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2-[3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)phenyl]-3H,4H,5H,6H,7H,8H,9H-cyclohepta[d]pyrimidin-4-one
3-[1-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
2-methyl-4-[4-(oxan-4-yl)piperazin-1-yl]quinoline
N-(2,4-dimethylphenyl)-2-({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)acetamide
4-(8-methyl-3-{[4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
5-ethyl-N-[(1-methylpyrrolidin-3-yl)methyl]-4-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
(3R,5S)-1-benzyl-N-[(4-fluorophenyl)methyl]-5-{4-[3-(trifluoromethyl)phenyl]piperazine-1-carbonyl}pyrrolidin-3-amine
1-[1'-(1-ethyl-1H-pyrazole-5-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(3-methylphenyl)ethan-1-one
1-(2-ethyl-6-methylphenyl)-4-{5H,6H,7H,8H-imidazo[1,5-a]pyrazine-7-carbonyl}pyrrolidin-2-one
[(8-methoxy-2H-chromen-3-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
(2S)-2-[(1-cyclohexylpiperidin-4-yl)formamido]-3-(4-hydroxyphenyl)propanamide
4-[4-(1-{[2-(1H-pyrazol-1-yl)phenyl]methyl}-1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]piperidine
6-ethoxy-2-[3-(4-methoxypiperidine-1-carbonyl)piperidin-1-yl]-4-methylquinazoline
5-(2,5-dimethylphenoxymethyl)-N-[(2S)-1-hydroxypropan-2-yl]-1,2-oxazole-3-carboxamide
7-fluoro-2-methyl-4-[4-(thiomorpholin-4-yl)piperidine-1-carbonyl]quinoline
N-{1-[1-(3-fluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
3-(butan-2-yl)-5-[(2-fluoro-3-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-N-methyl-5-{[(6-methylpyridin-3-yl)oxy]methyl}-1,2-oxazole-3-carboxamide
({4-cyclopropyl-5-[1-(1-methyl-1H-pyrazole-5-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-(4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl)ethan-1-ol
3-(3,4-difluorophenyl)-5-(2-ethoxybenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
2-[(1-{[2-(2-methylphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-yl)oxy]pyrimidine
(3aS,6aR)-3-[2-(4-fluorophenyl)ethyl]-5-(1H-imidazol-4-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-{3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrimidine
3-(1-{[5-(oxan-2-yl)thiophen-2-yl]methyl}piperidin-4-yl)-1-(pyrrolidin-1-yl)propan-1-one
2-(4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-3-fluoropyridine
2-(5-methylfuran-2-yl)-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazole
{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}(methyl)[1-(pyrazin-2-yl)propan-2-yl]amine
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
4-(3-{[3-(morpholin-4-ylmethyl)piperidin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carbonyl)morpholine
[(3R,4R)-1-(2-methyl-1-benzofuran-7-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
5-(4-{[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]methyl}phenyl)-2H-1,2,3,4-tetrazole
4,5-dimethyl 1-[(3S,5S)-1-(cyclohexylmethyl)-5-[(furan-2-ylmethyl)carbamoyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
1-[(1-ethyl-1H-pyrazol-3-yl)methyl]-4-phenylpyrrolidin-2-one
(2,2-dimethyl-3-{2-[2-(thiophen-2-yl)pyrimidin-5-yl]-1H-imidazol-1-yl}propyl)dimethylamine
[4-({1-[2-methyl-5-(trifluoromethyl)benzoyl]pyrrolidin-3-yl}methyl)phenyl]methanol
1-(oxan-4-yl)-4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperazine
8-[2-hydroxy-3-(2-methylphenoxy)propanoyl]-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(2,1,3-benzoxadiazol-5-ylmethyl)-4-phenoxypiperidine-4-carboxylic acid
4-[(3-methylpiperidin-1-yl)methyl]-N-[1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]benzamide
2-(2,3-dihydro-1H-inden-1-yl)-N-(piperidin-4-ylmethyl)acetamide
4-chloro-N,N-dimethyl-5-{[3-(4-phenylpiperazin-1-yl)piperidin-1-yl]methyl}-1,3-thiazol-2-amine
2-{3-[(4-cyclopentyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-5-methylpyrazine
3-(1-benzofuran-2-yl)-4-{[2-(3-methoxyphenyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
4-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-1-methyl-1H-pyrazole
N-[2-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)quinolin-5-yl]acetamide
N-[(2-methylphenyl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydroquinoline-2-carboxamide
1-benzyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(5-cyclohexyl-1,3,4-oxadiazol-2-yl)-1-[4-(6-methylpyridin-2-yl)piperazin-1-yl]propan-1-one