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(4aR,7aS)-4-(2,4-dimethylbenzoyl)-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1,6-dimethyl-N-[2-(5-phenyl-1,2,4-oxadiazol-3-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[({3-hydroxy-1-[(3-methylphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]-N-methylethane-1-sulfonamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(pyridin-2-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
2-{1-cyclopropyl-2,5-dioxo-3-[3-(trifluoromethyl)phenyl]pyrrolidin-3-yl}-N-methyl-N-(1,3-thiazol-2-ylmethyl)acetamide
methyl 2-{[(1,1-dioxo-1λ6-thiolan-3-yl)(ethyl)amino]methyl}-1,3-oxazole-4-carboxylate
1-(2,5-dimethylfuran-3-carbonyl)-4-[2-(1H-pyrazol-1-yl)ethyl]piperidine
3-(2-benzyl-3-oxopiperazin-1-yl)-N-(2-methylphenyl)-3-oxopropanamide
2-{1-[1-(2,2-diethylcyclopropanecarbonyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
3-{2-[3-(4-chlorophenyl)piperidin-1-yl]ethyl}pyridine
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}piperidin-2-one
N-[(3S,4R)-4-(4-methylphenyl)-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-(3-chloro-4-methylbenzoyl)-1,4-oxazepan-6-ol
(2R,3R)-2-amino-3-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
N-[(2R,3R)-2-methoxy-1'-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-(methylsulfanyl)acetamide
6-methyl-5-{[2-(naphthalen-1-ylmethyl)morpholin-4-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-{4-[(4-hydroxybutyl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
(4aS,8aS)-2-{5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}-decahydroisoquinolin-4a-ol
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-5-ethyl-1,2-oxazole-4-carboxamide
N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-2-methylthieno[2,3-d]pyrimidin-4-amine
2-(2-{4-[(5-methyl-2-phenyl-1H-imidazol-4-yl)methyl]piperazin-1-yl}ethoxy)ethan-1-ol
(2S)-2-[1-(2-fluorophenyl)-3-(5-methylfuran-2-yl)-1H-1,2,4-triazol-5-yl]pyrrolidine-1-carboxamide
2-methyl-9-(5-methyl-1,2-oxazole-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
(2S,4R)-1-[(2,4-dimethoxy-3-methylphenyl)methyl]-N-(2-methyl-1,3-benzothiazol-5-yl)-4-(pyridin-2-ylsulfanyl)pyrrolidine-2-carboxamide
ethyl 3-[(2-fluorophenyl)methyl]-1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidine-3-carboxylate
methyl 2-(N-methyl-2-{3-oxo-1-[(3-phenoxyphenyl)methyl]piperazin-2-yl}acetamido)acetate
1-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-3-[(1-methyl-2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)methyl]urea
2-cyano-N-ethyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)benzamide
1-[(3R,4R)-3-cyclobutyl-3-hydroxy-4-methylpyrrolidin-1-yl]-2-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
methyl 1-[3-(1-benzofuran-2-ylmethyl)-9-methoxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl]piperidine-2-carboxylate
3-{[1-(morpholine-4-sulfonyl)pyrrolidin-3-yl]methyl}benzoic acid
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-2-[2-(pyrrolidin-1-ylmethyl)-4-(thiophen-2-yl)phenoxy]acetamide
2-(1-methyl-1H-imidazol-2-yl)-1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidine
1-[1'-(pyridin-3-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-methyl-4-[2-(thiophen-2-yl)pyrimidine-5-carbonyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
2-{4-[(3,4-difluorophenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}pyridine-3-carbonitrile
methyl 1-(2-methoxyethyl)-5-[(6-methylhept-5-en-2-yl)amino]-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N,2-dimethylthieno[2,3-d]pyrimidin-4-amine
1-[5-({[(4-fluorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
3-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidine-1-carbonyl]-2,6-dimethyl-1,4-dihydropyridin-4-one
3-(3-methoxyphenyl)-1-methyl-3-{2-oxo-2-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]ethyl}pyrrolidine-2,5-dione
(3R,4R)-1-{4H,5H,6H,7H,8H-cyclohepta[b]thiophene-2-carbonyl}-4-(4-methylpiperazin-1-yl)piperidin-3-ol
(2S,4R)-4-amino-N-methyl-N-(quinolin-2-ylmethyl)pyrrolidine-2-carboxamide
7-(cyclobutylmethyl)-2-[1-(4-fluorophenyl)piperidin-4-yl]-2,7-diazaspiro[4.5]decane
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
2-amino-N-[2-(1H-indol-1-yl)ethyl]-N-methyl-4-phenylpyrimidine-5-carboxamide
(2S)-3-hydroxy-2-{[3-(4-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}propanamide
methyl 1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-(2-methylpropyl)-2-oxo-1H,2H,3H-imidazo[4,5-b]pyridine-6-carboxylate