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ethyl 1-{[2-(difluoromethoxy)phenyl]methyl}-4-[(3-methoxyphenyl)methyl]piperidine-4-carboxylate
N-[4-({[2-(1H-imidazol-4-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-{3-[(5-methylpyridin-2-yl)amino]propyl}-2-(phenylamino)pyrimidine-5-carboxamide
ethyl 3-[(2-methylphenyl)methyl]-1-[2-(2-oxopiperidin-1-yl)acetyl]piperidine-3-carboxylate
3-(4-{imidazo[1,2-b]pyridazin-6-yl}piperazine-1-carbonyl)-4,6-dimethyl-1,2-dihydropyridin-2-one
2-[1-(5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carbonyl)pyrrolidin-2-yl]-1,3-benzothiazole
(3aR,6aR)-2-(cyclobutylmethyl)-5-[4-(propan-2-yl)benzoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(2,5-dimethoxyphenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
(1-{1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-2-ylmethyl)amine
2-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-1-propyl-1H-imidazole
5-[3-(2-methyl-1,3-thiazol-4-yl)-1-[(4-methylphenyl)methyl]-1H-1,2,4-triazol-5-yl]piperidin-2-one
4-[({[3-(prop-2-en-1-yl)-4-(prop-2-en-1-yloxy)phenyl]methyl}amino)methyl]-1,3-thiazol-2-amine
3-{1-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}piperidine
1-({[2-(pyridin-3-yl)ethyl]carbamoyl}methyl)piperidine-4-carboxamide
2-(2,5-dimethoxyphenyl)-N-{[2-(3-hydroxypiperidin-1-yl)-7-methylquinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]acetamide
4-(5-ethyl-1,3-oxazole-4-carbonyl)-2-(6-methoxynaphthalen-2-yl)morpholine
1-[({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]cyclohexan-1-ol
(3R,4R)-1-[(4-methanesulfonylphenyl)methyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
N-methyl-3-(2-methyl-1H-indol-1-yl)-N-(1,2-oxazol-3-ylmethyl)propanamide
4-{[2-(2,5-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-oxazepane
(2R,3R)-3-amino-1'-[1-(methoxymethyl)cyclobutanecarbonyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-[(2-ethoxyphenyl)methyl]-3-[2-(4-methylpiperazin-1-yl)-2-oxoethyl]piperazin-2-one
2-cyclopropyl-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-hydroxypyrimidine-5-carboxamide
N-[4-(1H-1,3-benzodiazol-2-yl)phenyl]-1-[(1-ethyl-1H-pyrazol-4-yl)methyl]piperidine-4-carboxamide
1-(4-cyanopyridin-2-yl)-4-(2-fluorophenoxy)piperidine-4-carboxylic acid
N-benzyl-N-(2-hydroxyethyl)-4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzamide
8-methoxy-N-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-amine
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carbonitrile
2-[5-(furan-3-yl)-4-phenyl-1H-imidazol-1-yl]-3-hydroxypropanoic acid
1-(2,5-dimethylpyrimidin-4-yl)-4-(2-phenylethyl)piperidine-4-carboxylic acid
N-(1-{2,3-dimethyl-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-1-oxopropan-2-yl)methanesulfonamide
1-[2-(dimethylamino)ethyl]-4-(3-propyl-1,2,4-oxadiazol-5-yl)pyrrolidin-2-one
4-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyrimidine
N-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)-3-(1,2,3,6-tetrahydropyridin-1-ylmethyl)benzamide
(2S,4R)-4-amino-1-{2-[(1-ethyl-1H-indol-3-yl)sulfanyl]acetyl}-N-methylpyrrolidine-2-carboxamide
1-[(4-chlorophenyl)methyl]-N-[(4-phenyloxan-4-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2-(propan-2-yloxy)propanamide
4-(4-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
4-(1H-imidazol-1-yl)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
2-[4-(5-methylpyridin-2-yl)-4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenol
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-{3-oxo-2-azaspiro[4.4]nonan-2-yl}acetamide
4-(3-hydroxybenzoyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
5-(2,4-dimethoxypyrimidin-5-yl)thiophene-2-carboxylic acid
2-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-(propan-2-yl)acetamide
3-(4-hydroxyphenyl)-N-[(2-hydroxyphenyl)methyl]-N-methylbenzamide
N-(furan-3-ylmethyl)-3,4-dihydro-2H-1-benzopyran-3-carboxamide
3-{1-[3-(1H-pyrazol-1-ylmethyl)benzoyl]pyrrolidin-2-yl}pyridine
2-{4-[7,8-dimethyl-4-(3-methylpiperidine-1-carbonyl)quinolin-2-yl]-1H-pyrazol-1-yl}ethan-1-ol