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N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]morpholine-2-carboxylic acid
N-{[1-(cyclopentylmethyl)piperidin-3-yl]methyl}acetamide
(1S,5R)-6-(2-methyl-1H-pyrrole-3-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
7-[(3-ethoxy-4-methoxyphenyl)methyl]-3-phenyl-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[1-(4-chloro-1-methyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]benzoic acid
4-(4-methanesulfonylphenyl)-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-2-methoxy-N-(oxolan-2-ylmethyl)acetamide
5-ethyl-2-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridine
4-chloro-3-({[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]carbamoyl}amino)-N-methylbenzamide
3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-6-(1-methyl-1H-imidazol-2-yl)pyridazine
6-methyl-2-{3-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-3-carbonitrile
4-methoxy-6-(4-methoxy-2-methylphenyl)pyrimidin-2-amine
6-(benzyloxy)-4-[(1-methyl-1H-indol-3-yl)methyl]-1-(oxan-4-ylmethyl)-1,4-diazepan-2-one
2-(3-{[4-(4-methoxyphenyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyrimidine
6-{8-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
ethyl 3-(2-phenylethyl)-1-[3-(pyrazin-2-yl)propanoyl]piperidine-3-carboxylate
(3aS,7aR)-5-methyl-2-[2-(2-methylphenoxy)acetyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-({1-[(2-methoxyphenyl)methyl]piperidin-4-yl}methyl)-N-(2-methylpropyl)-1H-indole-5-carboxamide
1-{1'-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}-2-methoxyethan-1-one
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-ethylpiperidine-4-carboxamide
N-[1-(1-{[3-(5-methylfuran-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]cyclopropanecarboxamide
(1R,5R)-3-[3-(4-fluorophenyl)benzoyl]-6-methyl-3,6-diazabicyclo[3.2.2]nonane
(1S,4S)-2-(2-methoxy-5-phenylphenyl)-5-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-(2-{[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]amino}ethyl)-1,3-oxazolidin-2-one
N-[(3R,5S)-5-(diethylcarbamoyl)-1-(1H-imidazol-2-ylmethyl)pyrrolidin-3-yl]-3-methyl-1,2-oxazole-5-carboxamide
(2R,6S)-4-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-2,6-dimethylmorpholine
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(dimethyl-1,3-thiazol-5-yl)acetamide
ethyl 4-[3-(4-hydroxyphenyl)benzamido]piperidine-1-carboxylate
N-{[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]methyl}-3-(trimethyl-1H-pyrazol-4-yl)propanamide
1-cyclopentyl-4-(1-ethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-1-methyl-1H-pyrazole-4-carboxamide
3-{[(4-methoxy-2,5-dimethylphenyl)methyl]amino}-N-(4-methoxyphenyl)-5-(methylsulfamoyl)benzamide
[(2,3-difluoro-6-methoxyphenyl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl][(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amine
N-[(3R,4S)-1-(2-methanesulfonylethyl)-4-(propan-2-yl)pyrrolidin-3-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)acetamide
N-ethyl-5-{imidazo[1,2-a]pyridine-2-carbonyl}-1-[(3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-(4-{[2-(cyclohex-3-en-1-yl)-1H-imidazol-1-yl]methyl}-1,3-thiazol-2-yl)pyrimidine
8-(3-chloropyridin-2-yl)-2-[(dimethyl-1,2-oxazol-4-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
(furan-2-ylmethyl)[3-(methylsulfanyl)propyl][2-(morpholin-4-yl)ethyl]amine
N-[(7-{[3-(benzyloxy)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)methyl]pyridine-2-carboxamide
(3S,9aR)-3-(1H-indol-3-ylmethyl)-8-[(5-methylthiophen-2-yl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4,6-dimethoxy-2-{4-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidine
methyl (2S)-1-{9-methoxy-3-[(5-methylfuran-2-yl)methyl]-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carbonyl}pyrrolidine-2-carboxylate
3-(3,5-dimethylphenyl)-N-(1,1-dioxo-1λ6-thian-4-yl)propanamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
(3S,4R)-N,N-dimethyl-1-(2-methyl-1,3-benzothiazole-5-carbonyl)-4-(4-methylphenyl)pyrrolidin-3-amine
1,9-dimethyl-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
(2S,4S)-4-amino-N-ethyl-1-(4-methanesulfonylbenzoyl)pyrrolidine-2-carboxamide
3-{1-[2-(1H-indol-1-yl)ethyl]-1H-imidazol-2-yl}phenol