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2-ethyl-4-(4-methyl-1,3-thiazole-5-carbonyl)-1-(propan-2-yl)piperazine
N-[1-(2-phenylethyl)piperidin-3-yl]pyrazine-2-carboxamide
(2R)-2-amino-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-phenylacetamide
N-(2-{7-[(2-fluoro-5-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)cyclobutanecarboxamide
3-{1-[(4-acetamidophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)propanamide
2-[5-(5-chloropyrimidin-2-yl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
N-methyl-2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}acetamide
5-{4-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-1H-1,2,3,4-tetrazole
3-[cyclopropyl(1-methyl-1H-1,2,4-triazol-5-yl)methyl]-1-(2-fluoro-5-methanesulfonamidophenyl)urea
1-(4-methoxyphenyl)-4-[1-(3-methylthiophene-2-carbonyl)piperidin-3-yl]piperazine
1-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-(pyridin-3-yl)propan-1-one
[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]({[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl})amine
2-(2-chlorophenyl)-N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-3-methyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[2-(benzyloxy)ethyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-cyclopropyl-1-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
N-[(2-chloro-6-fluorophenyl)methyl]-2-(1H-imidazol-2-yl)benzamide
9-{[4-(2-methylphenyl)phenyl]methyl}-1,4,9-triazaspiro[5.5]undecan-5-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(pyridin-2-yl)pyrimidin-2-amine
(1R,4S)-N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-1,7,7-trimethyl-3-oxo-2-oxabicyclo[2.2.1]heptane-4-carboxamide
N-[2-({[4-(butan-2-yloxy)-3-chlorophenyl]methyl}amino)ethyl]acetamide
N-{1-[1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-phenylacetamide
N-ethyl-1-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}pyrrolidine-3-carboxamide
(1R,2R,4R)-N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
N-ethyl-4-({[(1-ethyl-1H-imidazol-2-yl)methyl](methyl)carbamoyl}amino)-3-methylbenzamide
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]-N-methyl-4-propylpyrimidine-5-carboxamide
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-2-(quinazolin-4-yloxy)acetamide
2-[4-(1-tert-butyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]-N,N-dimethylacetamide
3-(benzyloxy)-1-{[2-(2-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
2-methoxy-1-{1'-[2-(2-methyl-1H-imidazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
7,7-dimethyl-2-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-[1-(6-methylpyridin-2-yl)propan-2-yl]propanamide
2-benzyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1,3-thiazole-4-carboxamide
9-(4,6-dimethylpyrimidin-2-yl)-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
(1R,3S,5S)-8-[3-(piperidin-4-ylmethyl)benzoyl]-8-azabicyclo[3.2.1]octan-3-ol
N-({1-[(2,5-dimethylthiophen-3-yl)sulfonyl]piperidin-3-yl}methyl)-1H-indole-2-carboxamide
N-[1-(2-phenylethyl)piperidin-4-yl]pyrimidin-4-amine
ethyl 2-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-2-yl)acetate
5-{4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-2-methylpyrimidine
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methoxybenzoyl)piperazine
N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-{4-[(1S,2S)-2-hydroxycyclohexyl]piperazin-1-yl}propan-1-one
N-[5-(dimethylamino)pentyl]-6-(propan-2-yl)pyrimidin-4-amine
5-(2-fluoro-3-methylphenyl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(3-fluoro-4-hydroxyphenyl)ethan-1-one
2-{[cyclopropyl(4-methylpyridin-2-yl)methyl]amino}propane-1,3-diol
N-[(2S,3S)-1-hydroxy-3-methylpentan-2-yl]-3-(pyridin-4-yl)propanamide
2-[(4-acetyl-1,4-diazepan-1-yl)sulfonyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-methyl-8-(2-propylpyridine-4-carbonyl)-2,8-diazaspiro[4.5]decane