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2-(propan-2-yl)-9-[2-(pyrrolidin-1-yl)benzoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2,6-dimethylphenoxy)pyridin-3-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
N-[(1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidin-3-yl)methyl]thiophene-2-sulfonamide
N-[3-(1H-1,2,3-benzotriazol-1-yl)propyl]-8-chloroquinoline-2-carboxamide
5-[2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl]-1,2-oxazole
2-tert-butyl-6-(2-fluoro-6-methoxybenzoyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
1-(benzenesulfonyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine
(4aS,7aR)-1-(pyrazine-2-carbonyl)-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2,6-dimethylphenyl)-2-(3-acetamidopropanamido)benzamide
2-methyl-2-[(4-methylphenyl)amino]-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}propanamide
methyl 5-[(1-acetylpiperidin-4-yl)amino]-3-(furan-3-amido)-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
[1-(3,6-dimethylpyrazin-2-yl)-4-(2-phenylethyl)piperidin-4-yl]methanol
2-{[ethyl(oxan-4-ylmethyl)amino]methyl}benzonitrile
N-[(3-chlorophenyl)methyl]-3-[1-(thiophene-2-carbonyl)piperidin-4-yl]propanamide
5-ethyl-2,3-dimethyl-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-[4-(3-hydroxyphenyl)piperazine-1-carbonyl]-1H-imidazole-4-carboxylic acid
N,1-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}azepane-2-carboxamide
N-benzyl-N-ethyl-1-{2-[(4-methyl-1,3-thiazol-2-yl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}piperidine-3-carboxamide
5-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
1-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-[1-(propan-2-yl)-1H-pyrazol-4-yl]urea
1-[1-(methoxymethyl)cyclopropanecarbonyl]-3-phenylpiperazine
(1s,4s)-4-{4-[2-(4-methylpentyl)morpholine-4-carbonyl]-1H-1,2,3-triazol-1-yl}cyclohexan-1-amine
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1,2-oxazol-3-ylmethyl)piperidine-3-carboxamide
4-({4-[2-(1,3-thiazol-2-yl)pyrrolidine-1-carbonyl]furan-2-yl}methyl)morpholine
N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-3,4-dihydro-2H-1-benzopyran-3-amine
methyl 4-[4-(2-methyl-1,3-thiazole-5-carbonyl)piperazin-1-yl]benzoate
4-{1-[1-(4-methylpyridine-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
N-methyl-2-[methyl(pyridin-3-ylmethyl)amino]-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]acetamide
1-(2-methylpropyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
2-[5-(1-methyl-2-oxo-1,2-dihydropyridin-4-yl)-1-[(2-methylphenyl)methyl]-1H-1,2,4-triazol-3-yl]acetamide
[(1-butyl-2-cyclobutylmethanesulfonyl-1H-imidazol-5-yl)methyl](methyl)[2-(pyridin-2-yl)ethyl]amine
1-{[1-(8-chloroquinolin-2-yl)piperidin-4-yl]methyl}pyrrolidin-2-one
7-fluoro-3-methyl-2-[3-(propan-2-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazol-6-yl]-1H-indole
(3S,4R)-4-(3-methoxyphenyl)-1-[(2,3,4-trifluorophenyl)methyl]pyrrolidine-3-carboxylic acid
1-{1-[(5-hydroxy-2-methoxyphenyl)methyl]piperidin-4-yl}pyrrolidin-2-one
2-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-N-[(2-methoxyphenyl)methyl]acetamide
2-(4-ethylpiperazin-1-yl)-N-[(4-methoxyphenyl)methyl]-N-(2-methylpropyl)acetamide
8-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{[3-(azepane-1-carbonyl)-1H-pyrazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
3-(4-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperazin-1-yl)benzonitrile
methyl 2-[3-(2-methylphenyl)-3-phenylpropanamido]acetate
1-[(3-methoxyphenyl)methyl]-6-oxo-N-[(4-phenyloxan-4-yl)methyl]piperidine-3-carboxamide
N-[2-(4-fluorophenyl)ethyl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide
1-(2,2-dimethylpropyl)-3-hydroxy-3-({methyl[(5-methyl-1H-pyrazol-3-yl)methyl]amino}methyl)piperidin-2-one
2-methyl-5-({2-[3-(trifluoromethyl)phenyl]-1H-imidazol-1-yl}methyl)pyrazine
1-(4-tert-butylphenyl)-4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
({2-[(dimethylamino)methyl]phenyl}methyl)(1H-imidazol-2-ylmethyl)methylamine
4-(4-methoxybutyl)-N-[4-(3-methyl-1,2,4-oxadiazol-5-yl)phenyl]piperazine-1-carboxamide
N3-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-1,3-dicarboxamide
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-hydroxy-4-methylbenzamide