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N-cyclopropyl-N-(1-{1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}-2-phenylethyl)furan-2-carboxamide
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-ethyl-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
2-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]phenol
1-(2,1,3-benzothiadiazol-5-ylmethyl)-3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-methylurea
2-(1-methanesulfonylpiperidin-3-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(6-methoxypyridine-3-carbonyl)-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4-chlorophenoxy)ethyl]-N-ethyl-1-(2-hydroxyethyl)-1H-1,3-benzodiazole-5-carboxamide
1-[(2S,4S)-4-amino-1-methylpyrrolidine-2-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
1-cyclopropanecarbonyl-4-[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-1,4-diazepane
4-(4-methoxypyrimidin-2-yl)-N-(2-methyl-1-benzofuran-5-yl)piperazine-1-carboxamide
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methoxyphenyl)ethan-1-one
N-(2-phenyl-5,6,7,8-tetrahydroquinazolin-5-yl)pyridine-3-sulfonamide
3-(1,2-oxazinan-2-yl)-1-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)propan-1-one
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-phenylquinoline-4-carboxamide
2-(3-methyl-1H-pyrazol-1-yl)-1-[2-(3-phenylpropyl)morpholin-4-yl]ethan-1-one
N-[1-(1-cyclopentylpiperidin-4-yl)-1H-pyrazol-5-yl]pyridine-3-carboxamide
8-(2-aminopyridine-4-carbonyl)-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]piperidin-4-ol
N-[(2-chlorophenyl)methyl]-N-(2-hydroxyethyl)-3-(1H-pyrazol-4-yl)propanamide
1-{1-[(5-propylfuran-2-yl)methyl]azetidin-3-yl}piperidine
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-{[3-(trifluoromethyl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
methyl 2-{4-[2-(4-fluorophenyl)ethyl]-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-2-yl}acetate
1-phenoxy-2-[4-(quinolin-8-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]propan-2-ol
(4aS,8aR)-6-(5-fluoropyrimidin-2-yl)-1-(2-phenylethyl)-decahydro-1,6-naphthyridin-2-one
3-(5-amino-1H-1,2,4-triazol-3-yl)-N-[(2-methoxyphenyl)methyl]-N-propylpropanamide
[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl){[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}amine
2-methyl-4-[3-(thiomorpholine-4-carbonyl)phenyl]butan-2-ol
2-({5-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
1-[2-oxo-2-(4-phenyl-1,4-diazepan-1-yl)ethyl]-4-phenylpyrrolidin-2-one
3,3-dimethyl-1-{[5-(3-phenylbutyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}urea
dimethyl({[(1R,5S,6S)-3-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-(1-{[3-(2,3-dihydro-1,4-benzodioxin-6-yl)-1-methyl-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-2-oxo-2-(pyridin-3-yl)acetamide
1-(4-{[5-(hydroxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-3-phenylpropan-1-ol
2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)-N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
6-(5-methoxypyridin-3-yl)-2-methyl-3,4-dihydroquinazolin-4-one
5-cyclopropyl-N-({1-[(2-methylphenyl)methyl]pyrrolidin-3-yl}methyl)-1,3,4-oxadiazol-2-amine
N-[2-(2,2-dimethyl-4-phenyloxan-4-yl)ethyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
ethyl 3-[(2E)-3-phenylprop-2-en-1-yl]-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxylate
2-(1-{1-[2-(dimethylamino)-6-ethylpyrimidin-4-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)propan-2-ol
1-(2-{[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)amino}ethyl)piperidin-2-one
N-{2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]ethyl}-2-(4-oxo-3,4-dihydrophthalazin-1-yl)propanamide
N-cyclopentyl-N-({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)pyridine-2-carboxamide
N-benzyl-5-({methyl[2-(oxan-2-yl)ethyl]amino}methyl)pyrimidin-2-amine
N-cyclopropyl-1-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-5-(quinolin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N,1-dimethyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-1H-indole-2-carboxamide
7-methyl-2-[4-(pyridin-4-yl)piperidine-1-carbonyl]-4H-chromen-4-one
1,3-dimethyl-5-({[4-(trifluoromethyl)pyrimidin-2-yl]amino}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
N-[(3S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide