrolidin-2-one
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N,5-dimethyl-1H-pyrazole-3-carboxamide