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2-benzyl-8-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-2,8-diazaspiro[5.5]undecane
N-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)-3-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]propanamide
N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-(propan-2-yl)-1,3-thiazole-2-carboxamide
(7S,9aR)-7-ethyl-N-(3-fluorophenyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
4-benzyl-5-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
2-(2-methoxyphenyl)-N-[1-(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1H-pyrazol-4-yl]acetamide
2-[4-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)morpholin-3-yl]acetic acid
1-cyclopentyl-6-oxo-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}piperidine-3-carboxamide
2-chloro-6-methoxy-4-{1-[(5-methylfuran-2-yl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenol
N-{2-[({3-[2-hydroxy-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propoxy]phenyl}methyl)amino]ethyl}acetamide
(1R,5R)-3-(2,3-dimethyl-1H-indole-5-carbonyl)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane
(2E)-1-[7-(2-phenylethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-(pyridin-3-yl)prop-2-en-1-one
1,9-dimethyl-4-(4-methylpent-3-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[4-({[3-(dimethylamino)propyl](methyl)amino}methyl)phenyl]-6-(pyridin-4-yl)-3,4-dihydropyrimidin-4-one
ethyl 4-{9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl}piperidine-1-carboxylate
3-[(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)methyl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(4,5-dimethyl-1H-pyrazol-3-yl)propan-1-one
N-benzyl-1-(1-butanoylpiperidin-4-yl)piperidine-3-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
2-(3,4-dimethoxyphenyl)-N-{[5-fluoro-7-(pyrimidin-5-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}acetamide
(3S,4R)-1-(2-ethylpyridine-4-carbonyl)-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
4-{[1-(4-methoxy-2-methylbenzoyl)pyrrolidin-3-yl]methyl}benzoic acid
5-(dimethylamino)-2-{2-oxo-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethyl}-2,3-dihydropyridazin-3-one
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
1-(4-methoxyphenyl)-N-[2-(1H-pyrazol-4-yl)ethyl]cyclopentane-1-carboxamide
(2R,6R)-4-(4-methyl-1,3-thiazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-benzyl-2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-sulfonamide
(3S,4R)-1-{2-[4-(hydroxymethyl)phenyl]acetyl}-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-{1-[2-(4H-1,2,4-triazol-4-yl)pyridine-4-carbonyl]piperidin-4-yl}phenol
(2S,4R)-4-amino-N-ethyl-1-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}pyrrolidine-2-carboxamide
2-({3-[4-(piperidine-1-carbonyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)phenol
4-[4-methyl-6-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-4-(1H-1,2,4-triazol-1-yl)butanamide
4-{[1-(3-methoxypropanoyl)piperidin-4-yl]oxy}-N-[3-(propan-2-yloxy)propyl]benzamide
6-[4-(4-fluorophenyl)-1,4-diazepane-1-carbonyl]-1H-indole
5-(6-aminopyridin-3-yl)-4-(4-methylphenyl)-N-[2-(1H-1,2,3,4-tetrazol-5-yl)ethyl]pyrimidin-2-amine
1-(cyclohexylmethyl)-N-[2-(methylsulfanyl)ethyl]-6-oxopiperidine-3-carboxamide
2-(dimethylamino)-4-methyl-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidine-5-carboxamide
N-[1-(2-chlorophenyl)ethyl]-1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
{[1-(benzenesulfonyl)-1H-pyrrol-2-yl]methyl}(methyl)[1-(pyridin-2-yl)ethyl]amine
1-(4-{[1-(dimethylamino)propan-2-yl]amino}-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
1-{[4-(propan-2-yloxy)phenyl]methyl}-N-[3-(1,3-thiazol-4-yl)phenyl]piperidine-4-carboxamide
(1R,2R)-N-methyl-2-phenyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]cyclopropane-1-carboxamide
(3R,4S)-1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-cyclopropylpyrrolidin-3-amine
6-cyclopentyl-N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-(2-cyclopentylacetyl)-7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-(2,2-diphenylethyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(2R,3S,6R)-5-[1-(methoxymethyl)cyclobutanecarbonyl]-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
4-hydroxy-2-[(4-methyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]quinoline-6-carboxamide