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3-(4-fluorophenyl)-N-[(3-methyl-1H-pyrazol-5-yl)methyl]-3-phenylpropanamide
2-{4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
2-(1H-pyrazol-1-yl)-1-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]butan-1-one
1-(diethylamino)-3-[2-methoxy-4-({[2-(3-methylpyridin-2-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
3-benzyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-4,5-dihydro-1,2-oxazole-5-carboxamide
(4aS,8aR)-1-(3-hydroxypropyl)-6-[(5-methylthiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1'-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
[(3R,4S)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-{[3-(methylsulfanyl)phenyl]methyl}pyrrolidin-3-yl]methanol
N,1,3-trimethyl-N-(1-{1-[(4-methylphenyl)methyl]piperidin-4-yl}-2-phenylethyl)-1H-pyrazole-5-carboxamide
N-(furan-2-ylmethyl)-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(3-{[3-(3-chlorobenzoyl)piperidin-1-yl]sulfonyl}phenyl)acetamide
2-[(4-chlorophenyl)methyl]-8-(3-fluoropyridin-4-yl)-2,8-diazaspiro[4.5]decan-3-one
3-{[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]amino}-1-(3-methylpiperidin-1-yl)propan-1-one
N2-methyl-N1-[3-(2-methylphenyl)phenyl]pyrrolidine-1,2-dicarboxamide
2-(cyclopropylmethyl)-8-(6-methylpyridazin-3-yl)-2,8-diazaspiro[5.5]undecan-3-one
(1S,3R)-N-[(2-methyl-1,3-thiazol-4-yl)methyl]-3-(2-methylbenzenesulfonamido)cyclopentane-1-carboxamide
(3S,4R)-1-(3-methanesulfonamidopropanoyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
2-{2-[4-(4-methoxybenzoyl)piperazin-1-yl]-2-oxoethyl}-6-methyl-2,3-dihydropyridazin-3-one
1-{2-[3-methyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridin-2-one
2-methyl-5-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidine-1-carbonyl}phenol
N,N-diethyl-1-[3-(4-methylthiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]piperidine-3-carboxamide
N-cyclopentyl-N-(3-phenylprop-2-yn-1-yl)-2-(pyrrolidin-1-yl)acetamide
(4aS,7aR)-1-(2-fluoro-4-methylbenzoyl)-4-(2-methoxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-2-(4-fluorophenyl)imidazo[1,2-a]pyridine
1-[3-(3-methoxyphenoxy)azetidin-1-yl]-4-(4-methylpiperazin-1-yl)pentan-1-one
5-{1-[2-(3-methoxyphenyl)acetyl]piperidin-4-yl}-3-(oxolan-2-ylmethyl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
2-(4-cyclohexylpiperazin-1-yl)-2-(4-fluoro-2-methoxyphenyl)acetic acid
1-[(3R,4S)-3-amino-4-propylpyrrolidin-1-yl]-4-(4-fluorophenyl)butane-1,4-dione
(benzylsulfamoyl)(methyl){[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}amine
1,3-dimethyl-5-[({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)({[5-(methoxymethyl)furan-2-yl]methyl})methylamine
2-ethyl-1-[(2-methoxyphenyl)methyl]-3-[4-(4-methoxyphenyl)piperazine-1-carbonyl]-6-methyl-1,4-dihydropyridin-4-one
(1S,5R)-3-[2-(4-fluorophenoxy)ethyl]-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane
9-(7-chloroquinolin-4-yl)-1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane
(3S,4R)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
8-fluoro-2-{[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}quinolin-4-ol
N-(2-ethoxyphenyl)-3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}propanamide
1-[1-(furan-2-ylmethyl)piperidin-4-yl]-3-(4-phenyl-1,2,3-thiadiazol-5-yl)urea
{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
3-(pyridin-3-yl)-1-[4-(pyrrolidin-1-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]propan-1-one
(4S,4aS,8aS)-1-(2-aminopyridine-4-carbonyl)-4-phenyl-decahydroquinolin-4-ol
5-(1H-indol-3-ylmethyl)-N-(3-methoxypropyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-3-methyl-1-phenyl-1H-pyrazol-5-amine
4-(morpholin-4-yl)-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidin-2-amine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-[(3-methoxyphenyl)amino]butanamide
9-[2-(2-ethyl-1H-imidazol-1-yl)acetyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-(azepan-1-yl)-3-{[2-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-yl]amino}propan-2-ol
ethyl 1-(oxane-4-carbonyl)-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-{[2-(dimethylamino)-5,6,7-trimethoxyquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
{4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}(phenyl)methanol