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(4aR,7aS)-1-benzyl-4-(1,2,4-oxadiazol-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[(2S,4S)-1-[2-(dimethylamino)-4-methylpyrimidine-5-carbonyl]-4-fluoropyrrolidin-2-yl]methyl}ethane-1-sulfonamide
3-cyclopropyl-5-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazole
N2-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}-N4-methyl-5H,6H,7H-cyclopenta[d]pyrimidine-2,4-diamine
1-[3-(aminomethyl)phenyl]-3-(2-propoxypropyl)urea
1-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(morpholin-4-yl)butan-1-one
N-cyclopropyl-N-ethyl-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)-1,3-oxazole-4-carboxamide
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-{octahydropyrrolo[1,2-a]piperazin-2-yl}ethan-1-one
1-(2-chloro-6-methylphenyl)-3-{[1-(hydroxymethyl)cyclobutyl]methyl}-3-methylurea
2-(1H-indol-4-yl)pyridin-4-amine
1-(4-benzylpiperidin-1-yl)-3-{1-[3-(pyridin-4-yl)propanoyl]piperidin-4-yl}propan-1-one
2-methyl-5-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1,4-dihydropyridin-4-one
methyl 2-[8-(1H-indol-2-ylmethyl)-2,4-dioxo-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
N-cyclopropyl-1-[(1s,4s)-4-(3-cyclopentylpropanamido)cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(4aS,7aR)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(3S,4S)-1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-methylpiperidine-3,4-diol
2-(1H-imidazol-2-yl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]benzamide
ethyl 5-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
2-{4-[2-(4-chloro-2-methylphenoxy)ethyl]piperazine-1-carbonyl}morpholine
3-{[1-(2,4-dimethylphenyl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
5-phenyl-N-(quinolin-4-ylmethyl)pyrazolo[1,5-a]pyrimidin-7-amine
(2R,6R)-4-(5-ethyl-2-methylpyrimidin-4-yl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
(2E)-3-(2-chlorophenyl)-N-cyclopropyl-N-{[3-(2-methylpropoxy)phenyl]methyl}prop-2-enamide
N-(1-{imidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)-1-[2-(piperazin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-[(1-cyclopropyl-1H-imidazol-2-yl)methyl]-7-methyl-3,4-dihydro-2H-1,4-benzothiazin-3-one
8-fluoro-2-[({[4-(hydroxymethyl)phenyl]methyl}amino)methyl]quinolin-4-ol
(propan-2-yl)({[4-(pyrimidin-2-yloxy)phenyl]methyl})[(trimethyl-1H-pyrazol-4-yl)methyl]amine
2-(1-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1H-imidazol-2-yl)pyridine
1-(cyclohexylmethyl)-N-[3-(1H-indol-1-yl)propyl]-6-oxopiperidine-3-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-[1-(1,2,5-thiadiazole-3-carbonyl)piperidin-3-yl]propanamide
N3-butyl-N5-cyclooctyl-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
2-(1-benzofuran-2-yl)-4-(3,3,3-trifluoropropyl)pyrimidine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-3-yl]methyl}-N-(2-methoxyethyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-[2-(thiophen-2-yl)acetyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-methyl-N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
{2-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidin-1-yl]-1,3-thiazol-4-yl}methanol
1-[4-({[(4-fluorophenyl)methyl](methyl)amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
1-[(3-chlorophenyl)methyl]-4-(1H-imidazol-2-ylmethyl)piperazine
N-[2-(2-chlorophenyl)-1-[1-(quinolin-6-ylmethyl)piperidin-4-yl]ethyl]-N-methylfuran-2-carboxamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-N-[2-(diethylamino)ethyl]-6-methyl-4-oxo-2-propyl-1,4-dihydropyridine-3-carboxamide
1-{5-methoxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-(1H-1,2,4-triazol-1-yl)butan-1-one
1-cyclopentyl-N-[2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-6-oxopiperidine-3-carboxamide
(3R,5S)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[3-(morpholin-4-yl)propyl]-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
2-{[4-(2,2-dimethyloxan-4-yl)-1H-1,2,3-triazol-1-yl]methyl}pyridine
2-[4-(1H-pyrazol-1-yl)phenyl]-2-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]acetic acid
3-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridin-2-ol
6-methyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1,2-dihydroquinolin-2-one
2-(3-fluorophenyl)-N-({7-[(4-methoxyphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}methyl)acetamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-oxazole-3-carboxamide