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1-(2-methoxyethyl)-4-{1-[4-(1,3-thiazol-4-yl)phenyl]piperidin-4-yl}piperazine
N-methyl-3-{[3-(3-methylphenyl)propyl]sulfamoyl}-N-propylbenzamide
3-[2-(piperidin-1-yl)ethyl]-5-(piperidin-4-yl)-5-(pyridin-2-yl)imidazolidine-2,4-dione
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]methanesulfonamide
(4aS,7aR)-1-[2-(2-hydroxyphenyl)acetyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[(2-methyl-1,3-oxazol-4-yl)methyl]-2-(2-phenylethyl)piperidine
N-cycloheptyl-4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)piperidine-1-carboxamide
N-[2-(cyclohex-1-en-1-yl)ethyl]-2,4-dimethylpyrimidine-5-carboxamide
3-[2-(4-{[1,2,4]triazolo[4,3-a]pyrimidin-5-yl}piperazin-1-yl)ethyl]-2,3-dihydro-1,3-benzoxazol-2-one
3-({[(2-amino-1,3-thiazol-4-yl)methyl]amino}methyl)-3-hydroxy-1-(2-methoxyethyl)piperidin-2-one
2-methyl-6-{3-[3-(trifluoromethyl)phenoxymethyl]phenyl}-2,3-dihydropyridazin-3-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(pyrrolidine-1-carbonyl)piperidine
(2S)-2-[5-(2-methoxypyrimidin-5-yl)-4-phenyl-1H-imidazol-1-yl]-4-(methylsulfanyl)butan-1-ol
(3S,4S)-1-(5-methoxyfuran-2-carbonyl)-4-propylpyrrolidine-3-carboxylic acid
{1-[(6-methoxy-2H-chromen-3-yl)methyl]piperidin-4-yl}(1-methyl-1H-imidazol-2-yl)methanol
2-cyclopropyl-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-ethyl-5-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
methyl({[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-[(2-methyl-1,3-thiazol-4-yl)methyl]-2-azaspiro[4.5]decan-3-one
{3-ethyl-1-[4-methoxy-3-(prop-2-en-1-yl)benzoyl]piperidin-3-yl}methanol
1-[1-(2-hydroxy-3-methylbenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
N-phenyl-4-[3-(pyridin-4-yl)propanamido]piperidine-1-carboxamide
(2S)-2-{[6-(4-ethylphenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}propanamide
N-[(3S,4R)-1-(1,3-benzoxazol-2-yl)-4-propylpyrrolidin-3-yl]acetamide
2-methyl-N-(3-{4-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]phenoxy}propyl)-1,3-thiazole-4-carboxamide
[(2-cyclohexylpyrimidin-5-yl)methyl][(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]methylamine
4-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-2-(pyrrolidin-1-ylmethyl)-1,4-oxazepane
N-[(2R,3R)-1'-(4-methyl-1H-imidazole-2-carbonyl)-2-(pyridin-3-ylmethoxy)-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]propanamide
1-ethyl-3-(2-methylpropyl)-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1H-pyrazole-5-carboxamide
3-(4-chlorophenyl)-1-(4-methoxypiperidin-1-yl)-3-phenylpropan-1-one
2-(2-methoxyethoxy)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)acetamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
1-(4-cyano-2-fluorophenyl)-3-(pyrrolidin-3-yl)urea
5-chloro-N-[(3-methylphenyl)methyl]-6-oxo-N-(propan-2-yl)-1,6-dihydropyridine-3-carboxamide
2-hydroxy-1-[(1S,5R)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]-1-(4-phenyl-1,3-thiazol-2-yl)piperidine
1-(4-aminopyrimidin-2-yl)-4-(3-fluorophenoxy)piperidine-4-carboxylic acid
N-(furan-2-ylmethyl)-3-{3-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}propanamide
2-{[4-(2,2-dimethylpropyl)-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-5-methoxyphenol
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-3-(1H-indol-3-yl)propan-1-one
3-{1-[5-(1H-1,3-benzodiazol-1-ylmethyl)-1H-pyrazol-3-yl]-N-(propan-2-yl)formamido}propanamide
N-[(7S,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-5-chlorothiophene-2-carboxamide
3-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidin-1-yl}-N-(pyridin-3-yl)propanamide
methyl 7-oxo-9-[2-(piperidin-1-yl)ethoxy]-3-(1,3-thiazole-5-carbonyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
1-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(1-ethyl-1H-1,2,4-triazol-3-yl)urea
N-(3,4-difluorophenyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carboxamide
3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]-N-[1-(2-phenylethyl)piperidin-3-yl]propanamide
4-{4-[2-(morpholin-4-yl)-2-(pyridin-3-yl)acetyl]piperazin-1-yl}benzonitrile
8-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(1-methyl-1H-imidazol-2-yl)methyl]-1-phenylpiperazin-2-one