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N-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(pyrazin-2-yl)propanamide
N-(1-ethyl-1H-1,2,3-triazol-4-yl)-1-[3-(2-methylpyrimidin-4-yl)phenyl]piperidin-4-amine
2-(2H-indazol-2-yl)-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}-5,6-dimethylpyridine-3-carboxamide
2-{[({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}phenol
2-[(3,4-dimethoxyphenyl)methyl]-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1,3-benzoxazole-6-carboxamide
3-methyl-5-{6-[(pyridin-4-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}pyridin-2-amine
ethyl 4-{7-[3-chloro-5-(trifluoromethyl)pyridin-2-yl]-9-(oxolan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidine-1-carboxylate
N-{[4-(2,3-dihydro-1H-inden-2-yloxy)-3-methoxyphenyl]methyl}-N-(pyridin-4-ylmethyl)cyclohexanecarboxamide
2-[5-(3-{imidazo[1,2-a]pyridin-2-yl}-1,2,4-oxadiazol-5-yl)-1H-pyrazol-3-yl]phenol
N-[(1-hydroxycyclohexyl)methyl]-3-(3-methoxyphenyl)-1H-pyrazole-4-carboxamide
1'-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
1-({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-2-methylpiperidine
N-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-4-yl)ethyl]-5-(propan-2-yl)thiophene-3-carboxamide
3-({[4-(trifluoromethyl)-5,6,7,8-tetrahydroquinazolin-2-yl]amino}methyl)-1λ6-thiolane-1,1-dione
methyl 2-[2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamido]acetate
N-{[5-(furan-2-yl)-1,2-oxazol-3-yl]methyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
8-acetyl-2-[(1-phenyl-1H-pyrazol-4-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)(methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
1,6-dimethyl-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(5S,9aS,9bS)-2-[(5-methylfuran-2-yl)methyl]-5-[3-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
5-(4-chlorophenyl)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methyl-1H-pyrazole-3-carboxamide
3-[(4,4-difluoropiperidin-1-yl)methyl]-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
2-amino-4-[5-(hydroxymethyl)furan-2-yl]-6-methyl-5,6,7,8-tetrahydroquinoline-3-carbonitrile
ethyl 3-[(4-cyclobutaneamidophenyl)formamido]-4,4,4-trifluorobutanoate
N-[(2-chlorophenyl)methyl]-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(3,5-difluoropyridine-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
1-({1-[2-(4-fluorophenyl)azetidine-1-carbonyl]cyclopropyl}methyl)-1H-pyrazole
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
5-[4-(1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-N-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
N,2-dimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,3-benzothiazole-6-carboxamide
2-[(3-methoxyphenyl)methyl]-4-[(4-methyl-1H-imidazol-5-yl)methyl]morpholine
4-(4-methylphenyl)-5-(pyrimidin-5-yl)-N-[1-(1H-1,2,4-triazol-3-yl)ethyl]pyrimidin-2-amine
N-(2-methylpropyl)-5-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}pyridin-2-amine
N,7,8-trimethyl-2-[2-(propan-2-yl)pyrimidin-5-yl]-N-propylquinoline-4-carboxamide
2-(1-propylpiperidin-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N,N-dimethyl-5-{1-[5-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]pyrrolidin-2-yl}thiophene-2-carboxamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methylacetamide
1-[2-(morpholin-4-yl)ethyl]-5-[3-(morpholin-4-ylmethyl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
[(3R,4R)-4-{[(2-methoxyethyl)(methyl)amino]methyl}-1-[4-(propan-2-yl)benzoyl]pyrrolidin-3-yl]methanol
[(2,6-difluorophenyl)methyl](methyl){2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl}amine
4-phenyl-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-one
1-cyclohexyl-N-methyl-N-(quinolin-5-ylmethyl)piperidine-4-carboxamide
ethyl 4-[(3-methoxyphenyl)methyl]-1-(pyridin-3-ylmethyl)piperidine-4-carboxylate
3-[5-(pentan-2-yl)-1,3,4-thiadiazol-2-yl]-1-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}urea
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-ethyl-N-(2-methoxyethyl)piperidine-3-carboxamide
N-(4-chloro-2-fluorophenyl)-2-{[2-(4,6-dimethylpyrimidin-2-yl)ethyl]amino}acetamide
2-phenyl-7-(pyrrolidine-1-sulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
N-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-3-yl]methyl}-1-phenylmethanesulfonamide
4-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-1-(4-methylphenyl)piperazin-2-one