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N-(1-methoxybutan-2-yl)-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
4'-methyl-1-(2-methylpentanoyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(1S,9S)-11-[6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-yl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3,3-dimethyl-4-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]acetyl}piperazin-2-one
1-(4,4-difluoropiperidin-1-yl)-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
N3-benzyl-N3-(2-hydroxyethyl)-N5-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[4-(1H-pyrazol-4-yl)butanoyl]-decahydro-1,6-naphthyridin-2-one
4-[(2-aminopyridin-3-yl)methyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
N-{imidazo[1,2-a]pyridin-2-ylmethyl}-2-(morpholin-3-yl)acetamide
2-methoxy-5-{4-[4-(2-methylpropyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carbonyl}pyrimidine
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4,5,6,7-tetrahydro-1,3-benzothiazole-2-carboxamide
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-(4-methoxypyrimidin-2-yl)-decahydro-1,6-naphthyridin-2-one
1-(4-phenylazepan-1-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propan-1-one
4-{3-[2-(3-fluorophenyl)ethyl]piperidine-1-carbonyl}-1-(propan-2-yl)piperidine
N-benzyl-N-ethyl-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyridine-2-carboxamide
1-[(3-phenyloxolan-3-yl)methyl]-4-(pyrrolidine-1-carbonyl)piperidine
3-cyclohexyl-4-[2-(furan-2-yl)pyrrolidine-1-carbonyl]-1H-pyrazole
1-ethyl-N-[(4-methylphenyl)methyl]-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-amino-4-(2-methoxypyrimidin-5-yl)-8-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
2-cyclopropyl-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
6-{4-[4-(2-methoxyethyl)phenoxymethyl]phenyl}pyrimidin-4-amine
N-(4-chloro-3-methylphenyl)-2-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]amino}acetamide
2-(dimethylamino)-4-methyl-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
N-[(3R,4S)-4-cyclopropyl-1-(2-{[(2-fluorophenyl)methyl](methyl)amino}acetyl)pyrrolidin-3-yl]acetamide
N-benzyl-N-methyl-3-(1-phenylmethanesulfonylpiperidin-4-yl)propanamide
N-[2-(6-methylpyridin-2-yl)ethyl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
5-{[3-oxo-4-(2-phenylphenyl)piperazin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(4-methyl-1H-imidazole-2-carbonyl)-4-(4-methyl-1H-pyrazol-3-yl)piperidine
1,9-dimethyl-4-(2,5,7-trimethylquinoline-4-carbonyl)-1,4,9-triazaspiro[5.5]undecane
2-[4-(2-aminopyrimidin-4-yl)-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl]ethan-1-ol
5-[3-chloro-5-methoxy-4-(pyrrolidin-1-ylmethyl)phenoxy]-1-azabicyclo[3.2.1]octane
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-methyl-1,3-oxazole-5-carboxamide
5-(2-{[(3-methoxyphenyl)methyl]amino}ethyl)-1-[2-(piperidin-1-yl)ethyl]pyrrolidin-2-one
2-{1-cyclopentyl-4-[(3-methylquinoxalin-2-yl)methyl]piperazin-2-yl}ethan-1-ol
7-(2-hydroxy-5-methoxybenzoyl)-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-[3-(1,2-oxazolidin-2-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
[5-({[2-(2,4-dimethylphenoxy)ethyl](methyl)amino}methyl)furan-2-yl]methanol
2-(4-{[3-(2-hydroxyethyl)-4-[(5-methylfuran-2-yl)methyl]piperazin-1-yl]methyl}phenoxy)ethan-1-ol
(2R,3R,6R)-3-phenyl-5-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-benzyl-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-3-(2-phenoxyethyl)piperidin-3-yl}methanol
2-{[4-(3-acetylphenyl)-5-(pyridin-3-ylmethyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
N-{[2-(2-benzamidophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-methyl-5,6-dihydro-1,4-dioxine-2-carboxamide
(2S)-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-5-oxopyrrolidine-2-carboxamide
4-(4-methoxy-3-methylphenyl)-6-methyl-N-(oxan-4-yl)-2-oxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{1-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
N-(2-methoxy-5-{[1,3]oxazolo[4,5-b]pyridin-2-yl}phenyl)-2-(1H-pyrazol-1-yl)butanamide
4-[1-(2-{[(4-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-3-yl]benzoic acid
2-(5-{1-[(4-methylphenyl)sulfanyl]ethyl}-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-1-yl)ethan-1-ol