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1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
3-(4-fluorophenyl)-6-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}pyridazine
1-benzoyl-N-{2-[methyl(phenyl)amino]propyl}piperidin-4-amine
3-{[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1,2-dihydroquinolin-2-one
6-hydroxy-4-(naphthalen-1-ylmethyl)-1-[3-(2-oxopyrrolidin-1-yl)propyl]-1,4-diazepan-2-one
N-butyl-4-ethanesulfonamido-N-(thiophen-3-ylmethyl)benzamide
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-3-(pyridin-2-yl)propan-1-one
1-[4-(benzenesulfonyl)piperazin-1-yl]-2-(3-methyl-1,2-oxazol-5-yl)ethan-1-one
1-ethyl-3-(oxan-4-yl)-5-(5-phenyl-1,2-oxazol-3-yl)-1H-1,2,4-triazole
1-[(2-fluorophenyl)methyl]-4-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperazin-2-one
N-[2-(4-methyl-1H-1,2,3-triazol-1-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-[4-(2-cyclopentyl-2-phenylacetyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
(2S,4R)-1-[(2,4-difluorophenyl)methyl]-N-(1,1-dioxo-1λ6-thiolan-3-yl)-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
1-{2-[1-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
4-({1-[(2S)-2-aminopropanoyl]piperidin-4-yl}oxy)-N-(2-phenylethyl)benzamide
(1-benzothiophen-2-ylmethyl)(methyl)[(4-{[1-(4-methylbenzoyl)piperidin-4-yl]oxy}phenyl)methyl]amine
N-benzyl-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}pyrimidin-2-amine
methyl[(5-methylfuran-2-yl)methyl]{[2-(propan-2-yl)pyrimidin-4-yl]methyl}amine
(3aR,6aS)-5-[(1,5-dimethyl-3-oxo-2-phenyl-2,3-dihydro-1H-pyrazol-4-yl)methyl]-2-methyl-octahydropyrrolo[3,4-c]pyrrole-1,3-dione
2-methoxy-4-[8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl]pyridine-3-carbonitrile
1-{3-[(1S,3R)-1-(2-aminoethoxy)-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-3-oxopropyl}pyrrolidin-2-one
5-(3-{1-[(4-methyl-1,3-thiazol-5-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1-phenyl-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-2-(3-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-ylmethyl}-1H-indol-1-yl)acetamide
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
1-{2-[2-(4-fluorophenyl)piperidin-1-yl]-2-oxoethyl}azepan-2-one
methyl 3-(1-methylcyclohexanecarbonyl)-7-oxo-9-[2-(2-oxopyrrolidin-1-yl)ethoxy]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
[2-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)ethyl]dimethylamine
3,4-difluoro-N-[(3R,4R)-3-hydroxypiperidin-4-yl]benzamide
N-({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-4-(trifluoromethyl)benzamide
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)benzenesulfonamide
3-{[({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)carbamoyl]methyl}-1,2,3-oxadiazol-3-ium-5-olate
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-1-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]ethan-1-one
6-({4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}methyl)-1,4-oxazepan-6-ol
1'-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]-1,2-dihydrospiro[indole-3,4'-piperidine]
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-(diphenylmethyl)acetamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-6-ethyl-2-methylquinoline-4-carboxamide
(2S,4S)-N-ethyl-1-[(5-methylfuran-2-yl)methyl]-4-[(9H-purin-6-yl)amino]pyrrolidine-2-carboxamide
(4aR,7aS)-1-cyclopropanecarbonyl-4-(pyridine-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-({3-[3-(morpholin-4-yl)azetidine-1-carbonyl]-1H-pyrazol-5-yl}methyl)-1H-1,3-benzodiazole
{1-[(4-chloro-3-fluorophenyl)methyl]-3-[(4-fluorophenyl)methyl]piperidin-3-yl}methanol
N-[2-(5-{[(3-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(pyridin-2-ylsulfanyl)acetamide
3-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)pyridine
N-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]propanamide
N-methyl-1-(piperidin-3-ylmethyl)-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
2-methyl-6-{2-[({2-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]ethyl}pyrimidin-4-ol
N-(3,4-dihydro-2H-1-benzopyran-6-ylmethyl)-1-(methoxymethyl)cyclobutane-1-carboxamide
1-{[2-(3,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
1-(3-{4-[(4-methylphenyl)methyl]-3-oxopiperazin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
ethyl 2-(N-methyl-1-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazol-4-yl}formamido)acetate