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N-ethyl-7,8-dimethyl-N-(pentan-2-yl)-2-(pyrimidin-5-yl)quinoline-4-carboxamide
2-amino-N-[(5-cyclopropyl-1,2-oxazol-3-yl)methyl]-3-ethyl-3H-imidazo[4,5-b]pyridine-6-carboxamide
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridine
3-(3-chlorobenzoyl)-1-{2-methylpyrido[2,3-d]pyrimidin-4-yl}piperidine
methyl 3-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
8-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-1-oxa-8-azaspiro[4.5]decane
2-{[bis(2-hydroxyethyl)amino]methyl}-8-fluoroquinolin-4-ol
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-[(3-methylthiophen-2-yl)methyl]piperidin-4-ol
1,3-dimethyl-6-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-benzyl-N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-1,3-thiazole-4-carboxamide
N'-(3,5-dimethylphenyl)-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]propanediamide
2-(6-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
8-fluoro-N-methyl-N-[3-(oxolan-2-yl)propyl]quinoline-2-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-phenylbenzamide
1-(4-methylphenyl)-4-{3-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]propanoyl}piperazin-2-one
(2R,3S,6R)-5-(2,4-dimethylpyrimidine-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-methoxy-2-methylphenyl)-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]acetic acid
6-(2-aminoethyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}pyrimidin-4-amine
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(3-methoxyphenyl)-5-methyl-4-[3-(piperidin-1-yl)propanoyl]piperazin-2-one
methyl 4-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-4-oxobutanoate
(2S)-6-amino-2-[2-methyl-2-(thiophen-2-ylformamido)propanamido]hexanoic acid
methyl[2-(oxan-4-yl)ethyl]{[4-(trifluoromethyl)phenyl]methyl}amine
2-cyclohexyl-6-[4-(furan-2-carbonyl)-1,4-diazepane-1-carbonyl]-1,3-benzoxazole
6-[(2,4-dichloro-6-methylphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
2-methyl-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-1,3-thiazole-4-carboxamide
5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-{2-[(2-fluoro-5-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(pyridin-2-yl)propan-2-yl]propanamide
4-cyano-N-({1-[(3-hydroxyphenyl)methyl]pyrrolidin-3-yl}methyl)benzamide
N2-[2-(4-methoxyphenyl)phenyl]-N1-(propan-2-yl)pyrrolidine-1,2-dicarboxamide
2-cyclopentyl-8-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
2-[4-(1-benzofuran-2-ylmethyl)-1-[(4-fluorophenyl)methyl]piperazin-2-yl]ethan-1-ol
2-{[(2,3-difluoro-4-methoxyphenyl)methyl]amino}-N-(4-methylphenyl)propanamide
(4S)-3,3,4-trimethyl-1-[2-(1,1,2,2-tetrafluoroethoxy)benzoyl]piperidin-4-ol
2-cyclopropyl-4-methyl-5-[3-(oxan-4-yl)-1H-1,2,4-triazol-5-yl]pyrimidine
2-[4-(3,6-dimethylpyrazin-2-yl)-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
4-ethyl-3-{1-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-3-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(1-methyl-6-oxopiperidin-3-yl)-3-[5-(thiophen-2-yl)-1,3,4-thiadiazol-2-yl]urea
4-(2-{2-[2-(benzyloxy)phenyl]-1H-imidazol-1-yl}ethyl)-4H-1,2,4-triazole
(3R,4R)-4-cyclobutyl-3-methyl-1-(4-methyl-1H-imidazole-2-carbonyl)piperidin-4-ol
methyl 3-(2-methoxyacetamido)-1-[2-(4-methoxyphenyl)ethyl]-5-[(2-methylpropyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-cyclopropyl-5-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidine-1-carbonyl}piperidin-2-one
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-(4-fluorophenyl)cyclopropane-1-carboxamide
3-{[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}-2,2-dimethylpropan-1-ol
1-(2-{7-[(2,3-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)piperidin-2-one
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepane-1-carbonyl}quinoxaline
4-(2-cyclohexyl-1,3-benzoxazole-6-carbonyl)-3,3-dimethylpiperazin-2-one
N-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethyl}cyclohex-3-ene-1-carboxamide
N-[(1S)-1-[1-methyl-3-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]-3-(methylsulfanyl)propyl]acetamide
5-butyl-4-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)-1-(3-methylphenyl)piperazin-2-one