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3-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]-1H,2H,5H,6H,7H-cyclopenta[b]pyridin-2-one
1-[(4,6-dimethylpyrimidin-2-yl)methyl]-3-[3-methyl-4-(2-oxopyrrolidin-1-yl)phenyl]urea
5-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-2-(3-methylphenyl)pyrimidine
1-methyl-5-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
5-(1,4-dioxane-2-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
N-[2-(3-methoxyphenyl)-1-[1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
5-{1-[2-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-imidazol-2-yl}-2-(furan-2-yl)pyrimidine
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2E)-2-methyl-3-phenylprop-2-en-1-yl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
4-ethyl-5-{3-[2-(2-methylphenyl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
3-(3-chloro-1,2-oxazol-5-yl)-N-[(3-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
[1-(4-{[(3-methoxyphenyl)methyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidin-4-yl]methanol
(5R)-5-[3-(2-phenoxypyridin-3-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-2-one
2-{4-[(2,5-difluorophenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-[2-methyl-3-({[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]amino}methyl)-1H-indol-1-yl]acetamide
2-hydroxy-5-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]benzamide
1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(cyclopropylsulfamoyl)-5-[4-(1H-pyrazol-5-yl)phenyl]benzoic acid
N-[2-(N-methylmethanesulfonamido)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
N-[3-(4-{[(2,3-difluorophenyl)methyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
4-cyclopentyl-N-[3-(2-methoxyethoxy)phenyl]-1,4-diazepane-1-carboxamide
1-(4-benzylpiperazin-1-yl)-3-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-3-yl]propan-1-one
N-[3-(3-{[cyclohexyl(methyl)amino]methyl}phenoxy)propyl]-1-methylpiperidine-4-carboxamide
2-[(3aR,5S,6S,7aS)-5,6-dihydroxy-octahydro-1H-isoindol-2-yl]-N-(3,5-dimethoxyphenyl)acetamide
(2S)-2-amino-1-[4-(2-methylphenoxy)piperidin-1-yl]-2-phenylethan-1-one
4-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
8-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-(cyclohex-1-en-1-yl)-N-({2-[3-(4-methoxybenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)acetamide
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]but-3-enamide
N-(1-cycloheptylpiperidin-3-yl)-2-(phenylsulfanyl)acetamide
(3S,5S,9S)-5-{[(3-methylphenyl)methyl]amino}-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
7-chloro-N-[(6-hydroxypyrimidin-4-yl)methyl]-3,5-dimethyl-1-benzofuran-2-carboxamide
[3-(4-methyl-1,3-thiazol-5-yl)propyl]({[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
1-{1-[(2-chloro-6-fluorophenyl)methyl]piperidin-4-yl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
5-methanesulfonamido-N-[(3S)-2-oxoazepan-3-yl]-1-(2-phenylethyl)-1H-1,3-benzodiazole-7-carboxamide
N-(pyridin-3-ylmethyl)-1-[1-(pyrimidin-2-yl)piperidin-4-yl]piperidine-3-carboxamide
11-[(2,3-dihydro-1H-inden-2-yl)amino]-4-[(2-fluorophenyl)methyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N,6-dimethyl-2-oxo-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-1,2-dihydropyridine-4-carboxamide
11-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-4,6,10,12-tetraazatricyclo[7.3.0.03,7]dodeca-1,3(7),8,10-tetraen-5-one
5-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-1,2,3-benzotriazole
4-{2-[2-(3-methylbut-2-en-1-yl)-3-oxo-2,8-diazaspiro[4.5]decan-8-yl]-2-oxoethyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
2-[(ethylsulfanyl)methyl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-[(2R,3R,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(propan-2-yloxy)ethan-1-one
(2R,3R,6R)-3-(4-methylphenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
{1-[2-(3,4-dimethylphenoxy)ethyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
4-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}quinoline
2-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]ethan-1-ol
1-benzyl-3-methyl-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
9-(3,5-dimethylbenzoyl)-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
1-(2-fluoroethyl)-4-phenyl-5-(2,4,5-trimethoxyphenyl)-1H-imidazole