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1-[2-methyl-4-({[3-(propan-2-yl)-4,5-dihydro-1,2-oxazol-5-yl]methyl}amino)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]ethan-1-one
1-[(4-fluorophenyl)methyl]-4-[3-(propan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
2,2-dimethylpropyl N-(1,4-oxazepan-6-ylmethyl)carbamate
4-(2-hydroxy-6-methoxyquinolin-3-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N'-cyclopentyl-N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]butanediamide
N-(2H-1,3-benzodioxol-5-ylmethyl)-N-{[7-chloro-2-(dimethylamino)quinolin-3-yl]methyl}-3-methylthiophene-2-carboxamide
(2S,4S)-N-ethyl-4-{3-[(3-methoxyphenyl)formamido]propanamido}-1-methylpyrrolidine-2-carboxamide
(4-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}oxan-4-yl)methanol
(3aS,6aR)-5-(3-fluoropyridin-2-yl)-3-[3-(morpholin-4-yl)propyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
2-amino-7-[2-(1-methyl-1H-imidazol-2-yl)benzoyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-benzyl-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperazine
4-(2-hydroxypropanoyl)-1-[(3-methylphenyl)methyl]piperazin-2-one
2-[5-(4-chloro-1-ethyl-1H-pyrazol-3-yl)-3-cyclopropyl-1H-1,2,4-triazol-1-yl]pyridine
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[(4-methoxyphenyl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-benzyl-5-[2-(2-methoxyphenyl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
N-[(4-methanesulfonylmorpholin-2-yl)methyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
N-[2-(1H-imidazol-1-yl)ethyl]-4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}benzamide
({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
3-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridazine
1-cyclopropyl-6-oxo-N-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)ethyl]piperidine-3-carboxamide
1-cyclopropyl-N-[3-(1-methyl-1H-1,3-benzodiazol-2-yl)propyl]-5-oxopyrrolidine-3-carboxamide
1-[4-(3,4-dichlorophenyl)piperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-{[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-{1-[(3-ethoxy-4-hydroxyphenyl)methyl]piperidin-4-yl}-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
4-({1-[3-(3-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidin-4-yl}methyl)morpholine
(3S,4S)-1-[(3-phenoxyphenyl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol
4-phenyl-1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}azepane
1-[2-(2,3-dimethylphenoxy)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
(3S,4R)-1-(3-ethyl-1H-indole-2-carbonyl)-4-phenylpyrrolidine-3-carboxylic acid
[(2S,4R,5R)-4-[(benzylamino)methyl]-5-(4-chlorophenyl)-1-ethyl-2-methylpyrrolidin-2-yl]methanol
5-butyl-1-(3-chlorophenyl)-4-(5-methyl-1,3-oxazole-4-carbonyl)piperazin-2-one
4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-N,N-dimethylpiperazine-1-carboxamide
1-[2-(3-fluorophenyl)ethyl]-N-(2-hydroxyethyl)-6-oxo-N-(propan-2-yl)piperidine-3-carboxamide
2-(4-fluorophenoxymethyl)-N-[(2-fluorophenyl)methyl]-1,3-oxazole-4-carboxamide
3-(2,3-dihydro-1H-inden-2-yl)-8-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}pyrrolidin-3-yl)acetamide
7-chloro-1-methyl-N-[3-(3-oxopiperazin-1-yl)propyl]-1H-indole-2-carboxamide
(1S,6R)-9-(2-phenyl-1H-imidazole-4-carbonyl)-3,9-diazabicyclo[4.2.1]nonane
2-ethyl-9-(2,3,6-trifluorobenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1H-pyrrole-2-carboxamide
(2R,3S,6R)-3-phenyl-5-(pyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[4-(pyridin-2-ylmethoxy)phenyl]pyrrolidine-1-carboxamide
1-(2-{[2-(pyridin-3-yloxy)propyl]amino}pyrimidin-4-yl)piperidin-4-ol
N-[(3R,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-2,3-difluorobenzamide
ethyl 1-(1H-indole-5-carbonyl)-4-[(4-methoxyphenyl)methyl]piperidine-4-carboxylate
1-[(3S,4R)-1-(5-chlorothiophene-2-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-4-(cyclopropylmethyl)piperazine
[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl][4-(methylsulfanyl)butan-2-yl]amine
methyl 5-[(3-hydroxy-3-methylbutan-2-yl)amino]-3-(2-methylbutanamido)-1-(oxolan-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1-[4-(propylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one