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2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoxaline
3-[(3R,4S)-3-amino-4-cyclopropylpyrrolidine-1-carbonyl]-6-methyl-1,4-dihydroquinolin-4-one
N-(1-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)cyclopentanecarboxamide
3-(5-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
methyl 2-(5-{1-[2-(pyridin-2-yl)acetyl]piperidin-4-yl}-1H-pyrazol-3-yl)acetate
N-methyl-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-[2-(piperidin-1-yl)ethyl]acetamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
(1S,5R)-6-methyl-3-[1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
(1R,7S)-3-[(4-fluorophenyl)methyl]-6-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2-methyl-N-(propan-2-yl)imidazo[1,2-a]pyrimidine-3-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-methyl-5-[4-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
4-(1H-pyrazol-4-yl)-N-[2-(2,4,6-trimethylphenyl)ethyl]butanamide
2-(3-hydroxypropyl)-9-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-{1-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one
4-({3-hexyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-8-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
1-{5-[(3-methoxyphenyl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}-1,4-diazepan-5-one
1-[cyclohexyl(methyl)amino]-3-[2-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]propan-2-ol
ethyl 1-{3-[(2-hydroxypropyl)carbamoyl]-6-(4-methylthiophen-2-yl)pyridin-2-yl}piperidine-4-carboxylate
2-methyl-8-{1H-pyrazolo[1,5-a]imidazole-7-carbonyl}-octahydro-1H-pyrazino[1,2-a]piperazine
3-{2-[7-(5-chloropyridin-2-yl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}-2,3-dihydro-1H-isoindol-1-one
1-(3-hydroxypropyl)-4-(1-phenylcyclopropanecarbonyl)-1,4-diazepan-6-ol
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetamide
[(3R,4R)-4-[(dimethylamino)methyl]-1-(2-ethoxy-5-methylbenzenesulfonyl)pyrrolidin-3-yl]methanol
N-(1,3-dihydroxy-2-methylpropan-2-yl)-2-{4-[(2-methyl-1,3-oxazol-4-yl)methyl]morpholin-3-yl}acetamide
4-[(1E,3E)-4-(4-chlorophenyl)buta-1,3-dien-1-yl]-1,3-dimethyl-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-({2-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
1-[2-(2H-1,3-benzodioxol-5-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]-N-(2,2-diphenylethyl)piperidine-4-carboxamide
(2S,4S)-1-benzyl-4-(2,5-dimethylfuran-3-amido)-N-ethylpyrrolidine-2-carboxamide
(2S)-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-[2-(thiophen-3-yl)acetyl]pyrrolidine-2-carboxamide
2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-2,8-diazaspiro[4.5]decane
2-{2-cyclopropyl-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}-6-(propan-2-yl)pyridine-3-carbonitrile
2-(benzyloxy)-N-methyl-N-(pyrazin-2-ylmethyl)acetamide
1-methyl-3-(4-phenoxyphenyl)-4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-ylmethyl}-1H-pyrazole
3-{[(1S,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}pyridin-2-amine
N-phenyl-2-{3-phenyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propanamide
3-[3-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenol
(3S,4R)-1-(3-cyclohexyl-1H-pyrazole-4-carbonyl)-4-(hydroxymethyl)piperidin-3-ol
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-(pyrimidin-4-ylmethyl)propanamide
2-(1-{1-[3-methyl-4-(1H-pyrrol-1-yl)benzoyl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)ethan-1-ol
1-(2-ethoxyethyl)-N-[(6-hydroxy-2-methylpyrimidin-4-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-[2-(4-phenyl-1H-imidazol-5-yl)-1H-pyrrol-1-yl]pyrimidine
methyl 3-[(2-methylphenyl)methyl]-7-oxo-9-[3-(pyridin-3-yl)propoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
(1-{5-[(2,3-dihydro-1H-inden-2-yl)amino]-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-yl)methanol
5-(2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethyl)-1,3,4-thiadiazol-2-amine
(3S,4R)-1-[4-(hydroxymethyl)benzoyl]-4-methyl-3-(2-methylpropyl)piperidin-4-ol
4-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2,5-dimethylpyrimidine
1-[(3-hydroxy-2-oxo-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-3-yl)methyl]piperidine-4-carboxamide
1-cyclopentyl-4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazine
ethyl 1-[(2-ethoxy-2-oxoethyl)carbamoyl]-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate