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N-tert-butyl-5-chloro-2-{[1-(2,2-dimethylpropyl)piperidin-4-yl]oxy}benzamide
5-({[(5-chlorothiophen-2-yl)methyl]amino}methyl)-N-methyl-N-(2-phenylethyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-methoxy-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide
1-[(5-chlorothiophen-2-yl)methyl]-3-methoxy-1,2-dihydropyridin-2-one
5-(2,5-dimethylphenoxymethyl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1,2-oxazole-3-carboxamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-3-(pyridin-3-yl)propanamide
7-(cyclohexylmethyl)-2-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-6-one
1-[1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidin-3-yl]-4-(4-fluorophenyl)piperazine
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(3-fluoro-4-methoxybenzoyl)piperidine
1-{4-[5-(2,6-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
2,7-dimethyl-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)imidazo[1,2-a]pyridine-3-carboxamide
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(2,5-dimethylthiophen-3-yl)-4-methyl-1H-pyrazol-1-yl]acetamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carboxamide
1-[(1S,5R)-3-cyclobutanecarbonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(pyridin-3-yl)propan-1-one
N-[2-(azepan-1-yl)-2-phenylethyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
4-{[1-(2-aminopyrimidin-4-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
ethyl 4-[3-({[(2-fluorophenyl)methyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
3-[2-({[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}amino)propyl]-3,4-dihydroquinazolin-4-one
2-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
4-[3-(3-chloro-1H-1,2,4-triazol-5-yl)propanoyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
5-(4-chloro-3,5-dimethylphenoxymethyl)-N-methyl-N-(oxan-4-yl)-1,2-oxazole-3-carboxamide
ethyl 1-[(6-methylpyridin-2-yl)methyl]-4-(oxan-2-ylmethyl)piperidine-4-carboxylate
N,N-dimethyl-5-{1-[(5-methylpyrazin-2-yl)methyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
1-methyl-3-(2-methylpropyl)-N-(2-oxo-1,2,3,4-tetrahydroquinolin-4-yl)-1H-pyrazole-5-carboxamide
N-[2-methyl-1-(7-{[3-(2-methylphenyl)phenyl]methyl}-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl)propyl]propanamide
6-[(3-methoxyphenyl)methoxy]-4-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
methyl 3-cyclobutaneamido-5-[(propan-2-yl)amino]-1-[2-(pyridin-2-yl)ethyl]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
2-[(1S,2R)-2-(ethoxycarbonyl)cyclopropyl]-1H-1,3-benzodiazole-6-carboxylic acid
2,2-dimethyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-1-phenylcyclopropane-1-carboxamide
(1S,5R)-3-(2-methyl-1,3-benzoxazole-6-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
1-{2-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[(5-methylpyrazin-2-yl)methyl]urea
N-{[4-(4-aminoquinazolin-6-yl)phenyl]methyl}acetamide
N-[4-({4-[(3-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)phenyl]acetamide
4-[3-(furan-2-yl)-5-[5-(methoxymethyl)thiophen-2-yl]-1H-1,2,4-triazol-1-yl]-1-methylpiperidine
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]({[5-(thiophen-2-yl)-1H-pyrazol-4-yl]methyl})amine
N,2-dimethyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-6-(propan-2-yl)pyrimidin-4-amine
1-[2-(1H-imidazol-1-yl)-1-phenylethyl]-2-(3-methylthiophen-2-yl)-1H-imidazole
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(2E)-3-phenylprop-2-en-1-yl]piperidin-4-yl}oxy)benzamide
N-cyclohexyl-3-{[(4-fluoro-3-methoxyphenyl)carbamoyl]amino}propanamide
1-(2-amino-4-ethyl-1,3-thiazole-5-carbonyl)-4-benzyl-3-ethyl-1,4-diazepan-5-one
(1R,6S)-3-[6-(methoxymethyl)pyrimidin-4-yl]-9-methyl-3,9-diazabicyclo[4.2.1]nonane
2-methyl-8-(3-phenyl-1,2,4-oxadiazol-5-yl)-2,8-diazaspiro[4.5]decan-3-one
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[4-(thian-4-yl)piperazin-1-yl]propan-1-one
1-benzyl-N-{1H-pyrrolo[2,3-b]pyridin-6-yl}pyrrolidin-3-amine
2-(1-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidine-3-carbonyl)pyridine
1-[(4-fluorophenyl)methyl]-2-methyl-3-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-4,5,6,7-tetrahydro-1H-indol-4-one
3-(2-methyl-1H-indol-1-yl)-1-[4-(pyridin-3-ylmethyl)piperazin-1-yl]propan-1-one
2-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-azaspiro[4.5]decan-3-one
{[4-(3-methoxyphenyl)-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)[(2E)-3-phenylprop-2-en-1-yl]amine