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(benzylsulfamoyl)({[2-(1H-1,2,4-triazol-1-yl)pyridin-3-yl]methyl})amine
1-(cyclohexylmethyl)-5-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]piperidin-2-one
N-{[6,7-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-4-(1H-pyrazol-1-yl)benzamide
6-[2,6-dimethyl-4-(piperidin-1-ylmethyl)phenoxy]pyridine-3-carbonitrile
1-[(3-fluorophenyl)methyl]-4-(oxolan-3-ylmethyl)piperazine
4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3-(4-methoxyphenyl)-1H-pyrazole
1-({[2-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]carbamoyl}methyl)piperidine-4-carboxamide
methyl[3-(1H-pyrazol-1-yl)propyl](pyridin-2-ylmethyl)amine
1-{2-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-5-methoxybenzoyl}-3-methoxypiperidine
N-[3-(4-fluorophenyl)phenyl]-1-(6-methylpyridine-2-carbonyl)piperidine-3-carboxamide
3-benzyl-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidine-3-carboxylic acid
2-(3-phenylpropyl)-N-[1-(pyrimidin-4-yl)ethyl]-1,3-benzoxazole-5-carboxamide
2-[3-(1H-imidazol-1-yl)propyl]-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-oxo-2,3-dihydro-1H-isoindole-5-carboxamide
N,N-diethyl-1-({1-[(2E)-3-(thiophen-2-yl)prop-2-enoyl]piperidin-3-yl}methyl)-1H-1,2,3-triazole-4-carboxamide
2-{[6-(2-chlorophenyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}-N-propylacetamide
(3R,4R)-4-[4-(2-phenylethyl)piperazin-1-yl]-1-(pyrazin-2-yl)piperidin-3-ol
N-ethyl-1-[(4-fluoro-2-methoxyphenyl)methyl]-N-(pyridin-4-ylmethyl)piperidin-3-amine
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(5-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)acetamide
6-[3-(1-methyl-5-oxo-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]-2,3-dihydropyridazin-3-one
3-(3-fluoro-4-methoxybenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
{[2-(3-methylphenyl)pyrimidin-5-yl]methyl}[(5-phenyl-1H-pyrazol-3-yl)methyl]amine
1'-(3-fluorobenzoyl)-5-(3-methylbut-2-en-1-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-({3-[2-(3,4-difluorophenyl)ethyl]piperidin-1-yl}methyl)-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-7-one
2-[1-(2,2-dimethylpropyl)-4-(oxan-4-yl)piperazin-2-yl]ethan-1-ol
N,2,5-trimethyl-N-[1-(1,2-oxazol-3-yl)ethyl]furan-3-carboxamide
N-[furan-2-yl(phenyl)methyl]-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
(1S,5R)-3-(5-acetyl-4-methylpyrimidin-2-yl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-[2-(pyridin-2-yl)ethyl]propanamide
(3aS,6aR)-5-(3-methylfuran-2-carbonyl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-phenylpyrrolidin-3-yl]cyclobutanecarboxamide
1-{2,7-diazaspiro[4.5]decan-2-yl}-3-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]propan-1-one
3-(3-fluorophenyl)-4-{[5-methyl-2-(5-methylfuran-2-yl)-1,3-oxazol-4-yl]methyl}piperazin-2-one
2-benzyl-8-[2-(1H-pyrazol-1-ylmethyl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-3-(methylsulfanyl)propanamide
N,N-dimethyl-5-[3-(thiophene-2-carbonyl)piperidine-1-carbonyl]pyridin-2-amine
1-[9-(but-3-yn-1-yloxy)-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
1-cyclohexyl-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]piperidine-3-carboxamide
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-(pyrrolidin-1-yl)piperidine
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-5-(oxolan-2-yl)thiophene-2-carboxamide
1-phenyl-N-{[1-(3-phenylprop-2-ynoyl)piperidin-3-yl]methyl}methanesulfonamide
1-{2-[2-(cyclopropylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]-2-oxoethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
9-(1H-imidazol-2-ylmethyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
N-[1-(1,3-benzothiazol-2-yl)piperidin-3-yl]-2-(pyrimidin-2-ylsulfanyl)acetamide
N-(2,2-difluoroethyl)-1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carboxamide
2-(4-{imidazo[1,2-a]pyridine-6-carbonyl}piperazin-1-yl)ethan-1-ol
4-(4-fluorophenoxy)-1-[(2S)-pyrrolidine-2-carbonyl]piperidine-4-carboxylic acid
2,6-dimethyl-4-{[(propan-2-yl)[(trimethyl-1H-pyrazol-4-yl)methyl]amino]methyl}phenyl acetate
1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(trifluoromethyl)-1,2-dihydropyridin-2-one
(3aR,5S,6S,7aS)-2-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-octahydro-1H-isoindole-5,6-diol