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1-ethyl-N-[2-(4-methoxyphenyl)ethyl]-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(3-chloro-4-fluorophenyl)-8-cyclopropyl-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]-N-methyl-1,3-thiazol-2-amine
3-[2-(3-methoxyphenyl)phenyl]-1-(oxan-3-ylmethyl)urea
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)(pyridin-2-ylmethyl)amine
6-methoxy-2-oxo-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-[(4-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]propanamide
N-(2-{4-[(3,4-dimethylphenyl)methyl]morpholin-2-yl}ethyl)methanesulfonamide
3-(3-fluoro-4-methoxybenzoyl)-1-{[4-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
4-(4-ethoxy-3-methylphenyl)-1-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl}butan-1-one
N-[3-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-4-(2-methylpyrimidin-4-yl)piperidine-1-carboxamide
1-[1-(1-benzylpiperidin-4-yl)piperidine-3-carbonyl]azepane
N-(2-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]carbamoyl}phenyl)-N-methylthiophene-2-carboxamide
2,5-dimethyl-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
8-{[3-(furan-2-yl)phenyl]methyl}-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]piperidine
2-hydroxy-1-[6-hydroxy-4-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-1,4-diazepan-1-yl]ethan-1-one
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-(oxan-4-ylmethyl)propanamide
4-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
3-methoxy-1-{2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}pyrrolidine
{[7-fluoro-2-(thiophen-3-yl)quinolin-3-yl]methyl}[2-(2-methoxyphenyl)ethyl]amine
(2S,4R)-N,N-diethyl-4-(furan-3-amido)-1-methylpyrrolidine-2-carboxamide
1-(4-{[1-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
(2R,3R,6R)-3-(3,5-difluorophenyl)-5-(5-methyl-1,2,4-oxadiazol-3-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-N-propylpyrimidin-2-amine
N2-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-fluoro-N4-methylpyrimidine-2,4-diamine
5-(2-chlorophenyl)-3-(pyridin-2-ylmethyl)-3H,4H-thieno[2,3-d]pyrimidin-4-one
N-benzyl-3-[(1-benzylpiperidin-4-yl)oxy]benzamide
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]pyridin-2-amine
[(3-methyl-1,2-oxazol-5-yl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
N-(1,3-benzoxazol-2-ylmethyl)-4-(piperidin-1-ylmethyl)benzamide
2-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)-N-methylpyrimidin-4-amine
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-6-oxo-1-(pyridin-2-ylmethyl)piperidine-3-carboxamide
5-(3-methyl-1,2,4-oxadiazol-5-yl)-1-(3-phenylpropyl)piperidin-2-one
N-[2-(dimethylamino)-1-phenylethyl]-N-methyl-4-(2-oxopyrrolidin-1-yl)butanamide
4-(4-ethyl-5-methylthiophene-3-carbonyl)-1-(2-methylphenyl)piperazin-2-one
N-ethyl-2-{4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-1-yl}acetamide
3-[1-(3-methylbenzoyl)piperidin-4-yl]-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
2-(2-hydroxyphenoxy)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]acetamide
3-chloro-N-cyclopentyl-4-{[1-(oxan-4-yl)piperidin-4-yl]oxy}benzamide
2-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-1-(piperazin-1-yl)ethan-1-one
1-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}piperazine
N-[2-(1H-imidazol-4-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(cyclopropylmethyl)-8-(1-propyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-(butan-2-yl)-5-(2-methoxyphenoxymethyl)-N-methyl-1H-pyrazole-3-carboxamide
4-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3-phenyl-1H-pyrazole
1-methyl-N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]pyrrolidine-2-carboxamide
(3S,4S)-1-[(6-methoxy-2H-chromen-3-yl)methyl]-4-[4-(pyridin-2-yl)piperazin-1-yl]pyrrolidin-3-ol