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(3ar,6ar)-N-{[3-(pyrrolidin-1-yl)phenyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
4-(4-{[3-(methoxymethyl)piperidin-1-yl]methyl}phenyl)-2-methylbutan-2-ol
1,5-dimethyl-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1H-pyrazole-3-carboxamide
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-{1-[(2-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
(3R,4R)-1-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-3-ol
1-[(1-benzylpiperidin-4-yl)methyl]-1-methyl-3-(quinolin-5-yl)urea
(2S,4S)-4-amino-N-ethyl-1-[4-(4-hydroxyphenyl)benzoyl]pyrrolidine-2-carboxamide
4-(dimethylamino)-1-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}butan-1-one
methyl 1-methyl-2-[(1R,2S,9R)-6-oxo-7,11-diazatricyclo[7.3.1.02,7]tridecan-11-yl]-1H-1,3-benzodiazole-5-carboxylate
1-(2,6-diaminopyrimidin-4-yl)-4-(2,3-dihydro-1H-inden-5-yloxy)piperidine-4-carboxylic acid
1-{1-[(4-methoxyphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-3-(2-methylphenyl)pyrrolidin-3-ol
ethyl 2-[4-(5-methylpyridine-3-carbonyl)morpholin-3-yl]acetate
6-{1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-8-yl}-9H-purin-2-amine
4-[3-(2-ethylphenoxy)azetidin-1-yl]piperidine
9-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-3-methyl-3,9-diazaspiro[5.6]dodecane
2-benzyl-8-(oxan-4-yl)-2,8-diazaspiro[4.5]decan-3-one
N-{1-[2-(4-fluorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-3-(5-methyl-1H-pyrazol-1-yl)propanamide
N-[3-hydroxy-2-(thiophen-2-ylmethyl)propyl]-2-methyl-1-benzofuran-5-carboxamide
2-[4-({4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}methyl)piperidin-1-yl]-6-methylpyridine-3-carbonitrile
(2S,4S)-N-ethyl-4-(4-methoxy-3-methylbenzamido)-1-(pent-2-yn-1-yl)pyrrolidine-2-carboxamide
6-methyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[4-(1H-pyrazol-1-yl)phenyl]urea
1-(4-{[(1R,2S,4R)-bicyclo[2.2.1]hept-5-en-2-ylmethyl]amino}-5-methylthieno[2,3-d]pyrimidine-6-carbonyl)piperidine-4-carboxamide
4-hydroxy-N-(2-hydroxyethyl)-2-(4-methylphenyl)-N-(2-methylpropyl)pyrimidine-5-carboxamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[3-(trifluoromethyl)phenyl]methyl}amine
N-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-3-methylbenzamide
4-methoxy-2-[(4-{1-[methyl(pyridin-3-ylmethyl)amino]-2-phenylethyl}piperidin-1-yl)methyl]phenol
1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
1-{1-[2-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]piperidin-4-yl}-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-tert-butyl-6-[2-(trifluoromethyl)benzoyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
N-[furan-2-yl(phenyl)methyl]-3-(2-phenylethyl)-1,2-oxazole-5-carboxamide
(benzylsulfamoyl)({2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl})amine
4-[(1R,5S)-3,8-diazabicyclo[3.2.1]octane-3-carbonyl]-2,6-dimethylquinoline
1-[1-(2-methylpropyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
5-(dimethylamino)-2-[2-(6-methyl-2-phenyl-1,2-diazinan-1-yl)-2-oxoethyl]-2,3-dihydropyridazin-3-one
3-{3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}-4-methylpyridine
4-{2-[cyclopentyl(methyl)amino]acetyl}-1-(2-methoxyphenyl)piperazin-2-one
N,N-dimethyl-2-[5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]pyrimidin-4-amine
5-[1-(3,3-dimethylbutanoyl)piperidin-4-yl]-3-[(4-fluorophenyl)methyl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
5-(4-methoxyphenyl)-3-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]-1,2,4-triazine
1-ethyl-1-[2-(2-methylphenoxy)ethyl]-3-(6-methylpyridin-3-yl)urea
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-[4-(1H-pyrazol-1-yl)butan-2-yl]piperidine
2-(5-tert-butyl-1H-pyrazol-3-yl)-1-[2-(1H-imidazol-1-yl)ethyl]-1H-imidazole
1-[1-(2-cyclohexylethyl)-1H-1,2,3-triazole-4-carbonyl]-4-(2-methoxyethoxy)piperidine
2-amino-4-(2-phenylpyrimidin-5-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-[(3S,5S)-5-(ethylcarbamoyl)-1-(prop-2-en-1-yl)pyrrolidin-3-yl]-1,3-dimethyl-1H-indole-2-carboxamide
ethyl 1-(2-methylpropyl)-5-(1H-pyrazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
7-[(2-fluorophenyl)methyl]-2-(5-methyl-1,3-oxazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
1-(2,3-dihydro-1H-inden-2-ylmethyl)-4-(2-methoxyethyl)piperazine
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(oxan-4-yl)acetamide