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9-[4-(hydroxymethyl)-1,3-thiazol-2-yl]-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
1-{[3-(2H-1,3-benzodioxol-5-yl)-1H-pyrazol-4-yl]methyl}-4-(furan-2-carbonyl)piperazine
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-5-oxo-2,5-dihydro-1H-pyrazole-3-carboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(4-methyl-1,3-thiazol-2-yl)methyl]amino}methyl)piperidin-2-one
N-[(3S)-1-benzylpyrrolidin-3-yl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)thiophene-2-carboxamide
N-(isoquinolin-5-ylmethyl)-N,1-dimethyl-3-propyl-1H-pyrazole-5-carboxamide
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-[2-(2-oxopyrrolidin-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[3-({[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]amino}methyl)-1H-indol-1-yl]propanamide
2-[1-(3-methylbutyl)-1H-pyrazol-4-yl]-2-[4-(pyrimidin-2-yl)-1,4-diazepan-1-yl]acetic acid
4-[3-(azepane-1-carbonyl)piperidin-1-yl]-2-(oxolan-2-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
3-(5-methyl-1H-1,2,4-triazol-3-yl)-1-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
5-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridin-2-amine
N-(3-hydroxyadamantan-1-yl)-2-[(prop-2-en-1-yl)amino]benzamide
2-hydroxy-N-(2-methoxy-6-methylphenyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
2-(azepan-1-yl)-1-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-{[2-(4-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
2-{1-[(3-methyl-1,2-oxazol-5-yl)methyl]azetidin-3-yl}-1H-1,3-benzodiazole
3-(2-methoxyphenyl)-N-[1-({methyl[2-(oxan-2-yl)ethyl]carbamoyl}methyl)-1H-pyrazol-4-yl]propanamide
N-cyclopropyl-2-[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
N-(propan-2-yl)-1-(1-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}piperidin-4-yl)piperidine-4-carboxamide
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[(3R)-pyrrolidin-3-yl]piperidin-4-amine
N-{imidazo[1,2-a]pyridin-3-ylmethyl}-3-(4-methoxyphenyl)-N-methyl-3-phenylpropanamide
1-[2-(1H-imidazol-2-yl)benzoyl]-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
1-[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
methyl 3-[4-(2-methoxybenzoyl)-2-oxo-6-(pyridin-4-ylmethoxy)-1,4-diazepan-1-yl]propanoate
N-[2-(5-cyclobutyl-1,2,4-oxadiazol-3-yl)ethyl]-4-ethyl-5-methyl-3H-1λ4-pyrimidin-2-amine
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-methyl-2-(2-methylpropanamido)benzamide
4-{[2-(3-methoxyphenyl)ethyl]amino}-5-methyl-N-(pyridin-3-ylmethyl)thieno[2,3-d]pyrimidine-6-carboxamide
5-[1-(2-chloropyridine-4-carbonyl)piperidin-4-yl]-3-[2-(dimethylamino)ethyl]-5-(2-phenylethyl)imidazolidine-2,4-dione
1-[1'-(5-chloro-3-fluoropyridin-2-yl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[9-methoxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-2-ol
5-[5-(2,3-dihydro-1H-inden-1-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl (2S,4S,5R)-5-(2-chlorophenyl)-4-[(2-methoxy-2-oxoethyl)(methyl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylate
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]imidazo[1,2-a]pyrimidine-2-carboxamide
(3aR,6aR)-2-cyclopentyl-5-(3-methylthiophene-2-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[2-(1-{[6-(dimethylamino)pyridin-3-yl]methyl}piperidin-2-yl)ethyl]pyrrolidin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-2-[4-(pyridin-4-ylmethyl)piperazin-1-yl]acetic acid
2-ethyl-9-[4-(1H-1,2,4-triazol-1-yl)butanoyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(6-methyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-4-yl)-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}acetamide
6-methyl-5-(5-methyl-1,2,4-oxadiazol-3-yl)-2-(5-methyl-4,5,6,7-tetrahydro-2H-indazole-3-carbonyl)-1,2,3,4-tetrahydro-2,7-naphthyridine
N-(1-cycloheptylpiperidin-3-yl)-7-methylimidazo[1,2-a]pyridine-2-carboxamide
N,2-dimethyl-N-(pentan-3-yl)-1H-1,3-benzodiazole-5-carboxamide
4-methyl-N-{2-[(trifluoromethyl)sulfanyl]ethyl}pyrimidine-5-carboxamide
2-(pyridin-2-yl)-5-[4-(pyridin-3-yl)piperazine-1-carbonyl]pyrimidin-4-ol
2-(morpholin-3-yl)-N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]acetamide
N-(butan-2-yl)-2-[7-(3-chlorophenyl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]acetamide
(2R)-1-(4-{[(4-methylphenyl)amino]methyl}benzoyl)pyrrolidine-2-carboxamide
N-[2-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]oxolane-2-carboxamide
4-[(1-methyl-1H-pyrazol-4-yl)methyl]-11-({[2-(trifluoromethoxy)phenyl]methyl}amino)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one