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1-[(2-phenylpyrimidin-5-yl)methyl]-4-(pyrimidin-2-yl)-1,4-diazepane
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-4-(4H-1,2,4-triazol-4-yl)benzamide
(5-{[1-(1H-indole-3-carbonyl)piperidin-4-yl]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)methanol
1-[3-(dimethylsulfamoyl)propyl]-3-(3-methylbut-2-en-1-yl)piperidine-3-carboxylic acid
1-({benzyl[(1R,2R)-2-hydroxycyclohexyl]carbamoyl}methyl)piperidine-4-carboxamide
5-cyclopropyl-N-[1-methyl-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
4-(2-chlorobenzoyl)-2-(3,4-dichlorophenyl)morpholine
6-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
2-(pyrrolidin-1-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-5,6,7,8-tetrahydroquinazoline-4-carboxamide
7-fluoro-1-methyl-2-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-1,2,3,4-tetrahydroisoquinoline
4-{[ethyl({[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl})amino]methyl}-N-methylbenzene-1-sulfonamide
3-{2-[8-(6-methylpyridazin-3-yl)-1,8-diazaspiro[4.5]decan-1-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(2-methoxyphenoxy)-N,2-dimethyl-N-(2,2,6,6-tetramethylpiperidin-4-yl)propanamide
4-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propanoyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
3-[(4-methylpiperazin-1-yl)sulfonyl]-N-[(5-methylpyrazin-2-yl)methyl]-5-phenylbenzamide
methyl (2S,4S)-4-(5-chloro-3-phenyl-1H-indole-2-amido)-1-(2,3-dihydro-1H-inden-2-yl)pyrrolidine-2-carboxylate
1-(cyclohexylcarbamoyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
{4-[(4-methoxyphenyl)methyl]-1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}methanol
4-(2-methoxy-5-methylbenzoyl)-5-methyl-1-(2-methylphenyl)piperazin-2-one
4-{5-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-1-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}propan-1-one
3-[2-(4-fluorophenyl)ethyl]-1-(1-methyl-1H-imidazole-5-carbonyl)piperidine
3-(2-butyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[(3-methylpyridin-2-yl)methyl]propanamide
2-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}-4-phenylphenol
3-(1H-imidazol-2-yl)-1-(3-phenylbenzoyl)piperidine
{1-[3-(2H-1,3-benzodioxol-5-yl)-2-methylpropyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperidin-4-yl}methanol
5,6-dimethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
4-[(3-cyclohexylpyrrolidin-1-yl)methyl]-1,5-dimethyl-1H-pyrazole
3-(1-methoxybutan-2-yl)-1-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]urea
(1S,5R)-3-{5-methyl-6-[(2-methylpyridin-3-yl)oxy]pyrimidin-4-yl}-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(6-methylpyridine-3-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
1-(4-aminopyrimidin-2-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(2H-1,3-benzodioxol-5-yl)-5-[(2R)-oxolan-2-yl]-3-(2-phenylethyl)-1H-1,2,4-triazole
(4aS,7aR)-1-[5-(propan-2-yl)thiophene-3-carbonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-[(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)methyl]-1-phenyl-1H-1,2,3-triazole
(3R,4R)-1-(4-amino-5-methylpyrimidin-2-yl)-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-3-ol
N-[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]-1-[2-(2-methyl-1,3-benzothiazol-5-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-4-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}butanamide
2-[4-(6-methyl-2-propylpyrimidin-4-yl)piperazin-1-yl]pyridine-3-carbonitrile
1-[3-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]-N-(4-fluorophenyl)piperidin-3-amine
1-methyl-6-(pyridin-4-yl)-N-[2-(pyrrolidin-1-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(3-methylbutyl)-1-(2-methylpropyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(prop-2-en-1-yl)-9-(quinoline-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-ethyl-5-[(2S)-2-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carbonyl]pyrimidin-2-amine
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[2-(1H-pyrrol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
2-chloro-N-methyl-5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]benzamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}benzamide
(1R,3S)-7-(2-fluoro-6-methoxybenzoyl)-3-methoxy-7-azaspiro[3.5]nonan-1-ol
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide