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(1R,5R)-6-methyl-3-[2-methyl-5-(1H-pyrazol-1-yl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
2-{methyl[1-(1,3-thiazol-5-yl)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
N-[(2-chloro-6-fluorophenyl)methyl]-N-cyclopropyl-2,6-dimethylpyridine-4-carboxamide
3,5-difluoro-N-(oxolan-3-yl)benzamide
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
4-[methyl({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl})amino]pyrimidine-5-carboxylic acid
butyl(furan-2-ylmethyl)[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]amine
1-(6-methanesulfonamidopyridin-3-yl)-1H-indazole-3-carboxylic acid
(3S,7S)-5-[2-methyl-2-(morpholin-4-yl)propanoyl]-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
3-(3-chloro-4-methoxyphenyl)-1-{[3-(pyrrolidin-1-ylmethyl)phenyl]methyl}urea
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-{[(2-methyl-1,3-benzothiazol-5-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
(3R)-1-{7-methanesulfonyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}pyrrolidin-3-ol
N-(butan-2-yl)-2-(1,2,3,6-tetrahydropyridin-4-yl)-N-(thiophen-3-ylmethyl)acetamide
N-[5-(diethylamino)pentan-2-yl]-N'-(4-methylphenyl)propanediamide
N-{1-[(3-methylphenyl)methyl]cyclopropyl}-3-(1-methylpiperidin-2-yl)propanamide
ethyl 4-[(3-fluorophenyl)methyl]-1-[(3-hydroxy-4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-{2-methyl-2,7-diazaspiro[4.5]decan-7-yl}-2-(morpholin-4-yl)ethane-1,2-dione
(2H-1,3-benzodioxol-5-ylmethyl)(1-methoxypropan-2-yl){[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amine
N-[2-(diethylamino)ethyl]-1-{2-[(2,4-dimethoxyphenyl)methyl]-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl}-N-methylpiperidine-4-carboxamide
6-[(1R)-2-hydroxy-1-phenylethyl]-2,5-dioxo-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(3S,7S,8aS)-7-{[(3-chloro-1-benzothiophen-2-yl)methyl]amino}-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
2-[ethyl({[(3S,4R)-4-(hydroxymethyl)-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methyl})amino]ethan-1-ol
N-cyclopropyl-1-[2-(4-methoxyphenyl)ethyl]-5-(oxolane-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(3S,4R)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
1-cyclohexyl-N-[(1-propyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
4-{5-cyclobutanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-ylmethyl}-1H-pyrrole-2-carbonitrile
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propanoic acid
8-{2-[4-(dimethylamino)phenyl]acetyl}-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
1-{2-[1-ethyl-3-(phenoxymethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(3-methylbutyl)-1H-pyrazole-4-carboxamide
2-[(3S,4R)-3-cyclopropyl-4-(dimethylamino)pyrrolidin-1-yl]-5,6-dimethylpyridine-3-carbonitrile
4-({3-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}methyl)morpholine
(3R,5R)-5-(morpholine-4-carbonyl)-N-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
[1-(2,1,3-benzoxadiazol-4-ylmethyl)-3-[(4-fluorophenyl)methyl]piperidin-3-yl]methanol
1-(propan-2-yl)-4-[4-(9H-purin-6-yl)piperazine-1-carbonyl]pyrrolidin-2-one
3,3,3-trifluoro-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]propanamide
N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-5-oxo-1-(prop-2-en-1-yl)pyrrolidine-3-carboxamide
5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]-2-(1-methyl-1H-pyrazol-4-yl)pyridine
ethyl 1-(3-acetyl-1H-pyrazole-5-carbonyl)-3-[(4-fluorophenyl)methyl]piperidine-3-carboxylate
(1R,5S)-8-{4-methyl-6H,7H,8H-cyclopenta[g]quinazolin-2-yl}-3,8-diazabicyclo[3.2.1]octane
1-{4-[(3S)-3-ethylmorpholin-4-yl]-4-oxobutyl}pyrrolidin-2-one
6-(4-fluorophenyl)-N-(2-hydroxyethyl)-N-(2-methylpropyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-(furan-2-ylmethyl)-N-(2-methylpropyl)-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
1-{3-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]phenyl}piperazine
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(5-methyl-4H-1,2,4-triazol-3-yl)propanamide
1-(3,5-dimethylphenyl)-4-{[2-(pyrrolidin-1-yl)pyrimidin-5-yl]methyl}piperazin-2-one
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}amine
N-[4-(furan-2-yl)phenyl]-1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidine-3-carboxamide
2-(5-{[(1S,5R)-7-oxo-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-yl)benzonitrile